MedPath

Trial of Rituximab and Mycophenolate Mofetil Without Oral Steroids for Lupus Nephritis

Phase 3
Terminated
Conditions
Systemic Lupus Erythematosus, Lupus Nephritis
Interventions
Registration Number
NCT01773616
Lead Sponsor
Imperial College London
Brief Summary

The treatment of the multisystem autoimmune disease systemic lupus erythematosus (SLE) remains a challenge, particularly when there is renal involvement (lupus nephritis). For the last 60 years corticosteroids have been the backbone of the treatment of lupus nephritis but they are associated with significant toxicity.

Although randomized placebo controlled trials of Rituximab in non-renal lupus and lupus nephritis did not meet their primary end-points, there is accumulating data that suggests that B cell depletion with Rituximab may be efficacious in lupus disease refractory to conventional therapy. Furthermore, our pilot data suggests that the addition of Rituximab to mycophenolate mofetil (MMF) without oral steroids is at least as effective at inducing a renal response as the standard of care therapy comprising MMF and high dose oral corticosteroids.

RITUXILUP is a proof of concept, open labeled, randomized, controlled, multicentre trial that aims to demonstrate whether the addition of Rituximab to MMF therapy is useful in treating a new flare of lupus nephritis and whether it has a long lasting steroid-sparing, beneficial effect with equal efficacy and greater safety than a conventional regimen of MMF and oral prednisolone. If successful, this trial has the potential to dramatically change the management of lupus nephritis.

Detailed Description

TRIAL SUMMARY

TITLE RITUXILUP - An open label randomised multicentre controlled trial of RITUXImab and mycophenolate mofetil (MMF) without oral steroids for the treatment of LUPus nephritis

OBJECTIVES

1. Is the combination of Rituximab, Methyl prednisolone and MMF as effective in treating lupus nephritis as Methyl prednisolone, oral steroids and MMF?

2. Does the omission of oral steroids increase the safety of the treatment regimen?

DESIGN This is a 1:1 randomised, international open label, controlled phase III multicentre trial

SAMPLE SIZE A total of 252 patients: 126 patients in each arm (As of April 2017 decided 25 patients will be maximum recruited following decision to close the study early)

ELIGIBILITY Children (12 years and above) and adults with lupus nephritis ISN/RPS Class III A or A/C, Class IV-G A or A/C, Class IV-S A or A/C, and/or Class V with a urine protein/creatinine ratio (PCR) ≥ 100mg/mmol.

TREATMENT

1. Experimental group - Rituximab, IV methyl prednisolone and mycophenolate mofetil

2. Control group - oral prednisolone, IV methyl prednisolone and mycophenolate mofetil.

PRIMARY OUTCOME The primary outcome is to demonstrate non-inferiority of the Rituximab arm in comparison to the control arm in the proportion of patients achieving complete renal response (CR) at week 52 without the need for steroid prescription.

SECONDARY OUTCOMES

Safety outcomes:

* Serious Infectious Episodes

* Serious Adverse Events

* Evidence of metabolic abnormalities particularly new onset diabetes

Disease control over time:

* Proportion of patients achieving Partial Response (PR)

* Time to stable CR

* Time to PR

* Proportion of patients in PR who achieve histological remission in those who have a repeat biopsy as part of local standard of care

* Proportion of patients with renal or extra flare

* Cumulative steroid exposure

* Deviation from the steroid taper in the steroid arm and/or introduction of steroids in the steroid-free arm

* Proportion of patients achieving a response as defined by the SLE Responder Index (SRI) at week 52 and annually thereafter as defined by:

* a \>4 point reduction in SELENA-SLEDAI score;

* no new BILAG A organ domain score;

* no more than I new BILAG B score;

* no worsening in physician's global assessment (PGA) by \>10%;

* must not have received non-protocol treatment.

