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An Investigational Study to Evaluate the Effect of Rifampin on the Singe Dose of Experimental Medication BMS-986224 in Healthy Participants

Phase 1
Completed
Conditions
Healthy Participants
Interventions
Registration Number
NCT03563950
Lead Sponsor
Bristol-Myers Squibb
Brief Summary

The purpose of this study is to investigate if the blood levels of experimental medication BMS-986224 will be changed when given together with Rifampin, an antibiotic that affects specific enzymes involved with the breakdown of BMS-986224.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
42
Inclusion Criteria
  • Healthy participant, as determined by no clinically significant deviation from normal in medical history, physical examination, ECGs, and clinical laboratory determinations
  • Body mass index (BMI)of 18.0to 30.0 kg/m2, inclusive, at screening
Exclusion Criteria
  • Women of childbearing potential
  • Any significant acute or chronic medical illness
  • Current or recent (within 3 months of study treatment administration) gastrointestinal disease that could affect absorption or history of cholecystectomy

Other protocol defined inclusion/exclusion criteria may apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Rifampin + BMS-986224RifampinOral administration
Rifampin + BMS-986224BMS-986224Oral administration
Primary Outcome Measures
NameTimeMethod
Area under the plasma concentration-time curve from time zero extrapolated to infinite time [AUC(INF)] of BMS-9862245 days
Maximum observed plasma concentration (Cmax) of BMS-9862245 days
Area under the plasma concentration-time curve from time zero to time of last quantifiable concentration [AUC(0-T)] of BMS-9862245 days
Secondary Outcome Measures
NameTimeMethod
Incidence of AEs leading to discontinuation17 days
Biomarker plasma concentrations of BMS-9862245 days
Time of maximum observed plasma concentration (Tmax) of BMS-9862245 days
Terminal elimination half-life (T-HALF) of BMS-9862245 days
Metabolite of BMS-986224 Cmax5 days
Metabolite of BMS-986224 AUC(0-T)5 days
Metabolite of BMS-986224 AUC(INF)5 days
Incidence of nonserious adverse events (AE)17 days
Composite results of vital signs, electrocardiograms, physical examinations,and clinical laboratory tests18 days
Incidence of serious adverse events (SAE)30 days

Trial Locations

Locations (1)

PRA Health Sciences

🇺🇸

Salt Lake City, Utah, United States

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