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Ibalizumab Plus Optimized Background Regimen in Patient With Multi-Drug Resistant HIV

Phase 3
Completed
Conditions
HIV
Interventions
Biological: ibalizumab
Drug: Optimized Background Regimen (OBR)
Registration Number
NCT02475629
Lead Sponsor
TaiMed Biologics Inc.
Brief Summary

This Phase 3, single arm, multicenter study will evaluate the safety and effectiveness of ibalizumab in treatment-experienced patients infected with multi-drug resistant HIV-1.

Detailed Description

This Phase 3, single arm, multicenter study will evaluate the safety and effectiveness of ibalizumab in treatment-experienced patients infected with multi-drug resistant HIV-1. Patients must have been treated with HAART for at least 6 months and be failing or have recently failed (i.e., in the last 8 weeks) therapy to determine baseline viral load.

Days 0-6 of the study will be a "control period." During Days 0 through 6 patients will be monitored on current failing therapy (or no therapy, if the patient has failed and discontinued treatment within the 8 weeks preceding Screening).

Days 7-13 of the study will be an "essential monotherapy period." During Days 7 through 13 patients will continue on current failing therapy and receive one 2000 mg dose (loading dose) of ibalizumab on Day 7. Day 7 is Baseline for the treatment period (Day 7-Week 25).

Day 14-Week 25 of the study will be the "maintenance period." On Day 14 (primary endpoint), the OBR will be initiated and must include at least one agent to which the patient's virus is susceptible. Beginning at Day 21, 800 mg of ibalizumab will be administered every 2 weeks through Week 23.

End of Study evaluations will be performed at Week 25, and a follow-up visit will be conducted at Week 29.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
40
Inclusion Criteria
  • Are capable of understanding and have voluntarily signed the informed consent document
  • Have documented HIV-1 infection by official, signed, written history (e.g., laboratory report), otherwise an HIV-antibody test will be performed
  • Have no acquired immunodeficiency syndrome (AIDS)-defining events in the 3 months before Screening, other than cutaneous Kaposi's sarcoma or wasting syndrome due to HIV
  • Are able and willing to comply with all protocol requirements and procedures
  • Have a life expectancy that is >6 months.
  • Have a viral load >1,000 copies/mL and documented resistance to at least one antiretroviral medication from each of three classes of antiretroviral medications as measured by resistance testing
  • Have a history of at least 6 months on antiretroviral treatment
  • Are receiving a stable highly active antiretroviral regimen for at least 8 weeks before Screening and are willing to continue that regimen until Day 14, OR (in the past 8 weeks) have failed and are off therapy and are willing to stay off therapy until Day 14
  • Have full viral sensitivity/susceptibility to at least one antiretroviral agent, other than ibalizumab, as determined by the screening resistance tests and be willing and able to be treated with at least one agent to which the patient's viral isolate is fully sensitive/susceptible according to the screening resistance tests as a component of OBR
  • If sexually active, are willing to use an effective method of contraception during the study and for 30 days after the last administration of the study drug
Exclusion Criteria
  • Any active AIDS-defining illness per Category C conditions according to the Centers for Disease Control and Prevention (CDC) Classification System for HIV Infection, with the following exceptions: cutaneous Kaposi's sarcoma and wasting syndrome due to HIV
  • Any significant diseases (other than HIV-1 infection) or clinically significant findings, including psychiatric and behavioral problems, determined from screening, medical history and/or physical examination that, in the investigator's opinion, would preclude the patient from participating in this study
  • Any significant acute illness within 1 week before the initial administration of study drug
  • Any active infection secondary to HIV requiring acute therapy; however, patients that require maintenance therapy (i.e., secondary prophylaxis for opportunistic infections) will be eligible for the study.
  • Any immunomodulating therapy (including interferon), systemic steroids, or systemic chemotherapy within 12 weeks before Enrollment
  • Any prior exposure to ibalizumab (formerly TNX-355 and Hu5A8)
  • Any vaccination within 7 days before Enrollment
  • Any female patient who either is pregnant, intends to become pregnant, or is currently breastfeeding
  • Any current alcohol or illicit drug use that, in the investigator's opinion, will interfere with the patient's ability to comply with the study schedule and protocol evaluations
  • Any previous clinically significant allergy or hypersensitivity to any excipient in the ibalizumab formulation
  • Any radiation therapy during the 28 days before first administration of investigational medication
  • Any Grade 3 or 4 laboratory abnormality according to the Division of AIDS grading scale, except for the following asymptomatic Grade 3 events triglyceride elevation total cholesterol elevation

