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A Clinical Trial To Evaluate PF-05089771 On Its Own And As An Add-On Therapy To Pregabalin (Lyrica) For The Treatment Of Pain Due To Diabetic Peripheral Neuropathy (DPN)

Phase 2
Completed
Conditions
Diabetic Neuropathy, Painful
Interventions
Drug: Matched placebo for PF-05089771 150 mg and pregabalin 300 mg
Registration Number
NCT02215252
Lead Sponsor
Pfizer
Brief Summary

The purpose of this study is to evaluate the efficacy and safety of PF-05089771 as a monotherapy and as an add-on to pregabalin for the treatment of painful diabetic peripheral neuropathy (DPN)

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
141
Inclusion Criteria
  • Men and women aged 18 years to 80 years.
  • Diagnosis of Type 2 diabetes mellitlus (T2DM) with current glycosylated hemoglobin A1c (HbA1c) levels of ≤ 11% at Screening and on a stable antidiabetic medication regimen for at least 30 days prior to randomization.
  • Presence of ongoing pain due to DPN for at least 6 months.
  • Willing to discontinue protocol-specified prohibited pain medications for DPN throughout the duration of the study.
Exclusion Criteria
  • Painful neuropathies or painful conditions other than DPN that may confound evaluation of pain due to DPN during the study.
  • Subjects who have failed previously on pregabalin (at the recommended label dose and for adequate duration) due to lack of efficacy.
  • Subjects with any clinically significant medical or psychiatric conditions or clinically significant laboratory test abnormalities.
  • Pregnant women, lactating mothers, men with partners currently pregnant, women suspected of being pregnant, and women who wish to be pregnant during the course of the clinical study.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PF-05089771 + PregabalinPF-05089771 150 mg + Pregabalin 300 mg-
PF-05089771PF-05089771 150 mg-
PregabalinPregabalin 300 mg-
PlaceboMatched placebo for PF-05089771 150 mg and pregabalin 300 mg-
Primary Outcome Measures
NameTimeMethod
Daily Pain Numeric Rating Scale (NRS)Baseline, Week 1, Week 2, Week 3 and Week 4

The endpoint average pain score, based on the mean of the last 7 days' daily pain numeric rating scale (NRS) scores at (NRS is an 11-point scale where 0 = no pain and 10 = worst possible pain) from the daily pain diaries while receiving study medication during the treatment period.

Secondary Outcome Measures
NameTimeMethod
Responder Rate Based on a 30% Improvement in Mean Pain Response Using the Daily Pain NRS ScoreBaseline, Week 1, Week 2, Week 3 and Week 4

Percentage of participants that received ≥30% improvement from baseline in mean pain response (from the daily pain diary).

Neuropathic Pain Symptom Inventory (NPSI) - Total ScoreBaseline, Week 2 and Week 4

Participant rated questionnaire to evaluate different symptoms of neuropathic pain (dimensions: burning \[superficial\] spontaneous pain, pressing \[deep\] spontaneous pain, paroxysmal pain, evoked pain, and paresthesia/dyesthesia \[P/D\]) including 10 descriptors quantified on a 0 (no symptoms) to 10 (worst symptoms imaginable) and 2 temporal items assessing duration of spontaneous ongoing and paroxysmal pain. A score in each dimension and also a total score (from 0-100) is generated using data from the questionnaire. Higher score indicates a greater intensity of pain.

Responder Rate Based on a 50% Improvement in Mean Pain Response Using the Daily Pain NRS ScoreBaseline, Week 1, Week 2, Week 3, and Week 4

Percentage of participants that received ≥50% improvement from baseline in mean pain response (from the daily pain diary).

Daily Sleep Interference Scale Score (DSIS).Baseline, Week 1, Week 2, Week 3 and Week 4

Participant rated 11-point Likert scale ranging from 0 (pain does not interfere with sleep) to 10 (pain completely interferes with sleep) during past 24-hour period. Higher score indicates a greater level of sleep disturbance. Self-assessment performed daily on awakening prior to taking study medication. This score was measured as a weekly average.

