MedPath

A Study of Avastin (Bevacizumab) in Combination With XELOX or FOLFOX-4 in Patients With Metastatic Colorectal Cancer.

Phase 3
Completed
Conditions
Colorectal Cancer
Interventions
Drug: XELOX
Drug: FOLFOX-4
Registration Number
NCT00349336
Lead Sponsor
Hoffmann-La Roche
Brief Summary

This 2 arm study will compare the pharmacokinetics and safety of Avastin at steady state under 2 different dosing regimens, in combination with XELOX (oxaliplatin + Xeloda) or FOLFOX-4 (oxaliplatin, leucovorin and 5-fluorouracil). Patients randomized to the XELOX arm will receive Avastin (7.5mg/kg iv) on Day 1 of each 3 week cycle; patients randomized to the FOLFOX-4 arm will receive Avastin (5mg/kg iv) on Day 1 of each 2 week cycle. The anticipated time on study treatment is 3-12 months, and the target sample size is \<100 individuals.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
64
Inclusion Criteria
  • adult patients, >=18 years of age;
  • adenocarcinoma of the colon or rectum, with metastatic or locally advanced disease;
  • >=1 target lesion.
Exclusion Criteria
  • patients who have previously received systemic treatment for advanced or metastatic disease;
  • patients who have received adjuvant treatment for non-metastatic disease in past 3 months;
  • previous therapy with oxaliplatin or Avastin.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
1bevacizumab [Avastin]-
1XELOX-
2bevacizumab [Avastin]-
2FOLFOX-4-
Primary Outcome Measures
NameTimeMethod
Weekly Steady-state Exposure of BevacizumabUp to 48 weeks

Area under the serum concentration-time curve per week, at steady state (AUCss per week). Estimation of the parameter was performed using non-compartmental methods.

Secondary Outcome Measures
NameTimeMethod
Time Zero to Last Measurable Plasma Concentration of BevacizumabUp to 48 weeks

Area under the serum concentration-time curve from time zero to the time of the last measurable plasma concentration (AUC 0-last). Estimation of the parameter was performed using non-compartmental methods.

Steady-state Exposure of Bevacizumab From Time Zero to TauUp to 48 weeks

Area under the serum concentration-time curve from time zero to tau, at steady state (AUCss 0-tau), where tau was the length of the cycle, i.e., tau = 3 weeks for XELOX+BV and tau = 2 weeks for FOLFOX-4+BEV. Estimation of the parameter was performed using non-compartmental methods.

Maximum Serum Concentration of Bevacizumab at Steady StateUp to 48 weeks

Maximum serum concentration at steady state (Css,max). Estimation of the parameter was performed using non-compartmental methods.

Minimum Serum Concentration of Bevacizumab at Steady StateUp to 48 weeks

Minimum serum concentration at steady state (Css, min). Estimation of the parameter was performed using non-compartmental methods.

Serum Clearance of BevacizumabUp to 48 weeks

Serum clearance (CL). Estimation of the parameter was performed using non-compartmental methods.

Time of Maximum Serum Concentration of BevacizumabUp to 48 weeks

Time of maximum serum concentration (tmax). Estimation of the parameter was performed using non-compartmental methods.

Volume of Distribution of Bevacizumab at Steady StateUp to 48 weeks

Volume of distribution at steady state (Vss). Estimation of the parameter was performed using non-compartmental methods.

Terminal Half-life of BevacizumabUp to 48 weeks

Terminal half-life (t1/2) (apparent elimination half-life). Estimation of the parameter was performed using non-compartmental methods.

© Copyright 2025. All Rights Reserved by MedPath