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Open-Label Ibalizumab plus OBRibalizumab2000 mg intravenous ibalizumab (loading dose) on Day 7 followed in 14 days (on Day 21) by 800 mg intravenous ibalizumab administered once every two weeks, plus an Optimized Background Regimen (OBR) beginning on Day 14.
Open-Label Ibalizumab plus OBROptimized Background Regimen (OBR)2000 mg intravenous ibalizumab (loading dose) on Day 7 followed in 14 days (on Day 21) by 800 mg intravenous ibalizumab administered once every two weeks, plus an Optimized Background Regimen (OBR) beginning on Day 14.
Primary Outcome Measures
NameTimeMethod
Efficacy: Proportion of Participants Achieving a Viral Load Reduction of at Least 0.5 Log 10: ITT-MEFDay 14

Proportion of participants (%) achieving a viral load reduction of at least 0.5 log from baseline (Day 7)

Efficacy: Proportion of Subjects With a Viral Load Decrease of at Least 0.5 Log 10 - Protocol CorrectDay 14

Proportion of patients (%) with a viral load decrease of at least 0.5 log 10 from baseline (day 7)

Secondary Outcome Measures
NameTimeMethod
End of Study Viral Load Reductions as a Measure of Efficacy - Protocol Correct Analysisat Week 25/End of Study

Proportion of patients achieving a \>/= 0.5 log10 and \>/= 1.0 log10 decrease from Day 7/Baseline in viral load at Week 25/End of Study

Efficacy: Proportion of Patients With Undetectable Viral Load: ITT-MEFWeek 25 /end of study

Proportion of patients with undetectable Viral Load (\<50 copies/mL, and \<400 copies/mL)

Efficacy: Proportion of Patients With Undetectable HIV-RNA Levels: Protocol CorrectWeek 25/End of Study

Proportion of patients (%) with HIV-RNA levels \< 50 copies/mL and \< 400 copies/mL at Week 25/End of Study

Mean Change in Viral Load as a Measure of Efficacy - ITT-MEFDay 7 and Day 14

Mean change from Day 7/Baseline in log 10 vial load measured at Day 14

Mean Change in Viral Load as a Measure of Efficacy - Protocol CorrectDay 7 and Day 14

Mean change from Day 7/Baseline in Log 10 viral load measured at Day 14

End of Study Viral Load Reductions as a Measure of Efficacy - Intent to Treat Analysisat Week 25/End of Study

Proportion of patients achieving a \>/= 0.5 log10 and \>/= 1.0 log10 decrease from Day 7/Baseline in viral load at Week 25/End of Study

Mean Change in CD4+ Cell Count as a Measure of Efficacy and Safety - ITTDay 7 and Week 25/End of Study

Mean change from Day 7/Baseline in CD4+ cell count at Week 25/End of Study

Mean Change in CD4+ Cell Count as a Measure of Efficacy and Safety - Protocol CorrectDay 7 and Week 25/End of Study

Mean change from Day 7/Baseline in CD4+ cell count at Week 25/End of Study

Safety: Proportion of Participants Experiencing Adverse EventsThrough Week 25/End of Study

Proportion of participants experiencing at least one treatment emergent adverse event to week 25/End of Study

