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Efficacy and Safety of Alpha1-Proteinase Inhibitor (Human), Modified Process (Alpha-1 MP) in Subjects With Pulmonary Emphysema Due to Alpha1 Antitrypsin Deficiency (AATD)

Phase 3
Active, not recruiting
Conditions
Pulmonary Emphysema in Alpha-1 PI Deficiency
Interventions
Other: 0.9% Sodium Chloride for Injection, USP
Biological: Alpha-1 MP
Registration Number
NCT01983241
Lead Sponsor
Grifols Therapeutics LLC
Brief Summary

This is a multi-center, randomized, placebo-controlled, double blind clinical study to assess the efficacy and safety of two separate dose regimens of Alpha-1 MP versus placebo for 156 weeks (i.e., 3 years) using computed tomography (CT) of the lungs as the main measure of efficacy. The two Alpha-1 MP doses to be tested are 60 mg/kg and 120 mg/kg administered weekly by IV infusion for 156 weeks. The study consists of an optional pre-screening phase, Screening Phase, a 156-week Treatment Phase, and an End of Study Visit at Week 160.

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
345
Inclusion Criteria
  • Have a documented total alpha1-PI serum level < 11 µM.
  • Have a diagnosis of congenital AATD with an allelic combination of ZZ, SZ, Z(null), (null)(null), S(null), or "at-risk" alleles.
  • At the Screening (Week -3) Visit, have a post-bronchodilator forced expiratory volume in 1 second (FEV1) ≥ 30% and < 80% of predicted and FEV1/forced vital capacity (FVC) < 70% (Global Initiative for Chronic Obstructive Lung Disease [GOLD] stage II or III).
  • Have a carbon monoxide diffusing capacity (DLCO) ≤ 60% of predicted (corrected for HgB) within the past 2 years OR evidence of pulmonary emphysema on CT scan within the past 2 years per the Investigator's judgment.
  • Have clinical evidence of pulmonary emphysema per the Investigator's judgment.
Exclusion Criteria
  • Has received alpha1-PI augmentation therapy for more than 1 month within the six months prior to the Screening Visit.
  • Has received alpha1-PI augmentation therapy within one month of the Screening Visit.
  • Has had a chronic obstructive pulmonary disease (COPD) exacerbation within the 5 weeks prior to the Screening Visit or during the Screening Phase.
  • Unable to physically (e.g., unable to fit inside the CT scanner) or mentally (e.g., claustrophobic) undergo a CT scan.
  • History of lung or liver transplant.
  • Any lung surgery during the past 2 years (excluding lung biopsy).
  • On the waiting list for lung surgery, including lung transplant.
  • Smoking during the past 12 months or a positive urine cotinine test at screening that is due to smoking. Maybe on Nicotine replacement, including vapor cigarettes.
  • History of anaphylaxis or severe systemic response to any plasma-derived alpha1-PI preparation or other blood product(s).
  • Use of systemic steroids above a stable dose equivalent to 5 mg/day prednisone (i.e., 10 mg every 2 days) within the 5 weeks prior to the Screening Visit (inhaled steroids are not considered systemic steroids) or during the Screening Phase.
  • Use of systemic or aerosolized antibiotics for a COPD exacerbation within the 5 weeks prior to the Screening Visit or during the Screening Phase.
  • Known selective or severe Immunoglobulin A (IgA) deficiency.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Placebo0.9% Sodium Chloride for Injection, USP0.9% Sodium Chloride for Injection, USP, administered weekly by IV infusion for 156 weeks
Alpha-1 MP 120 mg/kgAlpha-1 MPAlpha-1 MP 120 mg/kg administered weekly by IV infusion for 156 weeks
Alpha-1 MP 60 mg/kgAlpha-1 MPAlpha-1 MP 60 mg/kg administered weekly by IV infusion for 156 weeks
Primary Outcome Measures
NameTimeMethod
Change from Baseline in Whole lung PD15 (15th percentile point)Week -3 (baseline measure), Week 52, Week 104, Week 130, Week 156

Whole lung PD15 measured by CT scan

Secondary Outcome Measures
NameTimeMethod
Discontinuations from the study due to AEsWeek -3 through Week 160

Monitoring of discontinuations due to AEs

Changes from baseline in forced expiratory volume in 1 second (FEV1)Weeks 26, 52, 78, 104, 130 and 156

FEV1 performed according to ATS/ERS guidelines

Severe COPD ExacerbationsWeek -3 through Week 160

Severe COPD exacerbations as defined by American Thoracic Society/European Respiratory Society (ATS/ERS) criteria (i.e., COPD exacerbations requiring hospitalization)

Change from Baseline in PD15 of the basal lung regionWeek -3 (baseline measure), Week 52, Week 104, Week 130, Week 156

PD15 of the basal lung region measure by CT scan

Change from baseline in carbon monoxide diffusing capacity (DLco)Weeks 26, 52, 78, 104, 130 and 156

DLco performed according to American Thoracic Society/European Respiratory Society (ATS/ERS) guidelines

Adverse Events (AEs)Week -3 through Week 160

Monitoring of AEs

Serious Adverse Events (SAEs)Week -3 through Week 160

Monitoring of SAEs

Change from baseline in Saint George's Respiratory Questionnaire: Minimum value = 0, maximum value = 100, higher scores indicate worse conditionWeeks 26, 52, 78, 104, 130 and 156

