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BI836845 Plus Enzalutamide in Castrate Resistant Prostate Cancer (CRPC)

Phase 1
Completed
Conditions
Prostatic Neoplasms, Castration-Resistant
Interventions
Registration Number
NCT02204072
Lead Sponsor
Boehringer Ingelheim
Brief Summary

The overall aim of the trial is to investigate the safety and anti-tumour activity of an experimental drug BI 836845 taken together with the prostate cancer drug, enzalutamide, compared to enzalutamide given alone, in castrate resistant prostate cancer (CRPC) patients that have previously been treated and failed on docetaxel and abiraterone treatments. Initially, a tolerability and safety phase (phase Ib escalation) will be performed to confirm the maximum tolerated dose (MTD), or recommended doses of both BI 836845 and enzalutamide that can be taken together.

Once the MTD, or recommended phase II dose, have been determined an expansion cohort will also be explored (phase Ib expansion) in CRPC patients already taking enzalutamide and have a rise in prostate serum antigen (PSA) levels. Patients may not have received prior docetaxel or abiraterone. Patients in this cohort will receive the MTD, or recommended phase II dose, of BI 836845 and enzalutamide determined in the phase Ib escalation phase.

The randomised trial (phase II) will be an open label, parallel group study design in a 1:1 ratio to which patients will receive either BI 836845 plus enzalutamide (Arm A) at the MTD/recommended doses, or enzalutamide alone (Arm B).

In all parts of the trial safety, anti-tumour activity will be assessed, in addition to circulating tumour cells (CTC), prostate serum antigen (PSA) response and progression, and determination of Overall Survival (OS).

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
120
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
BI 836845 & EnzalutamideBI 836845-
EnzalutamideEnzalutamide-
BI 836845 & EnzalutamideEnzalutamide-
Primary Outcome Measures
NameTimeMethod
Prostate Surface Antigen (PSA) response - defined as a decline in PSA value >50% (which is confirmed by a second value 3 to 4 weeks apart) (phase Ib expansion)Up to 3 years
Maximum tolerated dose (phase Ib escalation)6 months
Number of patients with dose limiting toxicities (phase Ib escalation)6 months
Radiological Progression free survival - time from randomisation to disease progression based on investigator assessment in bone, or soft tissue, or death (phase II)Up to 3 years
Secondary Outcome Measures
NameTimeMethod
Maximum decline in PSA - compared to baseline that occurs at any point after treatment start (phase II)Up to 3 years
Overall survival - defined as the time from randomisation to death from any cause (phase II)Up to 3 years
PSA response - defined as a decline in PSA value >50%, which is confirmed by a second value 3 to 4 weeks apart (phase II)Up to 3 years
Time to prostate serum antigen (PSA) progression - defined as the date that a 25% or greater increase in PSA, and an absolute increase of 2 ng/mL or more from the nadir, is documented, which is confirmed by a second value 3 or more weeks later (phase II)Up to 3 years
Percentage change in PSA - from baseline to week 12 of treatment (phase II)Up to 3 years
CTC response-CTC reduction compared to baseline for at least one time point after treatment start assessed by maximum change in CTC counts compared to baseline that occurs at any point after treatment start (phase II)Up to 3 years
Changes in circulating tumour cells (CTC) response - CTC reduction compared to baseline for at least one time point after treatment defined as CTC decline from, equal to, or more than, 5 to <5 cells per 7.5ml blood (phase Ib expansion)Up to 3 years
Changes in CTC response - CTC reduction compared to baseline for at least one time point after treatment start assessed by CTC decline from, equal to, or more than, 5 to <5 cells per 7.5ml blood (phase II)Up to 3 years
Radiological progression free survival - defined as time from start of treatment to disease progression based on investigator assessment in bone based on PCWG2 or soft tissue based on modified RECIST 1.1 where applicable, or death (phase Ib expansion)Up to 3 years
Radiological progression free survival - defined as time from randomisation to disease progression based on central review in bone based on PCWG2 or soft tissue based on modified RECIST 1.1 where applicable, or death (phase II)Up to 3 years

Trial Locations

Locations (27)

Hospital Duran i Reynals

🇪🇸

L'Hospitalet de Llobregat, Spain

Hospital Ramón y Cajal

🇪🇸

Madrid, Spain

The Clatterbridge Cancer Centre

🇬🇧

Bebington, Wirral, United Kingdom

Velindre Cancer Centre

🇬🇧

Cardiff, United Kingdom

NewYork-Presbyterian/Weill Cornell Medical Center

🇺🇸

New York, New York, United States

Hospital Vall d'Hebron

🇪🇸

Barcelona, Spain

Samsung Medical Center

🇰🇷

Seoul, Korea, Republic of

Hospital General Universitario Gregorio Marañón

🇪🇸

Madrid, Spain

The Christie Hospital

🇬🇧

Manchester, United Kingdom

Churchill Hospital

🇬🇧

Oxford, United Kingdom

The Royal Marsden Hospital, Sutton

🇬🇧

Sutton, United Kingdom

Instituto Valenciano de Oncología

🇪🇸

Valencia, Spain

Karmanos Cancer Institute

🇺🇸

Detroit, Michigan, United States

Oregon Health and Sciences University

🇺🇸

Portland, Oregon, United States

Asan Medical Center

🇰🇷

Seoul, Korea, Republic of

Hospital Clínic de Barcelona

🇪🇸

Barcelona, Spain

Hospital Santa Creu i Sant Pau

🇪🇸

Barcelona, Spain

Taipei Veterans General Hospital

🇨🇳

Taipei, Taiwan

National Cancer Centre Singapore

🇸🇬

Singapore, Singapore

Taichung Veterans General Hospital

🇨🇳

Taichung, Taiwan

Erasmus MC - Daniel den Hoed

🇳🇱

Rotterdam, Netherlands

National Taiwan University Hospital

🇨🇳

Taipei, Taiwan

Tweesteden Ziekenhuis, locatie Tilburg

🇳🇱

Tilburg, Netherlands

OncoCare Cancer Centre

🇸🇬

Singapore, Singapore

Tan Tock Seng Hospital

🇸🇬

Singapore, Singapore

Prince of Wales Hospital

🇭🇰

Hong Kong, Hong Kong

Queen Mary Hospital

🇭🇰

Hong Kong, Hong Kong

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