Proportion of Participants Experiencing Adverse Event Related to Study Drug as a Measure of Safety and TolerabilityThrough Week 25/End of Study

Proportion of participants experiencing a treatment emergent adverse event determined by the investigator to be related to study drug

Proportion of Participants Experiencing Serious Adverse Event as a Measure of Safety and TolerabilityThrough Week 25/End of Study

Proportion of participants experiencing at least one serious treatment emergent adverse event, excluding death

Proportion of Participants Discontinuing Study Drug Due to Adverse EventThrough Week 25/End of Study

Proportion of participants discontinuing study drug due to occurrence of treatment emergent adverse event

Proportion of Participants Experiencing Adverse Event Grade 3 and Higher as a Measure of Safety and TolerabilityThrough Week 25/End of Study

Proportion of participants experiencing treatment emergent adverse event Grade 3 and higher

Proportion of Participants Experiencing Adverse Event With Death as Outcome as a Measure of Safety and TolerabilityThrough Week 25/End of Study

Proportion of participants experiencing treatment emergent adverse event with death as the outcome, regardless of relationship to study drug

Proportion of Participants Experiencing New AIDS-defining Adverse Event According to CDC Criteria as a Measure of Safety and TolerabilityThrough Week 25/End of Study

Proportion of participants experiencing treatment emergent adverse event that is AIDS-defining by the CDC adverse event classification criteria for HIV infection

Trial Locations

Locations (30)

University of Maryland, Institute of Human Virology

🇺🇸

Baltimore, Maryland, United States

Research Access Network

🇺🇸

Houston, Texas, United States

W King Health Care Group

🇺🇸

Los Angeles, California, United States

Midway Immunology and Research Center

🇺🇸

Fort Pierce, Florida, United States

Anthony Mills, MD, Inc.

🇺🇸

Los Angeles, California, United States

Triple O Research Institute

🇺🇸

West Palm Beach, Florida, United States

St. John Hospital and Medical Center

🇺🇸

Southfield, Michigan, United States

Georgetown University School of Medicine

🇺🇸

Washington, District of Columbia, United States

Henry Ford Health Systems

🇺🇸

Detroit, Michigan, United States

Gary Richmond, MD, PA

🇺🇸

Fort Lauderdale, Florida, United States

AIDS Research Consortium of Atlanta

🇺🇸

Atlanta, Georgia, United States

Clinical Research PR, Inc

🇵🇷

San Juan, Puerto Rico

Kaiser Foundation Research Institute

🇺🇸

San Francisco, California, United States

University of Miami

🇺🇸

Miami, Florida, United States

Long Beach Education and Research Consultants

🇺🇸

Long Beach, California, United States

Southern California Permanente Medical Group

🇺🇸

Los Angeles, California, United States

Ruane Medical and Clinical Research Institute

🇺🇸

Los Angeles, California, United States

Charles R. Drew Univ. of Med. & Science Clinical and Translational Research Center

🇺🇸

Los Angeles, California, United States

Quest Clinical Research

🇺🇸

San Francisco, California, United States

Orlando Immunology Center

🇺🇸

Orlando, Florida, United States

ACRIA

🇺🇸

New York, New York, United States

North Texas Infectious Disease Consultants

🇺🇸

Dallas, Texas, United States

Carolinas HealthCare System

🇺🇸

Charlotte, North Carolina, United States

Circle Care Center, LLC

🇺🇸

Norwalk, Connecticut, United States

Palmtree Clinical Research Inc.

🇺🇸

Palm Springs, California, United States

National Taiwan University Hospital

🇨🇳

Taipei, Taiwan

Yale University

🇺🇸

New Haven, Connecticut, United States

E-Da Hospital

🇨🇳

Kaohsiung, Taiwan

Montefiore Medical Center

🇺🇸

Bronx, New York, United States

AIDS Healthcare Foundation

🇺🇸

Los Angeles, California, United States

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