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Tesetaxel Plus Reduced Dose of Capecitabine in Patients With HER2 Negative, HR Positive, LA/MBC

Phase 2
Terminated
Conditions
Breast Cancer
Interventions
Registration Number
NCT03858972
Lead Sponsor
Odonate Therapeutics, Inc.
Brief Summary

CONTESSA 2 is a multinational, multicenter, Phase 2 study of tesetaxel in patients with HER2 negative, HR positive, locally advanced or metastatic breast cancer (LA/MBC) not previously treated with a taxane. The primary objective of the study is to establish the efficacy of tesetaxel plus a reduced dose of capecitabine based on objective response rate (ORR) as assessed by an Independent Radiologic Review Committee (IRC). 152 patients were enrolled.

Detailed Description

CONTESSA 2 is a multinational, multicenter, Phase 2 study of tesetaxel, an investigational, orally administered taxane, in patients with HER2 negative, HR Positive, LA/MBC not previously treated with a taxane in the neoadjuvant, adjuvant or metastatic setting. This Study complements CONTESSA, a multinational, multicenter, randomized, Phase 3 study in patients with HER2 negative, HR positive LA/MBC previously treated with a taxane in the neoadjuvant or adjuvant setting. 152 patients were enrolled, including 149 who received treatment. Patients are administered tesetaxel at 27 mg/m2 orally once every 21 days on the first day of each 21-day cycle plus capecitabine at 825 mg/m2 orally twice daily (for a total daily dose of 1,650 mg/m2) for 14 days of each 21-day cycle. Patients in the dense pharmacokinetics (PK) cohort receive a single dose of capecitabine monotherapy prior to starting the combination regimen. Capecitabine is an oral chemotherapy agent that is considered a standard-of-care treatment in LA/MBC. The primary efficacy endpoint is ORR as assessed by the IRC. The secondary efficacy endpoints are duration of response (DoR) as assessed by the IRC, progression-free survival (PFS) as assessed by the IRC, disease control rate (DCR) as assessed by the IRC and overall survival (OS). CONTESSA 2 also investigates the PK of tesetaxel.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
152
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Tesetaxel (oral) and capecitabine (oral)TesetaxelCohort 1: Tesetaxel (27 mg/m2) once every 21 days on Day 1 of each 21-day cycle; and capecitabine (825 mg/m2) twice daily (total daily dose of 1,650 mg/m2) beginning with the evening dose on Day 1 through the morning dose on Day 15 of each 21-day cycle. Cohort 2: On Cycle 1, Day -1, either a single morning dose of capecitabine at 825 mg/m2 (Cohort 2A) or 1,250 mg/m2 (Cohort 2B). On Cycle 1, Day 1, a single dose of tesetaxel (27 mg/m2), followed 2 hours later by capecitabine (825 mg/m2), followed by an evening dose of capecitabine (825 mg/m2). Capecitabine (825 mg/m2) twice daily (total daily dose of 1,650 mg/m2) beginning with the morning dose on Day 2 through evening dose on Day 14 of Cycle 1. Starting with Cycle 2, tesetaxel (27 mg/m2) once every 21 days on Day 1 of each 21-day cycle; and capecitabine (825 mg/m2) twice daily (total daily dose of 1,650 mg/m2) beginning with the evening dose on Day 1 through the morning dose on Day 15 of each 21-day cycle.
Tesetaxel (oral) and capecitabine (oral)CapecitabineCohort 1: Tesetaxel (27 mg/m2) once every 21 days on Day 1 of each 21-day cycle; and capecitabine (825 mg/m2) twice daily (total daily dose of 1,650 mg/m2) beginning with the evening dose on Day 1 through the morning dose on Day 15 of each 21-day cycle. Cohort 2: On Cycle 1, Day -1, either a single morning dose of capecitabine at 825 mg/m2 (Cohort 2A) or 1,250 mg/m2 (Cohort 2B). On Cycle 1, Day 1, a single dose of tesetaxel (27 mg/m2), followed 2 hours later by capecitabine (825 mg/m2), followed by an evening dose of capecitabine (825 mg/m2). Capecitabine (825 mg/m2) twice daily (total daily dose of 1,650 mg/m2) beginning with the morning dose on Day 2 through evening dose on Day 14 of Cycle 1. Starting with Cycle 2, tesetaxel (27 mg/m2) once every 21 days on Day 1 of each 21-day cycle; and capecitabine (825 mg/m2) twice daily (total daily dose of 1,650 mg/m2) beginning with the evening dose on Day 1 through the morning dose on Day 15 of each 21-day cycle.
Primary Outcome Measures
NameTimeMethod
ORR as assessed by the IRCApproximately 2.0-2.5 years
Secondary Outcome Measures
NameTimeMethod
OSApproximately 3.0-3.5 years
DoR as assessed by the IRCApproximately 2.0-2.5 years
PFS as assessed by the IRCApproximately 2.0-2.5 years
DCR as assessed by the IRCApproximately 2.0-2.5 years
Central nervous system (CNS) ORR as assessed by the CNS IRC in patients with CNS metastases at baselineApproximately 2.0-2.5 years
CNS DoR as assessed by the CNS IRC in patients with CNS metastases at baselineApproximately 2.0-2.5 years
CNS PFS as assessed by the CNS IRC in patients with CNS metastases at baseline or a history of CNS metastases and in the intent-to-treat (ITT) populationApproximately 2.0-2.5 years
CNS OS in patients with CNS metastases at baseline or a history of CNS metastasesApproximately 3.0-3.5 years

