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Ketamine for Thrombolysis in Acute Ischemic Stroke

Phase 1
Conditions
Stroke
Interventions
Drug: Placebo
Registration Number
NCT02258204
Lead Sponsor
University Hospital, Caen
Brief Summary

KETA trial is a nonprofit, double-blind, randomized, controlled pilot trial with aiming to determine if co-administration of ketamine with recombinant of tissue type plasminogen activator (tPA) for thrombolysis in acute ischemic stroke compared with tPA co-administered with placebo, decreases cerebral infarction growth in diffusion weighted imaging between admission and day 1. Eligibility applies to patients with symptomatic ischemic stroke seen within 4.5 h of onset with middle cerebral artery or distal internal carotid artery occlusion, no contraindication to intravenous tPA-mediated thrombolysis and eligible to endovascular treatment of stroke (i.e. thrombectomy). The study has been designed to have 80% power to detect a 80% decrease of infarct volume growth in the tPA-ketamine group at a two-sided type I error rate of 5%. For this purpose, at least 25 patients per arm should be enrolled.

Detailed Description

Rationale - Tissue-type plasminogen activator (tPA) is a double-sided molecule, with beneficial effect in acute ischemic stroke due to its intravascular fibrinolytic activity but with potential deleterious effect due to its ability to potentiate neuronal N-methyl-D-aspartate (NMDA) receptor signalling (Nicole et al., 2001). Co-administration of sub-anesthetic dose of ketamine - a non-competitive inhibitor of NMDA receptor - was shown to improve efficacy of tPA-mediated thrombolysis following stroke in rodents (Gakuba et al, 2011).

Aims - To assess efficacy and safety of co-administration of ketamine with tPA compared with tPA-placebo infusion in patients with acute ischemic stroke.

Sample size estimates -With 25 patients per group, the trial has a 80% probability of detecting a 80% decrease of infarct volume growth in the tPA-ketamine group compared with the tPA-placebo group on day 1 after admission at a two-sided type I error rate of 5%.

Study outcomes - The primary efficacy outcome is cerebral infarction growth on diffusion weighted imaging between admission and day 1. The primary safety measure is mortality and/or symptomatic intracerebral hemorrhage rate at 3 months.

Recruitment & Eligibility

Status
UNKNOWN
Sex
All
Target Recruitment
50
Inclusion Criteria
  • Sudden focal neurological deficit attributable to acute ischemic stroke.
  • Age between 18 and 85.
  • Time from symptom onset less than 4.5 hours.
  • NIHSS score between 7 and 20.
  • Informed consent for participation.
  • Ketamine can be administered within 15 minutes after onset of tPA infusion.
  • MRI-based AIS diagnosis.
  • Middle cerebral (M1 or M2 segment) and/or distal internal carotid artery occlusion.
  • No intracranial hemorrhage on MRI.
  • Patient eligible for thrombectomy.
Exclusion Criteria
  • Contraindication to IV tPA treatment.
  • Contraindication to ketamine.
  • Contraindication to MRI.
  • Contraindication to intravascular iodinated contrast media.
  • Consciousness level >1 on question 1a of NIHSS.
  • Pre-stroke mRS ≥3.
  • Concomitant medical illness that would interfere with outcome assessments and follow-up (e.g. advanced cancer or respiratory disease).
  • Previous participation in this trial or current participation in another investigational drug trial.
  • Infarct volume on diffusion weighted MRI more than 100 mL.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
tPA-placeboPlacebotPA infusion : 0.9 mg/kg (90 mg maximum), 10% of the total dose is administered as an initial IV bolus dose over 1 minute and the remainder of the dose is infused over 60 minutes. Saline infusion : 0.15 mL/kg IV bolus (maximum 15 mL) followed by an IV infusion of 0.15 mL/kg over 60 minutes (maximum 15 mL).
tPA-ketamineKetaminetPA infusion : 0.9 mg/kg (90 mg maximum), 10% of the total dose is administered as an initial IV bolus dose over 1 minute and the remainder of the dose is infused over 60 minutes. Ketamine infusion : 0.15 mg/kg IV bolus (maximum 15 mg) followed by an IV infusion of 0.15 mg/kg over 60 minutes (maximum 15 mg).
Primary Outcome Measures
NameTimeMethod
Cerebral infarction growth on diffusion weighted magnetic resonance imaging between admission and day 1.Day 1
Secondary Outcome Measures
NameTimeMethod
National Institute of Health Stroke Scaleday 0, day 1, day 7 and day 90
Modified Rankin Scaleday 90
Infarction volume on diffusion weighted magnetic resonance imagingday 1
T2-weighted Fluid Attenuated Inversion Recovery Imaging infarct volumeday 90
Symptomatic intracerebral hemorrhage and/or deathday 90
Arterial patencyday 0 (before and after thrombectomy) and day 1

Arterial patency will be assessed with the Thrombolysis in Cerebral Infarction (TICI) Score on day 0 before and after thrombectomy (digital subtraction angiography) and day 1 (magnetic resonance angiography).

Trial Locations

Locations (1)

CHU Caen

🇫🇷

Caen, France

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