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Open Label Extension Study Evaluating Safety and Tolerability of AAB-003 (PF-05236812) in Subject With Mild to Moderate Alzheimer's Disease

Phase 1
Completed
Conditions
Alzheimer's Disease
Interventions
Drug: AAB-003 (PF-05236812)
Registration Number
NCT01369225
Lead Sponsor
Pfizer
Brief Summary

This is a study to evaluate the safety and tolerability of multiple doses of AAB-003 (PF-05236812) in patients with mild to moderate Alzheimer's Disease. Patients who complete study B2601001 may participate in this trial and receive AAB-003 (PF-05236812). Each patient's participation will last approximately 52 weeks.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
52
Inclusion Criteria
  • Successful completion of study B2601001
  • MMSE 12 or greater
Exclusion Criteria
  • Study B2601001 Week 32 MRI with clinically important exclusionary findings.
  • Experienced SAE, vasogenic edema and/or intracranial hemorrhage in study B2601001

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
0.5 mg/kg AAB-003AAB-003 (PF-05236812)-
1 mg/kg AAB-003AAB-003 (PF-05236812)-
2 mg/kg AAB-003AAB-003 (PF-05236812)-
4 mg/kg AAB-003AAB-003 (PF-05236812)-
8 mg/kg AAB-003AAB-003 (PF-05236812)-
Primary Outcome Measures
NameTimeMethod
Number of Participants With Treatment-Emergent Adverse Events (AEs) and Serious Adverse Events (SAEs)Baseline up to Week 52

An AE was any untoward medical occurrence in a participant who received study drug. An SAE was an AE resulting in any of the following outcomes or deemed significant for any other reason: death; initial or prolonged inpatient hospitalization; life-threatening experience (immediate risk of dying); persistent or significant disability/incapacity; congenital anomaly. Treatment-emergent are events between first dose of study drug and up to 28 days after last dose that were absent before treatment or that worsened relative to pre-treatment state. AEs included both SAEs and non-SAEs.

Number of Participants With Potentially Clinically Important Electrocardiogram (ECG) FindingsBaseline up to Week 52

ECG parameters included PR interval, QRS interval, and QT interval. Criteria for ECG changes meeting potential clinical concern included: PR interval \>=300 milliseconds (msec) or \>=25% increase when baseline is \>200 msec and \>=50% increase when baseline is less than or equal to (\<=)200 msec; QRS interval \>=200 msec or \>=50% increase from baseline when baseline is less than or equal to 100 msec and \>=25% increase when baseline is \>100 msec; and QTcF \>=450 msec or \>=30 msec increase.

Number of Participants With Abnormal Physical Examination FindingsBaseline up to Week 52

A full physical examination consisted of an examination of the abdomen, genitourinary and cardiovascular systems, lungs, lymph nodes, mouth, musculoskeletal and neurological systems, skin, extremities, head, ears, eyes, nose, throat and thyroid gland. Criteria for abnormal physical findings was based on the investigator's discretion and any new physical examination findings were documented as AEs. Only sites with at least 1 participant abnormality are reported.

Number of Participants With Abnormal Neurological Examination FindingsBaseline up to Week 52

Neurological examinations were done to the extent needed to assess the subject for any potential changes in neurological status, as determined by the investigator. Examinations included level of consciousness, speech, cranial nerves, motor, sensory, coordination, gait, and tendon reflexes. Only tests with at least 1 participant abnormality are reported.

Number of Participants With Any New Magnetic Resonance Imaging (MRI) FindingsBaseline up to Week 52

Brain MRIs were collected to assess for potential drug-related changes that might have constituted a safety concern. Findings suggestive of either vasogenic edema or intracranial hemorrhage were to be reported as AEs of special circumstance.

