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Safety and Efficacy of Itacitinib in Combination With Corticosteroids for Treatment of Graft-Versus-Host Disease in Pediatric Subjects

Phase 1
Terminated
Conditions
Acute Graft-versus-host Disease
Interventions
Drug: Corticosteroids
Registration Number
NCT03721965
Lead Sponsor
Incyte Corporation
Brief Summary

The purpose of this study is to evaluate itacitinib in combination with corticosteroids for the treatment of Grades II to IV acute graft-versus-host disease (aGVHD) in steroid-naive pediatric participants.

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
2
Inclusion Criteria
  • Male and female participants: 12 to < 18 years old (Cohort 1), 6 to < 12 years old (Cohort 2), 2 to < 6 years old (Cohort 3), Weighing > 8 kg to < 2 years old (Cohort 4), and 28 days old to weighing ≤ 8 kg (Cohort 5).
  • Undergone 1 allogeneic hematopoietic stem cell transplantation (allo-HSCT) from any donor and source for hematological malignancies or disorders. Recipients of myeloablative and reduced-intensity conditioning regimens are eligible.
  • Clinically suspected Grade II to IV aGVHD as per Mount Sinai Acute GVHD International Consortium (MAGIC) criteria, occurring after allo-HSCT and any GVHD prophylactic medication.
  • Evidence of myeloid engraftment.
Exclusion Criteria
  • More than 1 allo-HSCT.
  • Received more than 2 days of systemic corticosteroids for aGVHD before the first study drug administration.
  • Presence of GVHD overlap syndrome.
  • Presence of an active uncontrolled infection.
  • Known HIV infection.
  • Active hepatitis B virus (HBV) or hepatitis C virus (HCV) infection that requires treatment or at risk for HBV reactivation.
  • Evidence of relapsed primary disease or have been treated for relapse after the allo-HSCT was performed.
  • Any corticosteroid therapy for indications other than GVHD at doses > 1 mg/kg once daily of methylprednisolone (or equivalent) within 7 days of the first study drug administration.
  • Receipt of live (including attenuated) vaccines or anticipation of need for such vaccines during the study.
  • Receipt of JAK inhibitor therapy after allo-HSCT for any indication.
  • Treatment with any other investigational agent, device, or procedure within 21 days (or 5 half-lives, whichever is greater) of enrollment.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Itacitinib + CorticosteroidsItacitinib-
Itacitinib + CorticosteroidsCorticosteroids-
Primary Outcome Measures
NameTimeMethod
Phase 1: Number of Participants With Treatment-emergent Adverse Events (TEAEs)up to 45 days

A TEAE was defined as an AE that began or worsened from Baseline after the first administration of study drug.

Phase 1: Cmax of Itacitinib When Administered With CorticosteroidsDay 1: 1, 2, 4, and 6 hours post-dose. Day 7: predose; 1, 2, 4, and 6 hours post-dose

Cmax was defined as the maximum observed plasma concentration.

Phase 1: Cmin of Itacitinib When Administered With CorticosteroidsDay 1: 1, 2, 4, and 6 hours post-dose. Day 7: predose; 1, 2, 4, and 6 hours post-dose

Cmin was defined as the minimum observed plasma concentration.

Phase 1: Tmax of Itacitinib When Administered With CorticosteroidsDay 1: 1, 2, 4, and 6 hours post-dose. Day 7: predose; 1, 2, 4, and 6 hours post-dose

Tmax was defined as the time to the maximum concentration.

Phase 1: AUC of Itacitinib When Administered With CorticosteroidsDay 1: 1, 2, 4, and 6 hours post-dose. Day 7: predose; 1, 2, 4, and 6 hours post-dose

AUC was defined as the area under the plasma concentration-time curve.

Phase 1: Cl/F of Itacitinib When Administered With CorticosteroidsDay 1: 1, 2, 4, and 6 hours post-dose. Day 7: predose; 1, 2, 4, and 6 hours post-dose

Cl/F was defined as the apparent oral dose clearance.

Phase 2: Overall Response Rate up to Day 28up to Day 28

Overall response rate was defined as the number of participants demonstrating a complete response (CR), a very good partial response (VGPR), or a partial response (PR).

Secondary Outcome Measures
NameTimeMethod
Phase 2: Relapse Rate of Malignant and Nonmalignant Disordersup to approximately 12 months

Relapse rate was defined as the number of participants whose underlying disease relapsed.

Phase 2: Malignant and Nonmalignant Disorders Relapse-related Mortality Rateup to approximately 12 months

Mortality rate was defined as the number of participants whose underlying hematologic disorder relapsed and had a fatal outcome.

Phase 2: Failure-free Survivalup to 6 months

Failure-free survival was defined as the number of participants who were still alive, had not relapsed, had not required additional therapy for acute graft-versus-host disease (aGVHD), and had not demonstrated signs or symptoms of chronic GVHD.

Phase 2: Overall Survivalup to approximately 12 months

Overall survival was defined as the interval from study enrollment to death due to any cause.

Phase 2: Incidence Rate of Secondary Graft Failureup to approximately 12 months

Analysis was to be conducted to assess the number of participants experiencing secondary graft failure.

Phase 2: Average Corticosteroid Useup to 180 days

The average number of participants who discontinued corticosteroids was to be assessed.

Phase 2: Number of Participants With TEAEsup to 12 months

A TEAE was defined as an AE that began or worsened from Baseline after the first administration of study drug.

Phase 2: Cmax of Itacitinib When Administered With CorticosteroidsDay 7: predose; 1, 2, and 4 hours post-dose

Cmax was defined as the maximum observed plasma concentration.

