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NAC Supplementation and Skeletal Muscle Performance

Not Applicable
Completed
Conditions
Skeletal Muscle Damage
Skeletal Muscle Performance
Inflammatory Status
Intgracellular Signaling in Skeletal Muscle
Interventions
Dietary Supplement: n-acetylcysteine supplementation
Registration Number
NCT01778309
Lead Sponsor
Democritus University of Thrace
Brief Summary

In this investigation the investigators utilized NAC administration to foster GSH availability during an 8-day period following eccentric exercise-induced muscle damage in order to test our hypotheses: i) antioxidant supplementation does not disturb performance and adaptations induced by exercise-induced muscle injury and ii) redox status perturbations in skeletal muscle are pivotal for the regulation of muscle' inflammatory response and repair.

Detailed Description

The major thiol-disulfide couple of reduced (GSH) and oxidized glutathione (GSSG) is a key-regulator of major transcriptional pathways regulating aseptic inflammation and recovery of skeletal muscle following aseptic injury. Antioxidant supplementation may hamper exercise-induced cellular adaptations.

Our objective was to examine how thiol-based antioxidant supplementation affects skeletal muscle's performance and redox-sensitive signalling during the inflammatory and repair phases associated with exercise-induced micro-trauma.In a double-blind, counterbalanced design, 12 men received placebo (PLA) or N-acetylcysteine (NAC, 20 mg/kg/day) following muscle-damaging exercise (300 eccentric contractions). In each trial, muscle performance was measured at baseline, post-exercise, 2h post-exercise and daily for 8 consecutive days. Muscle biopsies from vastus lateralis and blood samples were collected pre-exercise and 2h, 2d, and 8d post-exercise.

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
20
Inclusion Criteria

a) recreationally trained as evidenced by their maximal oxygen consumption levels (VO2max >45 ml/kg/min), b) were engaged in systematic exercise at least three times/week for ≥12 months), c) non-smokers, d) abstained from any vigorous physical activity during the study, e)abstained from consumption of caffeine, alcohol, performance-enhancing or antioxidant supplements, and medications during the study.

Exclusion Criteria

a) a known NAC intolerance or allergy, b) a recent febrile illness, c) history of muscle lesion, d) lower limb trauma

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
n-acetylcysteine/placebo supplementationn-acetylcysteine supplementationn-acetylcysteine supplementation, orally in three daily dosages, at 20 mg/kg/day, daily for eight days after exercise placebo, orally in three daily dosages, content: 500 mL drink that contained water (375 mL), sugar-free cordial (125 ml), and 2 g of low-calorie glucose/dextrose powder.
Primary Outcome Measures
NameTimeMethod
Change in reduced glutathione in bloodone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise

Concentration of reduced glutathione in red blood cells

Change in reduced glutathione in muscleone hour before exercise, 2 hours post-exercise, 2 days post-exercise, 8 days post-exercise

concentration of reduced glutathione in quadriceps skeletal muscle group

Change in protein carbonyls in red blood cells and serumone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise

concentration of protein carbonyls

Change in protein carbonyls in muscleone hour before exercise, 2 hours post-exercise, 2 days post-exercise, 8 days post-exercise

protein carbonyl concentration in vastus lateralis skeletal muscle

Change in thiobarbituric acid reactive substances in red blood cells and serumone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise

thiobarbituric acid reactive substances concentration in serum and red blood cells

Change in thiobarbituric acid reactive substances in muscleone hour before exercise, 2 hours post-exercise, 2 days post-exercise, 8 days post-exercise

thiobarbituric acid reactive substances concentration in vastus lateralis skeletal muscle

Change in oxidized glutathione in red blood cells and bloodone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise

Concentration of oxidized glutathione in red blood cells and whole blood

Change in total antioxidant capacity in serumone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise
Change in oxidized glutathione in muscleone hour before exercise, 2 hours post-exercise, 2 days post-exercise, 8 days post-exercise

concentration of oxidized glutathione in vastus lateralis skeletal muscle

Change in catalase activity in red blood cells and serumone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise
Change in glutathione peroxidase activity in red blood cellsone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise
Change in creatine kinase activity in plasmaone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise
Change in C-reactive protein in plasmaone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise
Change in macrophage infiltration in muscleone hour before exercise, 2 hours post-exercise, 2 days post-exercise, 8 days post-exercise
Change in white blood cell count in bloodone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise
Change in neutrophil count in bloodone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise
Change in fatty acid binding protein in plasmaone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise
Change in cortisol concentration in bloodone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise
Change in testosterone concentration in plasmaone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise
Change in cytokine concentration in plasmaone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise

Measurement of IL-1β, IL-4, IL-6, TNF-α, IL-8, IL-10, IL-12p70 concentrations in plasma

Change in adhesion molecule concentration in bloodone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise

Measurement of ICAM-1, VCAM-1, sP-selectin, sE-selectin concentrations in plasma

Change in intracellular signalling proteins in muscleone hour before exercise, 2 hours post-exercise, 2 days post-exercise, 8 days post-exercise

Measurement of phosphorylation levels of protein kinase B (Akt), mammalian target of rapamycin (mTOR), serine/threonine kinase (p70S6K), ribosomal protein S6 (rpS6), nuclear factor κB (NFκB), serine⁄threonine mitogen activated protein kinase (p38-MAPK) in vastus lateralis muscle.

Change in myogenic determination factor (MyoD) protein levels in muscleone hour before exercise, 2 hours post-exercise, 2 days post-exercise, 8 days post-exercise

MyoD expression in vastus lateralis muscle

Change in tumor necrosis factor α in muscleone hour before exercise, 2 hours post-exercise, 2 days post-exercise, 8 days post-exercise

Protein levels of TNF-α in vastus lateralis muscle

Secondary Outcome Measures
NameTimeMethod
Change in muscle function of knee extensor and flexor muscleone hour before exercise, 5 minutes post-exercise, 2 hours post-exercise, daily for 8 days post-exercise

assessment of muscle peak and mean torque of knee extensors and flexors on an isokinetic dynamometer at 0, 90 and 180 degrees/sec

Body compositionOne day before exercise

Assessment of percent (%) lean body mass.

Maximal aerobic capacityOne day before exercise

Assessment of maximal oxygen consumption, an indice of cardiovascular conditioning

Change in profile of dietary intakeone hour before exercise, daily for 8 days post-exercise

Assessment of dietary intake with emphasis on antioxidant element intake

Change in side effect occurenceone hour before exercise, daily for 8 days post-exercise

The prevalence of potential side-effects (such as headaches or abdominal pain or any other discomfort) was monitored using a subjective 0-10 side-effects scale on a daily bases by an unblinded investigator (for ethical reasons).

Trial Locations

Locations (1)

Laboratory of Physical Education & Sport Performance

🇬🇷

Komotini, Thrace, Greece

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