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Study of CP-383 in Patients With Advanced or Metastatic Solid Tumors

Phase 1
Not yet recruiting
Conditions
Solid Tumor Malignancies
Colorectal Carcinoma
Small Cell Lung Cancer ( SCLC )
Head and Neck (HNSCC)
Bladder Cancer
Non-Small Cell Lung Cancer
Pancreatic Cancer, Advanced or Metastatic
Interventions
Registration Number
NCT07030257
Lead Sponsor
Tasca Therapeutics
Brief Summary

The goal of this clinical trial is to learn if an investigational drug CP-383 works to treat advanced cancer. It will also learn about the safety of CP-383. The main questions if aims to answer are:

* Does CP-383 slow or stop the growth of cancer in patients with advanced cancer

* What medical problems do participants have when taking CP-383 Researchers will test CP-383 in all kinds of cancers at various dose levels to determine what the best dose is to study further. Researchers will also see if certain cancers that have gene mutations respond better to CP-383

Participants will:

* Take CP-383 every day by mouth until the researcher learns whether CP-383 is helping slow or reduce the cancer growth

* Visit the clinic weekly for the first 6 weeks for checkups and tests

* Visit the clinic every 3 weeks thereafter for checkups and tests

Detailed Description

Not available

Recruitment & Eligibility

Status
NOT_YET_RECRUITING
Sex
All
Target Recruitment
150
Inclusion Criteria
  • Measurable or non measurable cancer that the research can assess for changes

  • Not eligible or able to take existing standard therapies for cancer

  • Availability of a part of a tumor for laboratory testing or willing to have a safe biopsy taken from a tumor

  • Diagnosed with locally advanced, recurrent or metastatic incurable disease

  • Part 1: any solid tumor (with the exception of brain cancer) that has progressed, standard therapy is no longer or has not helped the cancer, or is too toxic and for whom a clinical trial is an option for continued treatment

  • Part 1: specific advanced, metastatic tumor types will also be enrolled: colorectal cancer, small cell lung cancer, head and neck cancer, non-small cell lung cancer, pancreatic cancer, bladder cancer - some of these will have a specific gene mutation in the cancer

  • Part 1: selected solid tumor cancer types (with the exception of brain cancers) that have a specific gene mutation in the cancer

  • Part 2: specific advanced, metastatic tumor types will also be enrolled: colorectal cancer, small cell lung cancer, head and neck cancer - some of these will have a specific gene mutation in the cancer

    _ Part 2: selected solid tumor cancer types (with the exception of brain cancers) that have a specific gene mutation in the cancer

  • Adequate blood and urine lab tests

  • Women and men of childbearing potential with adequate contraception

  • Provides written informed consent

  • Willing to comply with the requirements of the protocol

Exclusion Criteria
  • Inability to swallow pills
  • Known history of HIV, HCV, HBV unless cured, controlled with undetectable viral load
  • Active tumor in the brain
  • Clinically significant liver disease
  • Significant gastrointestinal diseases
  • History of other cancer within past 5 years with certain exceptions for cancers that are likely cured
  • Significant cardiac disease
  • Other diseases that are not well controlled that could make taking the drug unsafe
  • pregnant or lactating females
  • Exposure to certain anti-cancer or other drugs within a certain period before the start of study drug

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Dose Level 1CP-383CP-383, single daily oral capsule, 0.8 mg
Expansion Arm 3CP-383Expansion in selected tumor type at recommended Phase 2 Dose of CP-383
Dose Level 2CP-383CP-383, single daily oral capsule, 1.6 mg
Dose Level 4CP-383CP-383, single daily oral capsule, 5.0 mg
Dose Level 6CP-383CP-383, single daily oral capsule, 12 mg
Expansion Arm 4CP-383Expansion in selected tumor type at recommended Phase 2 Dose of CP-383
Dose Level 3CP-383CP-383, single daily oral capsule, 3.0 mg
Dose Level 5CP-383CP-383, single daily oral capsule, 8.0 mg
Expansion Arm 1CP-383Expansion in selected tumor type at recommended Phase 2 Dose of CP-383
Expansion Arm 2CP-383Expansion in selected tumor type at recommended Phase 2 Dose of CP-383
Primary Outcome Measures
NameTimeMethod
Part 1: Determine the maximum tolerated dose (MTD)21 days

Determine the MTD of CP-383 in subjects with advanced solid tumors

Part 2: Evaluate the efficacy of CP-383 at the recommended phase 2 dose in selected tumor typesFrom enrollment through study completion, an average of 1 year

Objective response rate assessed by the investigator according to RECIST

Secondary Outcome Measures
NameTimeMethod
Part 2: Evaluate safety and tolerability of CP-383 at the recommended Phase 2 dose in selected tumor typesFrom enrollment through study completion, an average of 1 year

Incidence of AEs and changes in test results

Part 2: Evaluate the efficacy of CP-383 at the recommended phase 2 dose in selected tumor typesFrom enrollment through study completion, an average of 1 year

Evaluate overall survival

Part 1: Determine the pharmacokinetics parameters of CP-383From enrollment through study completion, an average of 1 year

Assess standard PK parameters including AUC

Part 1: Assess safety and tolerability of CP-383 in participants with advanced solid tumorsFrom enrollment through study completion, an average of 1 year

Incidence and severity of Adverse events and changes in test results

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