Trial Locations

Locations (25)

Texas Oncology - Baylor Charles A. Sammons Cancer Center

🇺🇸

Dallas, Texas, United States

Asan Medical Center

🇰🇷

Seoul, Korea, Republic of

Hopital Maisonneuve-Rosemont

🇨🇦

Montréal, Canada

West Cancer Center

🇺🇸

Germantown, Tennessee, United States

Centre Hospitalier Universitaire de Sherbrooke CIUSSS de lEstrie CHUS patyre

🇨🇦

Sherbrooke, Canada

Ajou University Hospital

🇰🇷

Suwon, Korea, Republic of

Virginia Oncology Associates

🇺🇸

Norfolk, Virginia, United States

Fundacion Jimenez Diaz

🇪🇸

Madrid, Spain

National Cancer Center

🇰🇷

Goyang, Korea, Republic of

McGill University Health Center

🇨🇦

Montréal, Canada

National Taiwan University Hospital

🇨🇳

Taipei City, Taiwan

Hospital Teresa Herrera Materno-Infantil (CHUAC)

🇪🇸

A Coruña, Spain

Center Hospitalier de Montreal CHUM McPeak Sirois

🇨🇦

Montréal, Canada

Border Medical Oncology

🇦🇺

Albury, New South Wales, Australia

CIUSSS de Centre-Ouest-de-l'Île-de-Montréal Jewish General Hospital

🇨🇦

Montréal, Canada

Innovative Clinical Research Institute

🇺🇸

Whittier, California, United States

Sarah Cannon Research Institute - Florida Cancer Specialists

🇺🇸

Fort Myers, Florida, United States

Dana-Farber Cancer Institute

🇺🇸

Boston, Massachusetts, United States

Rocky Mountain Cancer Center

🇺🇸

Lakewood, Colorado, United States

Florida Cancer Specialists and Research Institute

🇺🇸

Saint Petersburg, Florida, United States

New York Cancer and Blood Specialists

🇺🇸

East Setauket, New York, United States

CHU de Quebec-University Laval

🇨🇦

Québec, Canada

Kyungpook National University Hospital

🇰🇷

Daegu, Korea, Republic of

Koo Foundation Sun Yat-Sen Cancer Center

🇨🇳

Taipei, Taiwan

Gangnam Severance Hospital

🇰🇷

Seoul, Korea, Republic of

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