Total Amount of Rescue Medication Per WeekBaseline, Week 1, Week 2, Week 3, and Week 4

Total amount of rescue medication participants take per week

Number of Days Participants Take Rescue MedicationBaseline, Week 1, Week 2, Week 3 and Week 4

Number of days participants take rescue medication per week.

Neuropathic Pain Symptom Inventory (NPSI) - Burning (Superficial) Spontaneous PainBaseline, Week 2, and Week 4

Participants rated questionnaire to evaluate different symptoms of neuropathic pain (dimensions: burning \[superficial\] spontaneous pain, pressing \[deep\] spontaneous pain, paroxysmal pain, evoked pain, and paresthesia/dyesthesia \[P/D\]) including 10 descriptors quantified on a 0 (no symptoms) to 10 (worst symptoms imaginable) and 2 temporal items assessing duration of spontaneous ongoing and paroxysmal pain. A score in each dimension and also a total score (from 0-100) is generated using data from the questionnaire. Higher score indicates a greater intensity of pain.

Fasted Total Cholesterol ValuesBaseline, Week 2 and Week 4

Percentage Change from Baseline in Fasted Total Cholesterol values

Neuropathic Pain Symptom Inventory (NPSI) - Pressing (Deep) Spontaneous PainBaseline, Week 2 and Week 4

Participant rated questionnaire to evaluate different symptoms of neuropathic pain (dimensions: burning \[superficial\] spontaneous pain, pressing \[deep\] spontaneous pain, paroxysmal pain, evoked pain, and paresthesia/dyesthesia \[P/D\]) including 10 descriptors quantified on a 0 (no symptoms) to 10 (worst symptoms imaginable) and 2 temporal items assessing duration of spontaneous ongoing and paroxysmal pain. A score in each dimension and also a total score (from 0-100) is generated using data from the questionnaire. Higher score indicates a greater intensity of pain.

Neuropathic Pain Symptom Inventory (NPSI) - Evoked PainBaseline, Week 2 and Week 4

Participant rated questionnaire to evaluate different symptoms of neuropathic pain (dimensions: burning \[superficial\] spontaneous pain, pressing \[deep\] spontaneous pain, paroxysmal pain, evoked pain, and paresthesia/dyesthesia \[P/D\]) including 10 descriptors quantified on a 0 (no symptoms) to 10 (worst symptoms imaginable) and 2 temporal items assessing duration of spontaneous ongoing and paroxysmal pain. A score in each dimension and also a total score (from 0-100) is generated using data from the questionnaire. Higher score indicates a greater intensity of pain.

Patient's Global Impression of Change Score (PGIC).Baseline, Week 2, and Week 4

Participant rated instrument to measure participant's change in overall status on a 7-point scale; range from 1 (very much improved) to 7 (very much worse) at week 4. The PGIC was combined to produce a 3-point scale, "Improved", "No Change" and "Worse".

Number of Participants With Laboratory Test Values of Potential Clinical ImportanceScreening, Day 1, Day 15 and Day 29

The total number of participants with laboratory test abnormalities (without regard to baseline abnormality) was assessed. Clinical laboratory tests included hematology, chemistry, urinalysis and some other tests.

Fasted Low Density Lipoprotein (LDL) CholesterolBaseline, Week 2 and Week 4

Percentage Change from Baseline in LDL cholesterol Friedewald by PEG

Neuropathic Pain Symptom Inventory (NPSI) - Paroxysmal PainBaseline, Week 2, and Week 4

Participant rated questionnaire to evaluate different symptoms of neuropathic pain (dimensions: burning \[superficial\] spontaneous pain, pressing \[deep\] spontaneous pain, paroxysmal pain, evoked pain, and paresthesia/dyesthesia \[P/D\]) including 10 descriptors quantified on a 0 (no symptoms) to 10 (worst symptoms imaginable) and 2 temporal items assessing duration of spontaneous ongoing and paroxysmal pain. A score in each dimension and also a total score (from 0-100) is generated using data from the questionnaire. Higher score indicates a greater intensity of pain.

