MedPath

Imaging Neural Correlates of Ketamine Using PET/MR

Phase 1
Recruiting
Conditions
Major Depressive Disorder
Interventions
Registration Number
NCT04587778
Lead Sponsor
Medical University of Vienna
Brief Summary

The purpose of this randomized, placebo-controlled study is to investigate pharmacodynamic differences between racemic ketamine and esketamine using functional fluorodeoxyglucose (\[18F\]FDG) positron emission tomography/magnetic resonance imaging (PET/MR)

Pilot study I:

A pilot study with healthy controls will be performed in order to investigate pharmacokinetic behavior and acute behavioral effects of intravenous ketamine infusion.

Pilot study II:

A pilot study including 15 healthy volunteers will be performed in order to optimize scanning procedures. The pilot study follows a randomized, placebo-controlled, double-blind, cross-over study design. After enrollment into the study all subjects will undergo two \[18F\]FDG PET/CT scans in the course of which they will receive either S-ketamine or placebo during the first scan and the respective other study medication during the second scan.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
65
Inclusion Criteria
  • General health based on medical history, physical examination and structured clinical interview for the Diagnostic and Statistical Manual of Mental Disorders (DSM-IV) (SCID)
  • Age 18 to 55 years
  • Right-handedness (due to potential lateralization effects of lefthanded subjects)
  • Willingness and competence to sign the informed consent form.
Exclusion Criteria
  • Current or history of psychiatric or neurological disease
  • Current medical illness requiring treatment
  • Pregnancy or current breastfeeding
  • Current or former substance abuse
  • Diagnosis of an Axis-1 psychotic disorder in a first-degree relative
  • Any contraindication for MRI (e.g., MR incompatible implants, etc.) including dental implants causing signal artifacts
  • For subjects participating in earlier studies using ionizing radiation, the total radiation exposure of 30 millisievert (mSv) over the last 10 years must not be exceeded, as specified in the Austrian legislation on radiation protection (www.ris.bka.gv.at). Accordingly, body weight >100kg is an exclusion criterion (5.1 Megabequerel (MBq)/kg * 100kg * 0.019 mSv/MBq* 0.885 = 8.58 mSv per scan, the factor 0.885 is considered due to continuous radioligand infusion, see PET scanning).
  • Failure to comply with the study protocol or to follow the instruction of the investigating team.

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Esketamine ((S)-Ketamine)PlaceboSingle-blind placebo (saline) infusion will be performed during the first PET/MR scan in all subjects, i.e. both arms. In a cross-over study design, esketamine will be administered during the second scan and racemic ketamine during the third scan.
Racemic ketamine ((R,S)-Ketamine)PlaceboSingle-blind placebo (saline) infusion will be performed during the first PET/MR scan in all subjects, i.e. both arms. In a cross-over study design, racemic ketamine will be administered during the second scan and esketamine during the third scan.
Esketamine ((S)-Ketamine)Ketamine HydrochlorideSingle-blind placebo (saline) infusion will be performed during the first PET/MR scan in all subjects, i.e. both arms. In a cross-over study design, esketamine will be administered during the second scan and racemic ketamine during the third scan.
Racemic ketamine ((R,S)-Ketamine)EsketamineSingle-blind placebo (saline) infusion will be performed during the first PET/MR scan in all subjects, i.e. both arms. In a cross-over study design, racemic ketamine will be administered during the second scan and esketamine during the third scan.
Esketamine ((S)-Ketamine)EsketamineSingle-blind placebo (saline) infusion will be performed during the first PET/MR scan in all subjects, i.e. both arms. In a cross-over study design, esketamine will be administered during the second scan and racemic ketamine during the third scan.
Racemic ketamine ((R,S)-Ketamine)Ketamine HydrochlorideSingle-blind placebo (saline) infusion will be performed during the first PET/MR scan in all subjects, i.e. both arms. In a cross-over study design, racemic ketamine will be administered during the second scan and esketamine during the third scan.
Primary Outcome Measures
NameTimeMethod
Change in cerebral blood flow (CBF)during PETMR/during 45 minutes of infusion

Change in CMRGlu between each PET/MR scan

Change in Cerebral metabolic rate of glucose (CMRGlu)during PETMR/during 45 minutes of infusion

Change in CMRGlu between each PET/MR scan

Secondary Outcome Measures
NameTimeMethod
Change in Positive and Negative Syndrome Scaleone hour after infusion to baseline

Minimum: 30, Maximum: 210; higher score indicates worse outcome

Change in Brief Psychiatric Rating Scaleone hour after infusion to baseline

Minimum: 18, Maximum: 126; higher score indicates worse outcome

Change in Clinician Administered Dissociative States Scaleone hour after infusion to baseline

Minimum: 0, Maximum: 92; higher score indicates worse outcome

Trial Locations

Locations (1)

Medical University of Vienna

🇦🇹

Vienna, Austria

© Copyright 2025. All Rights Reserved by MedPath