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Hydroxychloroquine for Thrombosis Prevention and Antiphospholipid Antibody Reduction in Primary Antiphospholipid Syndrome

Not Applicable
Completed
Conditions
Antiphospholipid Syndrome
Interventions
Registration Number
NCT04153201
Lead Sponsor
National and Kapodistrian University of Athens
Brief Summary

This is an interventional drug study designed as a pilot for a randomized clinical trial, aimed at assessing the effect of hydroxychloroquine on the incidence rate of thrombosis in patients with primary antiphospholipid syndrome as the main outcome, as well as the safety of hydroxychloroquine administration in this population. In addition, the effect of hydroxychloroquine on antiphospholipid antibody titers will be assessed.

Detailed Description

Patients with primary antiphospholipid syndrome (either thrombotic or obstetric) on regular follow-up at our outpatient rheumatology department and being treated with standard care (systemic anticoagulants and/or antiplatelet agents), are randomized to receive either hydroxychloroquine plus standard care, or standard care alone, on a 1:1 ratio using block size 2 randomization, after exclusion of patients with contraindications to hydroxychloroquine or prior hydroxychloroquine use within 12 months of consideration for enrollment. Patients are monitored clinically every 3 months and the development of thrombosis and/or adverse effects attributable to hydroxychloroquine is recorded. Antiphospholipid antibody titers (anti-cardiolipin immunoglobulin G (IgG)/Immunoglobulin M (IgM) and anti-beta2-glycoprotein I IgG/IgM isotypes) are measured semi-annually. Intention-to-treat survival analysis is applied for assessing the effect of hydroxychloroquine on the incidence of thrombosis. Longitudinal mixed linear models are applied for assessing the effect of hydroxychloroquine on longitudinal titers of antiphospholipid antibodies.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
50
Inclusion Criteria

Adult patients diagnosed with primary antiphospholipid syndrome (PAPS) [updated Sapporo criteria: Miyakis et al, J Thromb Haemost. 2006 Feb;4(2):295-306. PubMed 16420554]

Exclusion Criteria
  1. ≥4 American College of Rheumatology (ACR) classification criteria for Systemic Lupus Erythematosus (SLE)
  2. ACR classification criteria for other systemic autoimmune disorders
  3. active malignancy
  4. treatment with Hydroxychloroquine (HCQ) in the previous 12 months
  5. history of serious adverse events or contraindication to HCQ including a history of HCQ allergy, HCQ eye toxicity, or glucose-6-phosphate dehydrogenase deficiency, uncontrolled seizure disorder, liver enzyme elevation >2-fold the upper normal limit, and creatinine clearance <30ml/min

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
HydroxychloroquineHydroxychloroquinePatients with primary antiphospholipid syndrome started on hydroxychloroquine while continuing standard care (vitamin K antagonists or direct oral anticoagulants, and/or antiplatelet agents, depending on primary APS subgroup)
Primary Outcome Measures
NameTimeMethod
Incident acute thrombosis in the venous or arterial circulation3 years

incident acute arterial thrombosis (myocardial infarction, stroke, transient ischemic attack, occlusion of the peripheral limb and neck, splanchnic, or retinal arteries) or venous thrombosis (pulmonary embolism, deep vein thrombosis, splanchnic vein thrombosis, retinal vein occlusion) confirmed by appropriate imaging studies (doppler ultrasonography, computed tomography pulmonary angiogram, conventional angiography, magnetic resonance angiography, ventilation/perfusion lung scintigraphy)

Secondary Outcome Measures
NameTimeMethod
General safety outcomes3 years

* Hospitalization for any cause

* Death of any cause

* APS-related death (based on death certificate records)

Hydroxychloroquine-related safety outcomes3 years

* Retinal toxicity by ocular examination, visual field testing and optical coherence tomography yearly and upon reporting visual symptoms

* Toxic myopathy: new onset motor strength \<=4/5, myalgia and creatine kinase elevation

* Liver toxicity: liver enzyme elevations \>3x of upper limit of normal (ULN), or serum total bilirubin \>2x ULN, with no cholestasis

* Metabolism disorders (hypoglycemia, weight decrease) by quarterly body weight and blood glucose testing

* Bone marrow suppression: drop in hemoglobin to \< 10 mg/dl, white blood cells \< 3700/μL, platelets \< 150,000/μL according to a hematologist

* Cardiac complications (conduction defects, QT prolongation, cardiomyopathy) screened by interview, physical examination, and semi-annual electrocardiogram

* Seizures screened by interview and confirmed by electrocardiogram

* Gastrointestinal upset, allergic reactions, skin reactions by interview and physical exam

Anticoagulation treatment-related safety outcomes3 years

* Major bleeding, defined as fatal bleeding, or symptomatic bleeding in a critical area or organ, such as intracranial, intraspinal, intraocular, retroperitoneal, intra-articular or pericardial, or intramuscular with compartment syndrome, and/or bleeding causing a fall in hemoglobin level of 2 g/dL or more, or leading to transfusion of two or more units of whole blood or red cells.

* Minor bleeding defined as clinically evident bleeding not fulfilling the definition of major bleeding

Trial Locations

Locations (1)

Laikon General Hospital

🇬🇷

Athens, Attiki, Greece

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