Number of Participants With Laboratory Abnormalities Meeting the Criteria for Potential Clinical ConcernBaseline up to Week 52

The following laboratory parameters were analyzed: hematology (hemoglobin, hematocrit, red blood cell \[RBC\] count, RBC morphology, platelet count, white blood cell \[WBC\] count, total neutrophils, eosinophils, monocytes, basophils, lymphocytes); blood chemistry (blood urea nitrogen \[BUN\], creatinine, glucose, calcium, sodium, potassium, chloride, total bicarbonate, aspartate aminotransferase \[AST\], alanine aminotransferase \[ALT\], total bilirubin, alkaline phosphatase, uric acid, albumin, and total protein; urinalysis (pH, glucose, protein, blood, ketones, nitrites, leukocyte esterase, microscopy \[if urine dipstick was positive for blood, protein, nitrites or leukocyte esterase\]); others (coagulation panel, circulating immune complex, and complement activation).

Number of Participants With Potentially Clinically Important Vital Sign FindingsBaseline up to Week 52

Vital signs assessment included pulse rate and blood pressure. Criteria for vital sign values meeting potential clinical concern included: supine/sitting pulse rate \<40 or \>120 beats per minute (bpm); standing pulse rate \<40 or \>140 bpm; systolic blood pressure (SBP) of more than or equal to (\>=)30 millimeters of mercury (mm Hg) change from baseline in same posture or SBP \<90 mm Hg, diastolic blood pressure (DBP) \>=20 mmHg change from baseline in same posture or DBP \<50 mm Hg.

Number of Participants With Suicidal Ideation or Suicidal Behavior as Assessed by the Columbia-Suicide Severity Rating Scale (C-SSRS)Baseline up to Week 52

The C-SSRS captures the occurrence, severity, and frequency of suicide-related thoughts and behaviors during the assessment period. C-SSRS assesses whether participant experienced the following: completed suicide; suicide attempt; preparatory acts towards imminent suicidal behavior; suicidal ideation; self-injurious behavior, no suicidal intent. The results presented are the number of participants with completed suicide or non-fatal suicide events or behaviors. Worsening of suicidal ideation was an increase in severity of suicidal ideation from baseline.

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (21)

Borgess Research Institute

🇺🇸

Kalamazoo, Michigan, United States

MD Clinical

🇺🇸

Hallandale Beach, Florida, United States

Munroe Regional Medical Center

🇺🇸

Ocala, Florida, United States

DePaul Health Center-MRI Department

🇺🇸

St. Louis, Missouri, United States

Samsung Medical Center, Department of Neurology

🇰🇷

Seoul, Korea, Republic of

Renstar Medical Research

🇺🇸

Ocala, Florida, United States

Trinity Care Solutions

🇺🇸

Ocala, Florida, United States

Advanced Imaging of Ocala

🇺🇸

Ocala, Florida, United States

CBH Health, LLC

🇺🇸

Rockville, Maryland, United States

Atlanta Center for Medical Research

🇺🇸

Atlanta, Georgia, United States

Borgess Medical Center

🇺🇸

Kalamazoo, Michigan, United States

Foers Medical Arts Pharmacy

🇺🇸

Bethesda, Maryland, United States

KNI Southwest Michigan Imaging Center, LLC

🇺🇸

Kalamazoo, Michigan, United States

Memory Enhancement Center of America, Inc.

🇺🇸

Eatontown, New Jersey, United States

Seoul National University Hospital, Department Neurology

🇰🇷

Seongnam-si, Gyeonggi-do, Korea, Republic of

Inha University Hospital, Department of Neurology

🇰🇷

Incheon, Korea, Republic of

ASAN Medical Center

🇰🇷

Seoul, Korea, Republic of

Korea University Anam Hospital IRB

🇰🇷

Seoul, Korea, Republic of

Konkuk University Medical Center, Department of Neurology

🇰🇷

Seoul, Korea, Republic of

Millennium Psychiatric Associates, LLC

🇺🇸

Creve Coeur, Missouri, United States

Central Jersey Radiology

🇺🇸

Oakhurst, New Jersey, United States

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