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Controlled, 12-Week Study of Albuterol HFA Versus the Active Control, Proventil(R)-HFA in Asthmatic Patients

Phase 3
Terminated
Conditions
Asthma
Interventions
Registration Number
NCT00635505
Lead Sponsor
Amphastar Pharmaceuticals, Inc.
Brief Summary

This 12-week clinical study evaluates the safety and efficacy of Albuterol Sulfate HFA Inhalation Aerosol (Albuterol-HFA, or: A004), Armstrong's proposed HFA formulation of metered dose inhaler (MDI) of Albuterol (Treatment T), in comparison with:

1. Placebo control: (HFA propellant only, Treatment P); and

2. Active control: 3M/Key's Proventil-HFA (Treatment R).

The treatments will be given as self-administered oral inhalations in adult and adolescent patients with mild-to-moderate asthma, for 12-weeks. Dosing regimen throughout the 12-week study is two actuations four times daily (QID).

Detailed Description

This is a randomized, parallel, multicenter, 12-week study in adolescent and adult patients with mild-to-moderate asthma, to evaluate the efficacy and safety of Armstrong's Albuterol-HFA MDI, in comparison to a Placebo Control and an Active Control of Proventil-HFA. While Albuterol-HFA (Treatment T) and Placebo (Treatment P) will be double-blinded to both the subjects and investigational staff, the active comparator drug, Proventil-HFA (Treatment R), can only be evaluator-blinded, due to: (1) its physical appearance differing from that of the T and P devices; and (2) unavailability of a Proventil-HFA placebo which would otherwise be used for a double-dummy design. All study medications will have the canisters and all product-identifying text or graphics (e.g., molded text on actuator) masked so that the treatments cannot be identified. No subject in any study arm will be given any information that could reveal the nature of the treatment given. All study subjects will be instructed not to reveal or discuss the study medications to the study staff or other subjects. The designated study evaluator(s), who conduct the clinical visits and safety and efficacy evaluations and perform the data recording and transcription, will be blinded to the study medications.

All subjects will be screened for enrollment, and will be randomized into the following three treatment groups in a double-blinded (for Treatments T and P) or evaluator-blinded (for Treatment R) manner:

Treatment T (Albuterol-HFA, N=200): 216 mcg albuterol sulfate (equivalent to 180 mcg albuterol base), QID; Treatment R (Proventil-HFA, N=50): 216 mcg albuterol sulfate (equivalent to 180 mcg albuterol base), QID; Treatment P (Placebo-HFA, N=50): two actuations of placebo, QID.

Randomization is achieved with blocks of six (6), with four (4) patients receiving Albuterol-HFA for every one (1) patient receiving Proventil-HFA and every one (1) receiving the Placebo-HFA. At each Clinical Visit that takes place every 3 weeks, the double-blinded (T, P) or evaluator-blinded (R) study drugs will be distributed in resealable masking pouches to the subjects of each arm.

An additional aim of the study is to evaluate the effect of weekly cleaning on the Albuterol-HFA MDI device clinical performance throughout the four, 3-week life-of-device treatment cycles, in conformance with the FDA's specific requirements.

Arms:

All subjects will be screened for enrollment, and will be randomized into the following three treatment groups in a double-blinded (for Treatments T and P) or evaluator-blinded (for Treatment R) manner:

Treatment T (Albuterol-HFA, N=200): 216 mcg albuterol sulfate (equivalent to 180 mcg albuterol base), QID; Treatment R (Proventil-HFA, N=50): 216 mcg albuterol sulfate (equivalent to 180 mcg albuterol base), QID; Treatment P (Placebo-HFA, N=50): two actuations of placebo, QID.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
300
Inclusion Criteria
  • Male and female asthma patients aged 12 - 75 years, in general good health.
  • A documented history of mild to moderate asthma, for at-least 6-months prior to Screening, requiring inhaled B2-adrenergic agonists, with or without orally inhaled corticosteroids, for asthma treatment.
  • Satisfying criteria of asthma stability, defined as no asthma-related hospitalization or emergency visits, and no significant changes in asthma therapy, over 4 weeks prior to Screening (with exception for switching from long- to short-acting B2-agonists).
  • Can tolerate withholding treatment with inhaled bronchodilators and other allowed medications for the minimum washout periods indicated in Appendix II prior to the Screening Baseline FEV1 testing.
  • Having a Screening Baseline FEV1 test that falls within 50-90% of the predicted values.
  • Airway Reversibility PFT at screening should demonstrate a greater than 12% increase in FEV1 at 30 minutes of inhaling 2 actuations of Ventolin-HFA (180 mcg albuterol base).
  • Demonstrating satisfactory techniques in the use of metered-dose inhaler (MDIs) and a hand held peak flow meter.
  • Female patients of child-bearing potential being non-pregnant and non-lactating at Screening and throughout the study, and using an acceptable method of contraception during the study.
  • Has properly consented to participate in this study.
Exclusion Criteria
  • Male and female asthma patients aged 12 - 75 years, in general good health.
  • A documented history of mild to moderate asthma, for at-least 6-months prior to Screening, requiring inhaled B2-adrenergic agonists, with or without orally inhaled corticosteroids, for asthma treatment.
  • Satisfying criteria of asthma stability, defined as no asthma-related hospitalization or emergency visits, and no significant changes in asthma therapy, over 4 weeks prior to Screening (with exception for switching from long- to short-acting B2-agonists).
  • Can tolerate withholding treatment with inhaled bronchodilators and other allowed medications for the minimum washout periods indicated in Appendix II prior to the Screening Baseline FEV1 testing.
  • Having a Screening Baseline FEV1 test that falls within 50-90% of the predicted values.
  • Airway Reversibility PFT at screening should demonstrate a greater than12% increase in FEV1 at 30 minutes of inhaling 2 actuations of Ventolin-HFA (180 mcg albuterol base).
  • Demonstrating satisfactory techniques in the use of metered-dose inhaler (MDIs) and a hand held peak flow meter.
  • Female patients of child-bearing potential being non-pregnant and non-lactating at Screening and throughout the study, and using an acceptable method of contraception during the study.
  • Has properly consented to participate in this study.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Talbuterol HFA (Armstrong's)albuterol HFA 180 mcg QID
Ralbuterol HFA (Proventil HFA)180 mcg QID 12 weeks
PHFA placebo2 actuations QID 12 weeks or until use of rescue drug
Primary Outcome Measures
NameTimeMethod
The primary endpoint is the bronchodilator effect expressed as the mean area under the curve (AUC) of FEV1 (% change from Same-Day Baseline FEV1) versus time.Concurent with each visit
Secondary Outcome Measures
NameTimeMethod
The comparative analysis of AUC of FEV1 (% change from the Same-Day Baseline) versus time, for bronchodilator effect (between Albuterol-HFA and Proventil-HFA).End of Study
AUC of FEV1-time curve (changes of actual volumes from the Same-Day Baseline).End of Study
Time to onset of bronchodilator effect, determined by linear interpolation as the time point where FEV1 first reaches 12% over Same-Day Baseline.End of Study
The peak bronchodilator response, defined as the maximum FEV1 (% change from Same-Day Baseline) post-dose.end of study
The time to peak FEV1 effect, measured as the time point of peak response, as defined (4) above.End of Study
Duration of bronchodilator effect, defined as the total length of time when FEV1 is maintained 12% above the respective Same-Day Baseline values (time points calculated with linear interpolation).Concurrent with each visit
Percentage of positive responders including those whose FEV1 exceed the Same-Day Baseline by 12% within 30 minutes post-dose (quick responders), and during the entire 6 hr post-dose (overall responders).Concurrent with visit
Number of inhalations of the rescue inhalers taken.Concurrent with each visit
Global assessment of Overall Asthma Control Scores by investigators.End of Study
Total daytime asthma symptom scores.End of Study
Nighttime sleep disturbance scores.End of Study
Morning pre-dose Peak Expiratory Flow Rate (PEF).Concurrent with each visit
The clinical performances of the Albuterol-HFA MDI at the representative first, middle and last one third of the usable life stage, are compared with each other, and are also compared to those of the active control, Proventil-HFA.End of Study
The in vitro performance of the Albuterol-HFA MDI will be evaluated.Concurrent with each visit
Vital signs (SBP/DBP, and heart rate) will be monitored at Clinical Visit 1, 3 and 5, at baseline (within 30 minutes prior to dosing), and 90+/-15 min, and 360+/-30 min, post-dose.concurrent with study visits as noted
A 12-lead ECG (for HR, QT and QTc intervals) will be recorded at Screening Visit, and at baseline (within 30 min) pre-dose and at 90+/-15 min post-dose (predicted time of peak effect).Clinical Visits 1 and 5
Data for CBC, blood chemistry panel (8-hr fasted), and urinalysis.Screening and end-of-study
Study compliance and diaries will be reviewedat all cliniical visits
Concomitant medications will be reviewed and recordedeach study visit
Adverse events/side effects whether observed by investigators or reported by subjects, will be documented, evaluated, followed up, and treated if deemed necessary.concurrent with each study visit

