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Efficacy, Safety and Tolerability of KLU156 in Adults and Children ≥ 5 kg Body Weight With Uncomplicated P. Falciparum Malaria

Phase 3
Recruiting
Conditions
Uncomplicated Plasmodium Falciparum Malaria
Interventions
Registration Number
NCT05842954
Lead Sponsor
Novartis Pharmaceuticals
Brief Summary

This study aims to confirm the efficacy, safety and tolerability of KLU156, a fixed dose combination of ganaplacide (KAF156) and a solid dispersion formulation of lumefantrine (lumefantrine-SDF), when administered once daily for three days in adults and children ≥ 5 kg body weight and ≥ 2 months of age suffering from uncomplicated P. falciparum malaria (with or without other Plasmodium spp. co-infection).

In the Extension phase, the safety, tolerability and efficacy of repeated treatment with KLU156 will be assessed for a maximum of two years in patients who did not experience early treatment failure (ETF), who did not experience any study treatment-related SAE (Serious Adverse Event) previously and who gave informed consent to participate in the Extension phase.

Detailed Description

The purpose of this study is to confirm the efficacy, safety and tolerability of KLU156 in patients with uncomplicated P. falciparum malaria (with or without other Plasmodium spp. co-infection) by demonstrating that KLU156 is non-inferior to Coartem.

* The study duration will be 43 days (Core phase) plus 24 months (Extension phase).

* The treatment duration will be 3 days for each malaria episode.

* The visit frequency will be Days 1-3 (hospitalized) and 5 follow-up visits (Days 4, 8, 22, 29 and 43) in the Core phase and Days 1-3 (hospitalized) and 3 follow-up visits (Days 4, 8 and 29) in the Extension phase.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
1500
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
KLU156KLU156KLU156 once daily (QD) for 3 days under fed conditions (light meal).
CoartemCoartemCoartem twice a day (BID) for 3 days under fed conditions.
Primary Outcome Measures
NameTimeMethod
PCR-corrected adequate clinical and parasitological response (ACPR)Day 29 (i.e., 28 days post-first dose administration)

To confirm the efficacy of KLU156 in adults and children ≥ 5 kg body weight and ≥ 2 months of age suffering from uncomplicated malaria caused by P. falciparum (with or without other Plasmodium spp. co-infection) by demonstrating that KLU156 is non-inferior to Coartem (non-inferiority margin = 5%) based on the PCR-corrected ACPR at Day 29.

Secondary Outcome Measures
NameTimeMethod
Proportion of patients with parasitemia12, 24, 48 and 72 hours after treatment

For the parasitemia assessment, blood sampling can be done by means of a finger prick except when the timing for parasitology assessments coincides with time for clinical laboratory tests, in which case, blood sample can be taken from the venous blood collected for clinical laboratory analyses.

GametocytemiaFrom baseline up to Day 43

Disappearance or development of gametocytemia in patients with or without gametocytemia at baseline (pre-first dose administration), respectively

PCR-corrected and uncorrected ACPRDays 22 and 43 (i.e., 21 and 42 days post-first dose administration)

To confirm the efficacy of KLU156 by assessing uncorrected and PCR-corrected ACPR at additional time points

Fever Clearance TimeUp to Day 3

To confirm the efficacy of KLU156 by assessing fever clearance between the two treatment arms

Parasite Clearance TimeUp to Day 3

To assess parasite clearance time between the two treatment arms

Extension phase: PCR-corrected and uncorrected ACPRDay 29 of malaria episode

To evaluate efficacy over repeated treatment with KLU156 in adults and children ≥ 5 kg body weight and ≥ 2 months of age suffering from uncomplicated malaria caused by P. falciparum (with or without other Plasmodium spp. co-infection) for a maximum of 2 years

Extension phase: Gametocyte carriage over timeUp to 2 years

To assess gametocyte carriage over time by malaria episode in the extension phase

Uncorrected ACPRDay 29

To further confirm the efficacy of KLU156 by demonstrating non-inferiority of KLU156 to Coartem (NI margin 7.5%) based on the uncorrected ACPR at Day 29

Incidence and severity of Adverse Events (AEs) and Serious Adverse Events (SAEs)Day 43

Incidence and severity of AEs and SAEs by treatment group, including changes in vital signs, electrocardiograms (ECGs), and laboratory results qualifying and reported as AEs.

Incidence rate of recrudescence and new infectionDays 22, 29 and 43

Proportion of patients with recrudescence and new infections between the two treatment arms

Extension phase: KLU156-related AE/SAE incidence and severity by malaria episodeUp to 2 years

To assess the safety and tolerability over repeated treatment with KLU156 in adults and children ≥ 5 kg body weight and ≥ 2 months of age suffering from uncomplicated malaria caused by P. falciparum (with or without other Plasmodium spp. co-infection) for a maximum of 2 years

Trial Locations

Locations (1)

Novartis Investigative Site

🇿🇲

Ndola, Zambia

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