Phase 2: Cmin of Itacitinib When Administered With CorticosteroidsDay 7: predose; 1, 2, and 4 hours post-dose

Cmin was defined as the minimum observed plasma concentration.

Phase 2: Tmax of Itacitinib When Administered With CorticosteroidsDay 7: predose; 1, 2, and 4 hours post-dose

Tmax was defined as the time to the maximum concentration.

Phase 2: AUC of Itacitinib When Administered With CorticosteroidsDay 7: predose; 1, 2, and 4 hours post-dose

AUC was defined as the area under the plasma concentration-time curve.

Phase 2: Cl/F of Itacitinib When Administered With CorticosteroidsDay 7: predose; 1, 2, and 4 hours post-dose

Cl/F was defined as the apparent oral dose clearance.

Phase 2: Overall Response Rate up to 100 Daysup to 100 days

Overall response rate was defined as the number of participants demonstrating a CR, a VGPR, or a PR.

Phase 1: Overall Response Rateup to Day 28

Overall response rate was defined as the number of participants demonstrating a CR, a VGPR, or a PR.

Phase 2: Non Relapse Mortalityup to 24 months

Non relapse mortality was defined as the number of participants who died due to causes other than underlying hematologic disorders relapse.

Phase 2: Duration of Responseup to approximately 12 months

Duration of response was defined as the time of the onset of response to the loss of response.

Phase 2: Time to Responseup to approximately 12 months

Time to response was defined as the interval from treatment initiation to the first response.

Phase 2: Cumulative Corticosteroid Doseup to 180 days

The number of participants with various cumulative corticosteroid doses was assessed.

Phase 2: Number of Participants Who Discontinued Corticosteroidsup to 100 days

The number of participants who discontinued corticosteroids was assessed.

Phase 2: Number of Participants Who Discontinued Immunosuppressive Medicationup to 100 days

The number of participants who discontinued immunosuppressive medication was assessed.

Phase 2: Number of Participants With aGVHD Flaresup to 100 Days

The number of participants who experienced aGVHD flares requiring treatment was assessed.

Phase 2: Number of Participants With Chronic Graft-versus-host Disease (cGVHD)up to 365 days

The number of participants with a diagnosis of any cGVHD, including mild, moderate, severe, was assessed.

Trial Locations

Locations (36)

University of Minnesota Medical Center

🇺🇸

Minneapolis, Minnesota, United States

Duke University Medical Center

🇺🇸

Durham, North Carolina, United States

University Hospitals Cleveland Medical Center - Rainbow Babies and Children's Hospital

🇺🇸

Cleveland, Ohio, United States

Children's Hospital of Philadelphia - Center for Childhood Cancer Research

🇺🇸

Philadelphia, Pennsylvania, United States

Childrens Hospital of Orange County

🇺🇸

Orange, California, United States

Robert Debre Hospital

🇫🇷

Paris, France

Royal Marsden Hospital - Surrey

🇬🇧

Surrey Quays, United Kingdom

City of Hope National Medical Center

🇺🇸

Duarte, California, United States

CHU Nancy

🇫🇷

Vandœuvre-lès-Nancy, France

Universitatsklinikum Jena, Klinik fur Kinder und Jugendmedizin

🇩🇪

Jena, Germany

Doernbecher Children's Hospital - Division of Pediatric Hematology

🇺🇸

Portland, Oregon, United States

Sarah Cannon Research Institute, LLC

🇺🇸

Nashville, Tennessee, United States

Vanderbilt University Medical Center

🇺🇸

Nashville, Tennessee, United States

Children's Hospital Colorado - Center for Cancer and Blood Disorders

🇺🇸

Aurora, Colorado, United States

Memorial Sloan Kettering Cancer Center

🇺🇸

New York, New York, United States

Nicklaus Children's Hospital

🇺🇸

Miami, Florida, United States

Universitaetsklinikum Aachen, AoeR

🇩🇪

Aachen, Germany

Fred Hutchinson Cancer Research Center

🇺🇸

Seattle, Washington, United States

Centre Hospitalier Universitaire de Rennes

🇫🇷

Rennes, Cedex 2, France

CHU de Grenoble

🇫🇷

Grenoble, France

CHRU Nancy

🇫🇷

Vandœuvre-lès-Nancy, France

Policlinico S. Orsola-Malpighi

🇮🇹

Bologna, Italy

Azienda Ospedaliero Unversitatia Policlinico - Vittorio Emanuele - Presido Ospedaliero G. Rodolico

🇮🇹

Catania, Italy

Fondazione MBBM

🇮🇹

Monza, Italy

Ospedale Pediatrico Bambino Gesu

🇮🇹

Roma, Italy

AOU Citta della Salute e della Scienza di Torino - Ospedale Regina Margherita

🇮🇹

Torino, Italy

Hospital Vall D Hebron

🇪🇸

Barcelona, Spain

Hospital Clinico de Santiago de Compostela

🇪🇸

Santiago De Compostela, Spain

Hospital Universitari i Politecnic La Fe

🇪🇸

Valencia, Spain

Great Ormond Street Hospital for Children

🇬🇧

London, United Kingdom

Bristol Royal Hospital for Children

🇬🇧

Bristol, United Kingdom

Birmingham Childrens Hospital

🇬🇧

Birmingham, United Kingdom

Leeds Teaching Hospitals NHS Trust

🇬🇧

Leeds, United Kingdom

Central Manchester University Hospital - Royal Manchester Children's Hospital

🇬🇧

Manchester, United Kingdom

Hopitaux Universitaires De Strasbourg

🇫🇷

Strasbourg Cedex, France

Nemours/A.I. duPont Hospital for Children

🇺🇸

Wilmington, Delaware, United States

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