Neuropathic Pain Symptom Inventory (NPSI) - Paresthesia/DysethesiaBaseline, Week 2 and Week 4

Participant rated questionnaire to evaluate different symptoms of neuropathic pain (dimensions: burning \[superficial\] spontaneous pain, pressing \[deep\] spontaneous pain, paroxysmal pain, evoked pain, and paresthesia/dyesthesia \[P/D\]) including 10 descriptors quantified on a 0 (no symptoms) to 10 (worst symptoms imaginable) and 2 temporal items assessing duration of spontaneous ongoing and paroxysmal pain. A score in each dimension and also a total score (from 0-100) is generated using data from the questionnaire. Higher score indicates a greater intensity of pain.

Number of Participants With Treatment-Emergent Adverse Events (TEAEs), Serious Adverse Events (SAEs), and Withdrawals Due to Adverse Events (AEs)Screening to Day 36, and Day 64

An AE was any untoward medical occurrence attributed to study drug in a participant who received study drug. An SAE was an AE resulting in any of the following outcomes or deemed significant for any other reason: death; life threatening (immediate risk of death); initial or prolonged inpatient hospitalization; persistent or significant disability/incapacity; resulted in congenital anomaly/birth defect.

Plasma Concentration of PF-05089771Baseline, Week 2 and Week 4

All participants in this group were analysed. Only plasma PK concentration of PF-05089771 was analysed.

Trial Locations

Locations (28)

Pulmonary Associates of Brandon (PAB)

🇺🇸

Brandon, Florida, United States

Beacon Clinical Research, LLC

🇺🇸

Quincy, Massachusetts, United States

The Medical Research Network, LLC

🇺🇸

New York, New York, United States

Clinical Physiology Associates

🇺🇸

Fort Myers, Florida, United States

MD Clinical

🇺🇸

Hallandale, Florida, United States

Family Care Specialists

🇺🇸

Ocala, Florida, United States

Renstar Medical Research

🇺🇸

Ocala, Florida, United States

Oviedo Medical Research, LLC

🇺🇸

Oviedo, Florida, United States

Clinical Research Advantage, Inc

🇺🇸

Evansville, Indiana, United States

Meridien Research

🇺🇸

Tampa, Florida, United States

Novex Clinical Research, LLC

🇺🇸

New Bedford, Massachusetts, United States

Metabolic Research Institute, Inc

🇺🇸

West Palm Beach, Florida, United States

Columbus Regional Research Institute

🇺🇸

Columbus, Georgia, United States

Arizona Research Center

🇺🇸

Phoenix, Arizona, United States

Brigham and Women's Hospital

🇺🇸

Boston, Massachusetts, United States

Clinical Research Consortium

🇺🇸

Las Vegas, Nevada, United States

Nerve and Muscle Center of Texas

🇺🇸

Houston, Texas, United States

Clinical Research Consortium Arizona

🇺🇸

Phoenix, Arizona, United States

Neuro-Pain Medical Center

🇺🇸

Fresno, California, United States

PAB Clinical Research

🇺🇸

Brandon, Florida, United States

Internal Medicine Associates

🇺🇸

Tullahoma, Tennessee, United States

Trinity Clinical Research, LLC

🇺🇸

Tullahoma, Tennessee, United States

New Phase Research and Development

🇺🇸

Knoxville, Tennessee, United States

Michigan Head Pain and Neurological Institute

🇺🇸

Ann Arbor, Michigan, United States

National Clinical Research - Norfolk, Inc

🇺🇸

Norfolk, Virginia, United States

KRK Medical Research

🇺🇸

Arlington, Texas, United States

Rainier Clinical Research Center, Inc

🇺🇸

Renton, Washington, United States

Eastern Virginia Medical School

🇺🇸

Norfolk, Virginia, United States

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