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A Study to Assess How Food Affects the Safety and Pharmacokinetics of Galicaftor and Navocaftor

Phase 1
Completed
Conditions
Healthy Volunteers
Interventions
Registration Number
NCT05538585
Lead Sponsor
AbbVie
Brief Summary

Cystic Fibrosis (CF) is a rare, life-threatening, genetic disease that affects the lungs and digestive system, significantly impairing the quality of life, with those affected having a median age of death at 40. The objectives of this study are to assess the effect of food on the safety and pharmacokinetics of navocaftor and galicaftor.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
24
Inclusion Criteria
  • Body Mass Index (BMI) is => 18.0 to <= 32.0 kg/ m2 after rounding to the tenth's decimal.
  • A condition of general good health, based upon the results of a medical history, physical examination, vital signs, laboratory profile and a 12-lead electrocardiogram (ECG).
Exclusion Criteria
  • History of epilepsy, any clinically significant cardiac, respiratory (except mild asthma as a child), renal, hepatic, gastrointestinal, hematologic, or psychiatric disease or disorder, or any uncontrolled medical illness.
  • History of or active medical condition(s) or surgical procedure(s) that might affect gastrointestinal motility, pH, or absorption [e.g., Crohn's disease, celiac disease, gastroparesis, short bowel syndrome, gastric surgery (except pyloromyotomy for pyloric stenosis during infancy), cholecystectomy, vagotomy, bowel resection, etc.].
  • Evidence of dysplasia or history of malignancy (including lymphoma and leukemia) other than successfully treated non-metastatic cutaneous squamous cell, basal cell carcinoma or localized carcinoma in situ of the cervix.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Part 1: Navocaftor without foodNavocaftorParticipants will receive navocaftor administered without food
Part 1: Navocaftor with foodNavocaftorParticipants will receive navocaftor administered with food
Part 2: Galicaftor without foodGalicaftorParticipants will receive galicaftor administered without food
Part 2: Galicaftor with foodGalicaftorParticipants will receive galicaftor administered with food
Primary Outcome Measures
NameTimeMethod
Terminal Elimination Half-life (t1/2)Up to Day 4

Terminal elimination half-life (t1/2) will be assessed.

Time to Cmax (peak time, Tmax)Up to Day 4

Tmax will be assessed.

Number of Participants with Adverse Events (AEs)Up to Day 38

An adverse event (AE) is defined as any untoward medical occurrence in a patient or clinical investigation participant administered a pharmaceutical product which does not necessarily have a causal relationship with this treatment.

Area under the plasma curve (AUC)Up to Day 4

AUC will be assessed.

Maximum Observed Plasma Concentration (Cmax)Up to Day 4

Cmax will be assessed.

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (2)

Clinical Pharmacology of Miami /ID# 249531

🇺🇸

Miami, Florida, United States

Acpru /Id# 249532

🇺🇸

Grayslake, Illinois, United States

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