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The Effect of Metformin on Composition of Human Gut Bacteria

Phase 1
Completed
Conditions
Healthy
Interventions
Registration Number
NCT02546050
Lead Sponsor
Oluf Borbye Pedersen
Brief Summary

OBJECTIVE: Investigate structural changes in the human gut microbiota and associated changes in metabolic markers in urine, saliva, blood and fecal samples following metformin treatment.

DESIGN: An, 18 week, one-armed cross over intervention trial consisting of a 6-week pre-intervention period, 6-week intervention period and a 6-week post-intervention period. 25 healthy young men will be included in the trial.

INTERVENTION: Six-week Metformin treatment to young healthy men.

Detailed Description

An, 18 weeks, one-armed cross over intervention trial consisting of a 6-weeks pre-intervention period, 6-weeks intervention period and a 6-weeks post-intervention period. 25 healthy young men will be included in the trial. The pre-intervention period is the control period with no treatment. During the intervention period participants will receive 500 mg of metformin once daily the 1st week, then 500 mg twice daily the 2nd week, 1000 mg + 500 mg daily the 3rd week and 1000 mg + 1000 mg daily the remaining three weeks. Post-interventional investigators will examine gut microbiota of the participants 6 weeks after completion of the intervention period.

MESUREMENTS: Altered composition of gut microbiota as investigated by 16S rRNA sequencing is the primary outcome of this study. Secondary outcomes are to investigate changes in metabolic and inflammatory markers in blood and fecal samples. Blood, urine, saliva and fecal samples will be stored for future studies.

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
26
Inclusion Criteria
  • Male
  • HbA1c < 5.7 % (39 mmol/mol)
  • Caucasian (self-report of parental ethnicity)
  • Weight stabile with 18.5 kg/m2 < BMI < 27.0 kg/m2
  • Normal kidney function as evaluated by normal p-creatinine for age
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Exclusion Criteria
  • Oral intake of any form of prescribed medication two months prior to recruitment
  • Chronic or acute illness
  • Previous gastro-intestinal operation excluding appendicitis
  • Any other significant medical reason for exclusion as determined by the investigator
  • Unable to give informed consent
  • Need of medical treatment during the study period
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Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
MetforminMetformin18 weeks study with intervention during week 6 to 12: the intervention consist of 500 mg of metformin once daily for week 7, then 500 mg twice daily week 8, 1000 mg + 500 mg daily week 9 and 1000 mg + 1000 mg daily for weeks 10-12.
Primary Outcome Measures
NameTimeMethod
Structural changes in the human gut microbiota.Baseline, 4 , 7, 8, 10, 11 , 13, 16, and 18 weeks

Fecal samples are collected in order to characterize the gut microbiota composition.

Microbial DNA will be subjected to sequencing, microbial gene analyses, including taxonomic and functional annotation.

Secondary Outcome Measures
NameTimeMethod
Changes in insulin metabolismBaseline and at week 7,10,13 and 18

Venous blood will be collected. The samples will be analyzed for serum insulin and C-peptide levels. Changes will be correlated to changes in gut microbiota composition.

Changes in inflammatory markers in blood samples.Baseline and at week 7,10,13 and 18

Venous blood will be collected. The samples will be analyzed for markers of inflammation such as high sensitive C-reactive protein.

Changes in plasma glucose and HbA1c levelsBaseline and at week 7,10,13 and 18

Venous blood will be collected. The samples will be analyzed for plasma glucose and HbA1c, and correlated to changes in gut microbiota composition

Changes in kidney function tests.Baseline and at week 7,10,13 and 18

Venous blood will be collected. The samples will be analyzed for plasma creatinine and correlated to gut microbiota changes

Bio-electrical impedance.Baseline and at week 7,13 and 18

Body composition will be measured through bio-electrical impedance

GI symptomsBaseline and at week 7, 10, 13 and 18.

Changes in gastrointestinal symptoms of participants by validated VAS-questionnaire concerning following parameters: Overall abdominal symptoms, abdominal pain, bloating, flatulence, satisfaction with stool consistence, constipation, diarrhea, tiredness, nausea, metallic taste.

Changes in liver function tests.Baseline and at week 7,10,13 and 18

Venous blood will be collected. The samples will be analyzed for liver function test and correlated to gut microbiota changes

Serum CobalaminBaseline and at week 7,10,13 and 18

Venous blood will be collected. The samples will be analyzed for serum cobalamin and correlated to gut microbiota changes

Metformin plasma levelAt week 10 and 13.

Plasma levels of metformin will be measured at visits 3 and 4 in order to test for compliance. Plasma metformin concentrations will be correlated to changes in gut microbiota composition and function

Blood pressureBaseline and at week 7,13 and 18

Systolic and diastolic blood pressure are measured in the inclined position after a five minute rest using an automated sphygmomanometer. The measurement is repeated three times. Participants are instructed not to talk during the measurements.

Heart rateBaseline and at week 7,13 and 18

Heart rate is measured in the inclined position after a five minute rest using an automated sphygmomanometer. The measurement is repeated three times. Participants are instructed not to talk during the measurements.

Anthropometrics characteristicsBaseline and at week 7,13 and 18

Waist- and hip circumference are measured using standardized procedures.

Trial Locations

Locations (1)

The Novo Nordisk Foundation Center of Basic Metabolic Research, Section for Metabolic Genetics, University of Copenhagen

🇩🇰

Copenhagen, Copenhagen Ø, Denmark

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