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A Study to Assess the Effect of Famotidine on the Drug Levels of Afimetoran in Healthy Participants

Phase 1
Recruiting
Conditions
Healthy Volunteers
Interventions
Registration Number
NCT05866627
Lead Sponsor
Bristol-Myers Squibb
Brief Summary

The purpose of this study is to confirm there is no significant effect of gastric pH changes of famotidine on the drug levels of afimetoran in healthy participants.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
76
Inclusion Criteria
  • Weight ≥ 50 kilograms (kg), at screening and first admission, and body mass index between 18.0 kilogram per square meter (kg/m^2) and 32.0 kg/m^2, inclusive, at screening.
  • A negative QuantiFERON-TB Gold test result at screening or documentation of a negative result within 3 months before screening.
  • Normal renal function at screening as evidenced by an estimated glomerular filtration rate (eGFR) ≥ 80 milliliter per minute (mL/min)/1.732 m^2 calculated with the Chronic Kidney Disease Epidemiology Collaboration formula.
Exclusion Criteria
  • Any significant acute or chronic medical illness.
  • Current or recent (within 3 months of study drug administration) gastrointestinal (GI) disease that could impact upon the absorption of study treatment.
  • GI surgery, including cholecystectomy, that could impact upon the absorption of study treatment, at the investigator's discretion.

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Afimetoran, followed by famotidine + afimetoranAfimetoran-
Famotidine + afimetoran, followed by afimetoranFamotidine-
Famotidine + afimetoran, followed by afimetoranAfimetoran-
AfimetoranAfimetoran-
Afimetoran, followed by famotidine + afimetoranFamotidine-
Famotidine, followed by afimetoranFamotidine-
Famotidine, followed by afimetoranAfimetoran-
Primary Outcome Measures
NameTimeMethod
Time to attain maximum observed plasma concentration (Tmax)Up to 20 Days
Maximum observed plasma concentration (Cmax)Up to 20 Days
Area under the plasma concentration-time curve from time zero to time of the last quantifiable concentration (AUC[0-T])Up to 20 Days
Secondary Outcome Measures
NameTimeMethod
Number of participants with clinical laboratory abnormalitiesUp to 52 Days
Number of participants with vital sign abnormalitiesUp to 52 Days
Number of participants with electrocardiogram (ECG) abnormalitiesUp to 52 Days
Number of participants with adverse events (AEs)Up to 52 Days

Trial Locations

Locations (1)

Quotient Sciences

🇬🇧

Nottingham, Nottinghamshire, United Kingdom

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