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Efficacy and Pharmacokinetic-Pharmacodynamic Relationship of Intranasally Administered Sufentanil, Ketamine, and CT001

Phase 2
Completed
Conditions
Pain
Interventions
Registration Number
NCT05508594
Lead Sponsor
Cessatech A/S
Brief Summary

A randomised, double-blind, parallel-group, study comparing the analgesic effect of intranasal CT001 to intranasal sufentanil, intranasal ketamine or placebo for treatment of acute pain in adults undergoing surgical removal of an impacted mandibular third molar, where bone removal is judged to be needed.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
220
Inclusion Criteria
  • Healthy (The American Society of Anaesthesiologists' Physical Classification System (ASA) I-II) male or female participants scheduled for surgical removal of an impacted mandibular third molar, where bone removal is judged to be needed
  • Age: ≥ 18 and < 56 years
  • Body Mass index above (>)18.5 or below (<) 30.0 kg/m2
  • Prior to randomisation: Numeric Pain Rating Scale (NRS anchored by 0 = "no pain", 10 = "worst pain imaginable") ≥ 5 at rest within 4 hours after the administration of the last dose of local anaesthetic
Exclusion Criteria
  • Current or history of any clinically significant disease or disorder, which, in the opinion of the investigator, may put the potential subject at risk when participating in the study, or influence the potential subject's ability to participate in the study or influence the study results.
  • Any clinically significant illness, medical/surgical procedure or trauma within 4 weeks of the administration of investigational product that is likely to introduce additional risk factors, jeopardize study integrity, or to interfere with the study assessments or procedure
  • History of increased bleeding tendency
  • Clinically significant mental illness
  • Opioid Risk Tool score of >3
  • Pain Catastrophizing Scale score, total points >30
  • Hospital Anxiety and Depression Scale (HADS), points ≥ 11 for anxiety or ≥ 11 points for depression
  • Daily intake of analgesics
  • History of alcohol or drug abuse or use of illicit drugs or positive screen for drugs of abuse at screening or on admission to the Clinic prior to the administration of the investigational product.
  • Abnormal nasal cavity/airway

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Sufentanil 13 mcg/Ketamine 40 mgKetamine-
Sufentanil 40 mcg/Ketamine 40 mgKetamine-
Sufentanil 40 mcg/Ketamine 13 mgKetamine-
CT001CT001-
PlaceboPlacebo-
Sufentanil 27 mcgSufentanil-
Sufentanil 40 mcg/Ketamine 27 mgKetamine-
Ketamine 27 mgKetamine-
Sufentanil 13 mcgSufentanil-
Ketamine 40 mgKetamine-
Ketamine 13 mgKetamine-
Sufentanil 40 mcgSufentanil-
Sufentanil 13 mcg/Ketamine 13 mgSufentanil-
Sufentanil 13 mcg/Ketamine 13 mgKetamine-
Sufentanil 13 mcg/Ketamine 27 mgSufentanil-
Sufentanil 13 mcg/Ketamine 27 mgKetamine-
Sufentanil 27 mcg/Ketamine 13 mgSufentanil-
Sufentanil 13 mcg/Ketamine 40 mgSufentanil-
Sufentanil 27 mcg/Ketamine 13 mgKetamine-
Sufentanil 27 mcg/Ketamine 40 mgSufentanil-
Sufentanil 27 mcg/Ketamine 40 mgKetamine-
Sufentanil 40 mcg/Ketamine 13 mgSufentanil-
Sufentanil 40 mcg/Ketamine 27 mgSufentanil-
Sufentanil 40 mcg/Ketamine 40 mgSufentanil-
Primary Outcome Measures
NameTimeMethod
Sum of pain intensity differences at 55 min0-55 min

Derived from pain intensity scores measured by the Numerical Rating Scale (0-10, 0= no pain, 10= worst possible pain).

PK-PD relationship for analgesic efficacy IN sufentanil, IN ketamine and IN CT0010-180 min

To assess the relationship between analgesic efficacy and the plasma concentrations of intranasal sufentanil, intranasal ketamine and intranasal CT001.

Secondary Outcome Measures
NameTimeMethod
Time to meaningful pain relief0-180 min

Time when participants feel that the pain relief becomes meaningful to them

Maximum Pain intensity difference (PIDmax)0-180 min
Time to rescue medication0-180 min
Sum of pain intensity differences at 30 min0-30 min

Derived from pain intensity scores measured on the Numerical Rating Scale (0-10, 0= no pain, 10= worst possible

Mean pain intensity difference (PID) from baseline at rest0-180 min
Median time to a request for rescue medication0-180 min
Rescue medication0-180 min

Number of participants receiving rescue medication

Sum of pain intensity differences at 90 min0-90 min

Derived from pain intensity scores measured on the Numerical Rating Scale (0-10, 0= no pain, 10= worst possible

Time to perceptible pain relief0-180 min

Time when participants feel that the pain relief becomes meaningful to them

Number of patients who are considered a responder/non-responder, 30%0-30 min

Number of participants with at least 30% reduction in pain intensity score compared to baseline

Number of patients who are considered a responder/non-responder, 50%0-30 min

Participants with at least at least 50% reduction in pain intensity score compared to baseline

Ramsay sedation score0-179 min

Change from baseline in Ramsay sedation score (1= agitated, anxious, restless, 6= unarousable)

Mean pain intensity difference (PID) from baseline on jaw movement0-181 min

Trial Locations

Locations (1)

DanTrials

🇩🇰

Copenhagen, NV, Denmark

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