Health-related quality of life assessment tool

Change from baseline in the EuroQoL (Quality of Life)- 5 Dimension- 5 Level (EQ-5D-5L): Minimum value (for each one of the 5 levels) = 1, maximum value (for each one of the 5 levels) = 5, higher scores indicate worse conditionWeeks 26, 52, 78, 104, 130 and 156

Heath-related quality of life assessment tool

Trial Locations

Locations (52)

Institutul de Ftiziopneumologie "Chiril Draganiuc"

🇲🇩

Chisinau, Moldova, Republic of

St. Joseph's Hospital and Medical Center

🇺🇸

Phoenix, Arizona, United States

Washington University School of Medicine

🇺🇸

Saint Louis, Missouri, United States

University of Florida

🇺🇸

Gainesville, Florida, United States

Medical Research of Central Florida, LLC

🇺🇸

Leesburg, Florida, United States

Accellacare

🇺🇸

Wilmington, North Carolina, United States

Faculdade de Medicina do ABC

🇧🇷

Santo André, Sao Paulo, Brazil

University of Miami Miller School of Medicine

🇺🇸

Miami, Florida, United States

Oregon Health & Science University

🇺🇸

Portland, Oregon, United States

Penn State Univ. Milton S. Hershey Medical Center

🇺🇸

Hershey, Pennsylvania, United States

Medical University of South Carolina

🇺🇸

Charleston, South Carolina, United States

University of Texas Health Center at Tyler

🇺🇸

Tyler, Texas, United States

Hospital del Torax Dr. Antonio A. Cetrangolo

🇦🇷

Vicente Lopez, Buenos Aires, Argentina

Centro Dr. Lazaro Langer

🇦🇷

Cordoba, Argentina

St Vincent's Hospital Sydney

🇦🇺

Sydney, New South Wales, Australia

The Prince Charles Hospital

🇦🇺

Chermside, Queensland, Australia

Royal Adelaide Hospital

🇦🇺

Adelaide, South Australia, Australia

Institute for Respiratory Health Inc

🇦🇺

Nedlands, Western Australia, Australia

St Vincent's Hospital Melbourne

🇦🇺

Fitzroy, Victoria, Australia

UNIFESP - Universidade Federal de São Paulo

🇧🇷

São Paulo, Sao Paulo, Brazil

Instituto do Coração - Incor- HCFMUSP

🇧🇷

São Paulo, Brazil

Health Sciences Centre

🇨🇦

St. John's, Newfoundland and Labrador, Canada

Queen Elizabeth II Health Sciences Centre

🇨🇦

Halifax, Nova Scotia, Canada

Inspiration Research Limited

🇨🇦

Toronto, Ontario, Canada

Århus Universitetshospital

🇩🇰

Arhus C, Denmark

Gentofte Hospital

🇩🇰

Hellerup, Denmark

North Estonia Medical Centre Foundation

🇪🇪

Tallinn, Estonia

Tartu University Hospital

🇪🇪

Tartu, Estonia

Turku University Central Hospital, Department of Pulmonary Diseases

🇫🇮

Turku, Finland

Universitaetsklinikum Heidelberg

🇩🇪

Heidelberg, Baden Wuerttemberg, Germany

Universitaetsklinikum Giessen und Marburg GmbH

🇩🇪

Marburg, Hessen, Germany

Groupe Hospitalier Sud - Hôpital Haut-Lévêque

🇫🇷

Pessac, Gironde, France

Hôpital Cardio-Vasculaire et Pneumologique Louis Pradel

🇫🇷

Bron, Rhone, France

Ruhrlandklinik

🇩🇪

Essen, Nordrhein Westfalen, Germany

Univer des Saarlandes Innere

🇩🇪

Homburg Saar, Germany

New Zealand Respiratory and Sleep institute

🇳🇿

Auckland, New Zealand

Christchurch Hospital NZ

🇳🇿

Christchurch, New Zealand

Waikato Hospital

🇳🇿

Hamilton, New Zealand

SPZOZ Szpital Uniwersytecki w Krakowie

🇵🇱

Krakow, Poland

Instytut Gruzlicy i Chorob Pluc w Warszawie

🇵🇱

Warszawa, Poland

SAIH of Yaroslavl region "Clinical Hospital of Emergency Medical Care n.a. N. V. Solovyev

🇷🇺

Yaroslavl, Russian Federation

Clinic Dr.G Curteanu Oradea

🇷🇴

Oradea, Romania

Spitalul Clinic de Boli Infectioase si Pneumoftiziologie

🇷🇴

Timisoara, Romania

SBEI HPE Altai State Medical University of MoH and SD

🇷🇺

Barnaul, Russian Federation

Hospital Universitario Central de Asturias

🇪🇸

Oviedo, Asturias, Spain

Hospital de Cruces

🇪🇸

Barakaldo, Vizcaya, Spain

FSI Scientific Research Institute of Pulmonology

🇷🇺

Moscow, Russian Federation

Sahlgrenska Sjukhuset

🇸🇪

Göteborg, Sweden

CTC - Clinical Trial Consultants AB

🇸🇪

Linköping, Sweden

Skånes Universitetssjukhus, Malmö

🇸🇪

Malmö, Sweden

Karolinska Universitetssjukhuset, Solna

🇸🇪

Stockholm, Sweden

CTC Clinical Trial Consultants AB

🇸🇪

Uppsala, Sweden

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