Trial Locations

Locations (41)

Pulmonary Associates of Mobile, PC

🇺🇸

Mobile, Alabama, United States

MEDEX Healthcare Research, Inc.

🇺🇸

St. Louis, Missouri, United States

The Clinical Research Center, LLC

🇺🇸

St. Louis, Missouri, United States

Clinical Research Institute of Southern Oregon

🇺🇸

Medford, Oregon, United States

Allergy and Clinical Immunology Associates

🇺🇸

Pittsburgh, Pennsylvania, United States

Bensch Research Associates

🇺🇸

Stockton, California, United States

Allergy Asthma and Dermatology Research

🇺🇸

Lake Oswego, Oregon, United States

Allergy and Asthma Associates of Houston

🇺🇸

Houston, Texas, United States

Asthma, Inc.

🇺🇸

Seattle, Washington, United States

Clinical Trials of North Houston

🇺🇸

Houston, Texas, United States

Allergy Associates Medical Group

🇺🇸

San Diego, California, United States

CHOC PSF, AMC, Divison AA and I

🇺🇸

Orange, California, United States

Family Allergy and Asthma Research Institute

🇺🇸

Louisville, Kentucky, United States

Virginia Adult and Pediatric Allergy and Asthma, PC

🇺🇸

Richmond, Virginia, United States

Colorado Allergy and Asthma Centers

🇺🇸

Lakewood, Colorado, United States

Rocky Mountain center for Clinical Research

🇺🇸

Wheatridge, Colorado, United States

Park Nicollet Institute

🇺🇸

Minneapolis, Minnesota, United States

Allergy Associates Research Center

🇺🇸

Portland, Oregon, United States

Allergy Asthma & Respiratory Care Medical Center

🇺🇸

Long Beach, California, United States

Allergy & Asthma Care Center

🇺🇸

Long Beach, California, United States

Allergy & Asthma Specialists Medical Group

🇺🇸

Huntington Beach, California, United States

Clinical Trials of Orange County

🇺🇸

Orange, California, United States

Southern California Research

🇺🇸

Mission Viejo, California, United States

Allergy & Asthma Associates of Santa Clara Valley Research Centere

🇺🇸

San Jose, California, United States

Peninsula Research Associates

🇺🇸

Rolling Hills Estates, California, United States

Allergy and Asthma Care of Florida

🇺🇸

Ocala, Florida, United States

Atlanta Allergy and Asthma Clinic

🇺🇸

Woodstock, Georgia, United States

Northeast Medical Research Group

🇺🇸

N. Dartmouth, Massachusetts, United States

Clinical Research Group of Montana

🇺🇸

Bozeman, Montana, United States

Asthma and Allergy Center, PC

🇺🇸

Papillion, Nebraska, United States

New Horizons Clinical Research

🇺🇸

Cincinnati, Ohio, United States

Montant Medical Research

🇺🇸

Missoula, Montana, United States

Integrated Medical Research

🇺🇸

Ashland, Oregon, United States

Toledo Center for Clinical Research

🇺🇸

Sylvania, Ohio, United States

Allergy & Asthma Research Group

🇺🇸

Eugene, Oregon, United States

Pharmaceutical Research & Consulting, Inc.

🇺🇸

Dallas, Texas, United States

Kerrville Allergy and Asthma Associates

🇺🇸

Kerrville, Texas, United States

Biogenics Research Institute

🇺🇸

San Antonio, Texas, United States

Sylvania Research Associates

🇺🇸

San Antonio, Texas, United States

Waterbury Pulmonary Research

🇺🇸

Waterbury, Connecticut, United States

Brandon-Valrico Center for Allergy and Astham Research,LLC

🇺🇸

Valrico, Florida, United States

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