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A Study of the Safety and Tolerability of ASP0777 in Subjects With Alzheimer's Disease (AD) Taking a Stable Dose of Donepezil

Phase 1
Completed
Conditions
Alzheimer's Disease
Interventions
Drug: Placebo
Registration Number
NCT01406145
Lead Sponsor
Astellas Pharma Inc
Brief Summary

This study is intended to determine the safety and tolerability of ASP0777 in subjects with Alzheimer's Disease (AD) taking a stable dose of donepezil.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
60
Inclusion Criteria
  • Subject has a Mini-Mental Status Exam score of 18-26
  • Subject has a diagnosis of "probable" Alzheimer's Disease
  • Subject has used donepezil for at least 3 months and has been on a stable dose for at least 6 weeks prior to screening
  • Subject has a reliable adult who is residing with him/her during the outpatient portion of the study
  • Subject is medically stable
  • Subject has adequate cognitive, hearing, vision, and language skills
  • Subject is able to ingest oral tablets
Exclusion Criteria
  • Subject has received any investigational product in another clinical study or post-marketing clinical study within past 3 months
  • Subject has any clinically significant abnormal laboratory tests
  • Subject is a female who is pregnant, lactating or of childbearing potential who refuses to use a form of contraception during the study
  • Subject has a history of a drug allergy or intolerance to memantine or a related compound
  • Subject is currently using anti-dementia drugs (except for donepezil) or has used any such drugs within the last 4 weeks
  • Subject has a score of 2 on item 16 of Cornell Scale for Depression in Dementia (CSDD) or has an overall CSDD score > 10
  • Subject is using off-label medicines, non-medicinal compounds, or dietary aids/food supplements to improve cognition that have not been at a stable dose for at least 4 weeks prior to Screening and/or are anticipated to change dosing regimen during the study
  • Subject has a history of drug or alcohol abuse within the past 12 months or subject consumes > 1 drink of alcohol daily, or is unable to refrain from alcohol during the study
  • Subject is a current smoker or recently quit smoking (within the past 12 months)
  • Subject has a clinically significant medical condition that is unstable or is likely to become unstable during the course of the study
  • Subject has history of seizures, other than febrile seizures during infancy
  • Subject has history of repeated falls within past 6 months
  • Subject has a major psychiatric illness or has received treatment for symptoms of a major psychiatric illness within past 1 year. Mild psychiatric disorders are allowable

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
ASP0777 low dose, then high doseASP0777ASP0777 low dose for 1 week and ASP0777 high dose for 5 weeks
ASP0777 low doseASP0777ASP0777 low dose for 6 weeks
ASP0777 high doseASP0777ASP0777 high dose for 6 weeks
PlaceboPlaceboPlacebo for 6 weeks
Primary Outcome Measures
NameTimeMethod
Number and percentage of subjects with adverse eventsUp to 56 Days
Secondary Outcome Measures
NameTimeMethod
Pharmacokinetic assessment of AUC, maximum concentration (Cmax), minimum concentration (Cmin) and time to maximum concentration (tmax) through analysis of blood samplesUp to 56 Days

Trial Locations

Locations (2)

MD Clinical

🇺🇸

Hallandale Beach, Florida, United States

Pacific Research Network, Inc.

🇺🇸

San Diego, California, United States

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