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A Double-blinded, Randomised, Three-period Crossover Euglycaemic Clamp Trial Investigating the Pharmacokinetics, Glucodynamics and Safety of BioChaperone Human Insulin, Human Insulin (Huminsulin® Normal) and Insulin Lispro (Humalog®) in Subjects With Type 1 Diabetes

Phase 1
Completed
Conditions
Diabetes Mellitus Type 1
Interventions
Registration Number
NCT02213146
Lead Sponsor
Adocia
Brief Summary

The addition of BioChaperone to already marketed prandial human insulin preparations may accelerate the onset and shorten the duration of action due to facilitation of the insulin absorption after subcutaneous injection.

The aim of the trial is to assess the efficacy and safety of BioChaperone human insulin in subjects with type 1 diabetes under a dose of 0.2 U/kg.

This trial is a single center, randomised, double-blinded, three treatment, three-period cross-over, 10-hour euglycaemic clamp trial in subject with type 1 diabetes mellitus. Each subject will be randomly allocated to a single dose of BioChaperone human insulin 0.2 U/kg, a single dose of Huminsulin® Normal 0.2 U/kg and a single dose of Humalog® 0.2 U/kg on 3 separate dosing visits.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
38
Inclusion Criteria
  • Male subject with type 1 diabetes for at least 12 months
  • Treated with multiple daily insulin injections or insulin pump (CSII) for at least 12 months
  • Body mass index: 18.5-28.0 kg BW·m-2
  • HbA1c: ≤ 9.0%
Exclusion Criteria
  • Diabetes mellitus type 2
  • Receipt of any investigational product within 3 months prior to first dosing of investigational product in this trial
  • Clinically significant abnormalities as judged by the Investigator
  • Any systemic treatment with drugs known to interfere with glucose metabolism
  • History of alcoholism or drug/chemical abuse as per Investigator's judgement
  • Use of any tobacco or nicotine-contained product within one year prior to screening

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
BioChaperone human insulinBioChaperone human insulinBioChaperone Human Insulin
BioChaperone human insulinHuminsulin® NormalBioChaperone Human Insulin
BioChaperone human insulinHumalog®BioChaperone Human Insulin
Human insulinHuminsulin® NormalHuminsulin® Normal
Human insulinHumalog®Huminsulin® Normal
Insulin lisproBioChaperone human insulinHumalog®
Insulin lisproHuminsulin® NormalHumalog®
Insulin lisproHumalog®Humalog®
Human insulinBioChaperone human insulinHuminsulin® Normal
Primary Outcome Measures
NameTimeMethod
Area under the curve (AUCins(0-1h))1 hour

Area under the human insulin serum concentration - time curve from t=0 to 1 hour

Secondary Outcome Measures
NameTimeMethod
Safety and tolerability: adverse events, local tolerability, vital signs variation, ECG, laboratory safety parametersup to 7 weeks

Adverse events, local tolerability, vital signs variation, ECG, laboratory safety parameters

Pharmacokinetics: Cmax(ins/lisp)up to 10 hours

Maximum observed human insulin / insulin lispro serum concentration

Pharmacokinetics: AUCins/lisp(0-10h): Area under the human insulin / insulin lispro serum concentration10 hours

Area under the human insulin / insulin lispro serum concentration - Time curve from t=0 to 10 hours

Pharmacokinetics: Early t0.5max ins/lispup to 10 hours post administration

Time to first observed half maximum serum human insulin / insulin lispro concentration

Glucodynamics: Area under the glucose infusion rate - time curve from t=0 to 10 hours10 hours

Area under the glucose infusion rate - time curve from t=0 to 10 hours

Glucodynamics: Early t0.5 Glucose Infusion Rate max (GIRmax)10 hours

Time to first observed half maximum glucose infusion rate

Glucodynamics: GIRmax - Maximum glucose infusion rate10 hours

Maximum glucose infusion rate

Pharmacokinetics: Tmax(ins/lisp) - Time to maximum observed serum human insulin concentration and insulin lispro concentration10 hours

Time to maximum observed serum human insulin concentration and insulin lispro concentration

Glucodynamics: Area under the glucose infusion rate - time curve from t=0 to 2 hours2 hours post administration

Area under the glucose infusion rate - time curve from t=0 to 2 hours

Trial Locations

Locations (1)

Profil GmbH

🇩🇪

Neuss, Germany

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