* Proportion of patients achieving a response as defined by the BILAG-based Composite Lupus Assessment (BICLA) at week 52 and annually thereafter as defined by: BILAG-2004 improvement (BILAG A to B/C/D, BILAG B to C/D and no BILAG worsening, no deterioration in SLEDAI total score, no worsening in physician's global assessment (PGA) by \>10% and must not have received non-protocol treatment.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
24
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Oral prednisoloneOral prednisoloneOral prednisolone, methyl prednisolone and mycophenolate mofetil
Oral prednisoloneMethyl prednisoloneOral prednisolone, methyl prednisolone and mycophenolate mofetil
RituximabMethyl prednisoloneRituximab, methyl prednisolone and mycophenolate mofetil
RituximabMycophenolate mofetilRituximab, methyl prednisolone and mycophenolate mofetil
RituximabRituximabRituximab, methyl prednisolone and mycophenolate mofetil
Oral prednisoloneMycophenolate mofetilOral prednisolone, methyl prednisolone and mycophenolate mofetil
Primary Outcome Measures
NameTimeMethod
Complete renal response (CR) at week 52 without the need to prescribe oral steroids within 1 year1 year

The proportion of participants who achieve a complete renal response at week 52 without the need to prescribe oral steroids within 1 year, except for one course of maximum 30mg for a maximum of 14 days OR one intramuscular or intra-articular injection of steroids

Secondary Outcome Measures
NameTimeMethod
Mean time to stable CR and mean time to PR2 years
Metabolic abnormalities related to steroid exposure2 years
Mean time to renal flare in patients achieving CR and PR2 years
Proportion of patients achieving CR at 6, 18 and 24 months2 years
Proportion of patients with renal flare2 years

Flare is identified by:

i) Proteinuria \>50% increase ii) AND above 100mg/mmol for 2 visits iii) and / or in those with normal renal function and normal urinary sediment, a fall of \>20% in eGFR on 2 occasions Where possible flare should be proven by repeat renal biopsy.

Introduction of oral steroids in the B cell depleted patients2 years
Proportion of patients with only 1 or fewer BILAG 2004 Bs in any non-renal organ system at 1 year2 years
Serious Infectious Episodes, Serious Adverse Events and Adverse events2 years

4. Metabolic abnormalities related to steroid exposure: 5. Cumulative steroid exposure over 1 and 2 years 6. Introduction of oral steroids in the B cell depleted patients 7. Patients requiring \>10mg oral prednisolone at 1 year and 2 year

Cumulative steroid exposure over 1 and 2 years2 years
Patients requiring >10mg oral prednisolone at 1 year and 2 year2 years
Proportion of patients achieving PR at 6,12,8 and 24 months2 years

PR is defined as:

i) eGFR at baseline or \<20% decrease, ii) AND if not nephrotic at baseline (PCR\<300mg/mmol), 50% improvement in urine PCR iii) OR if nephrotic at baseline (PCR \>300mg/mmol), 50% improvement in urine PCR AND PCR \<300mg/mmol

Proportion of patients achieving normal serum C3,C4 and anti-dsDNA antibodies at week 522 years
Proportion of patients in PR who achieve histological remission as judged by absence of proliferative lesions and no new subendothelial or subepithelial deposits2 years

Trial Locations

Locations (11)

Royal Stoke Hospital, University Hospitals of North Midlands NHS Trust

🇬🇧

Stoke-on-Trent, United Kingdom

Hammersmith Hospital, Imperial College Healthcare NHS Trust

🇬🇧

London, United Kingdom

Churchill Hospital, Oxford University Hospitals NHS Trust

🇬🇧

Oxford, United Kingdom

Queen Elizabeth Hospital, University Hospitals Birmingham NHS Foundation Trust

🇬🇧

Birmingham, United Kingdom

Great Ormond Street Hospital for Children NHS Foundation Trust

🇬🇧

London, United Kingdom

King's College Hospital

🇬🇧

London, United Kingdom

Leicester General Hospital, University Hospitals of Leicester NHS Trust

🇬🇧

Leicester, United Kingdom

Chapel Allerton Hospital, The Leeds Teaching Hospitals NHS Trust

🇬🇧

Leeds, United Kingdom

Manchester Royal Infirmary, Central Manchester University Hospitals NHS Foundation Trust

🇬🇧

Manchester, United Kingdom

Royal Free London NHS Foundation Trust

🇬🇧

London, United Kingdom

Guy's and St Thomas' NHS Foundation Trust

🇬🇧

London, United Kingdom

© Copyright 2025. All Rights Reserved by MedPath