MedPath

A Phase 1 Study of AB521 Monotherapy and Combination Therapies in Renal Cell Carcinoma and Other Solid Tumors (ARC-20)

Phase 1
Recruiting
Conditions
Clear Cell Renal Cell Carcinoma
Solid Tumors
Interventions
Registration Number
2024-519142-70-00
Lead Sponsor
Arcus Biosciences Inc.
Brief Summary

The purpose of this study is to evaluate the safety and tolerability of:

* casdatifan when taken alone in participants with advanced solid tumor malignancies and clear cell renal cell carcinoma (ccRCC) during the dose escalation stage; and

* casdatifan monotherapy and casdatifan in combination with cabozantinib or zimberelimab in participants with ccRCC in the dose expansion stage

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
Not specified
Target Recruitment
7
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Dose Escalation Cohort 1casdatifanParticipants will receive casdatifan orally once daily
Dose Escalation Cohort 2casdatifanParticipants will receive casdatifan orally once daily
Dose Escalation Cohort 3casdatifanParticipants will receive casdatifan orally twice daily
Dose Escalation Cohort 4casdatifanParticipants will receive casdatifan orally once daily
Dose Escalation Cohort 5casdatifanParticipants will receive casdatifan orally once daily
Dose Expansion Cohort 1casdatifanParticipants will receive casdatifan orally
Dose Expansion Cohort 2casdatifanParticipants will receive casdatifan orally
Dose Expansion Cohort 3casdatifanParticipants will receive casdatifan orally
Dose Expansion Cohort 4casdatifanParticipants will receive casdatifan orally with with cabozantinib orally
Dose Expansion Cohort 4CabozantinibParticipants will receive casdatifan orally with with cabozantinib orally
Dose Expansion Cohort 5casdatifanParticipants will receive casdatifan orally
Dose Expansion Cohort 6casdatifanParticipants will receive casdatifan orally
Dose Expansion Cohort 7casdatifanParticipants will receive casdatifan orally with zimberelimab infusion
Dose Expansion Cohort 7ZimberelimabParticipants will receive casdatifan orally with zimberelimab infusion
Dose Expansion Cohort 8casdatifanParticipants will receive casdatifan orally
Primary Outcome Measures
NameTimeMethod
Number of participants with dose limiting toxicities (DLTs)Up to 4 months
Number of participants with adverse events (AEs)Up to 4 months
Secondary Outcome Measures
NameTimeMethod
Objective Response Rate as measured by Response Evaluation Criteria in Solid Tumors (RECIST) v1.1Up to 4 months
Area under the plasma concentration time curve (AUC) of casdatifanUp to 4 months
Maximum Observed Plasma Concentration (Cmax) of casdatifanUp to 4 months
Plasma concentration of casdatifanUp to 4 months

Trial Locations

Locations (28)

University of California at San Diego

🇺🇸

San Diego, California, United States

Medical Oncology Associates Summit Cancer Centers

🇺🇸

Spokane, Washington, United States

Chris O'Brien Lifehouse

🇦🇺

Camperdown, Australia

Box Hill Hospital

🇦🇺

Melbourne, Australia

Macquarie University Hospital

🇦🇺

Sydney, Australia

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

UCLA

🇺🇸

Santa Monica, California, United States

University of Miami

🇺🇸

Miami, Florida, United States

Emory University

🇺🇸

Atlanta, Georgia, United States

University of Louisville Brown Cancer Center

🇺🇸

Louisville, Kentucky, United States

Scroll for more (18 remaining)
University of California at San Diego
🇺🇸San Diego, California, United States

MedPath

Empowering clinical research with data-driven insights and AI-powered tools.

© 2025 MedPath, Inc. All rights reserved.