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A Phase 2 Study of RTA 901 (BIIB143) in Participants With Diabetic Peripheral Neuropathic Pain (CYPRESS)

Phase 2
Terminated
Conditions
Diabetic Peripheral Neuropathic Pain
Interventions
Drug: RTA 901-Matching Placebo
Registration Number
NCT05895552
Lead Sponsor
Reata, a wholly owned subsidiary of Biogen
Brief Summary

This is a 2-part, randomized, placebo-controlled, double-blind, Phase 2 study to evaluate the safety, tolerability, efficacy, and pharmacokinetics (PK) of RTA 901 in qualified participants with Diabetic Peripheral Neuropathic Pain (DPNP). Each study part will be randomized into 3 treatment arms; 2 different doses of RTA 901 and RTA 901-maching placebo. The doses of RTA 901 in Part 2 will be selected based on the Exposure-Response (E-R) analyses of data from Part 1. A total of 384 participants will be randomized in this study. Each part will have 192 participants, with 64 participants randomized 1:1:1 to each treatment arm.

The duration of each part of the study will be approximately 20 weeks, including a Screening period of up to 2 weeks, a Run-in-period of 2 weeks, a Treatment period of 12 weeks, and a Follow-up period of 4 weeks. All participants in Part 1 and Part 2 of the study will follow the same visit and assessment schedule. Eligibility will be assessed during the Screening and Run-in-periods.

Detailed Description

Study Sponsor, originally Reata Pharmaceuticals, Inc., is now Reata Pharmaceuticals, Inc., a wholly owned subsidiary of Biogen.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
209
Inclusion Criteria
  • Diagnosis of type 1 diabetes mellitus (T1DM) or type 2 diabetes mellitus (T2DM) at least 1 year prior to Screening
  • Clinical diagnosis of DPNP defined as symptomatic distal symmetric polyneuropathy (secondary to diabetes) in the lower extremities, which may include symptoms of pain that is burning, lancinating, tingling, or shooting (electric shock-like). Pain in the lower extremities may occur with paresthesia or dysesthesia (unpleasant sensations of burning). Neuropathic pain may be accompanied by an exaggerated response to painful stimuli (hyperalgesia) and pain evoked by light touch or contact, eg, with socks, shoes, and bedclothes (allodynia);
  • NPRS pain intensity score ≥ 4 on an 11-point scale at Screening
  • A score ≥ 2.5 on the Michigan Neuropathy Screening Instrument (MNSI) Part B

Run-in

Exclusion Criteria
  • Has neuropathy from a cause other than T1DM or T2DM
  • Has a condition other than DPNP that could confound the assessment of pain (eg, fibromyalgia or regional pain caused by lumbar or cervical compression);
  • Diabetic foot ulceration or infection within 90 days prior to Screening
  • Prior participation in a study with RTA 901;

NOTE: Other protocol-defined Inclusion/Exclusion criteria may apply.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Part 1 RTA 901 Dose 1RTA 901Participants will receive study drug, once daily (QD), during the 2-week Run-in Period. Following randomization, the participants will receive a dose of RTA 901, QD, for a 12-week treatment duration.
Part 1 RTA 901 Dose 2RTA 901Participants will receive study drug, QD, during the 2-week Run-in Period. Following randomization, the participants will receive a dose of RTA 901, QD, for a 12-week treatment duration.
Part 1 RTA 901-Matching PlaceboRTA 901-Matching PlaceboParticipants will receive study drug, QD, during the 2-week Run-in Period. Following randomization, the participants will receive a dose of RTA 901-matching placebo, QD, for a 12-week treatment duration.
Part 2 RTA 901-Matching PlaceboRTA 901-Matching PlaceboParticipants will receive study drug, QD, during the 2-week Run-in Period. Following randomization, the participants will receive a dose of RTA 901-matching placebo, QD, for a 12-week treatment duration.
Part 2 RTA 901 Dose 1RTA 901Participants will receive study drug, QD, during the 2-week Run-in Period. Following randomization, the participants will receive a dose of RTA 901, QD, for a 12-week treatment duration.
Part 2 RTA 901 Dose 2RTA 901Participants will receive study drug, QD, during the 2-week Run-in Period. Following randomization, the participants will receive a dose of RTA 901, QD, for a 12-week treatment duration.
Primary Outcome Measures
NameTimeMethod
Number of Participants With Clinically Significant Abnormality in Physical ExaminationsBaseline up to Week 16
Number of Participants With Clinically Significant Abnormality in Vital SignBaseline up to Week 16
Number of Participants With Clinically Significant Abnormality in Electrocardiogram (ECG)Baseline up to Week 16
Number of Participants With Clinically Significant Abnormality in Clinical Laboratory MeasurementBaseline up to Week 16
Number of Participants With Clinically Significant Abnormality in Body WeightBaseline up to Week 16
Change From Baseline in Average Daily Pain Intensity as Assessed by the Numeric Pain Rating Scale (NPRS) at Week 12Baseline, Week 12

The NPRS of pain intensity is a numeric scale, ranging from 0 (representing no pain at all) to 10 (representing the worst pain imaginable). The participant will select a whole number (0 to 10) that best indicates the intensity of his/her pain in the past 24 hours. Lower scores indicate less pain.

Number of Participants With Adverse Events (AEs) and Serious Adverse Events (SAEs) During and Following the Treatment PeriodFrom the first day of dosing up to end of follow-up period (Week 16)
Secondary Outcome Measures
NameTimeMethod
Number of Participants who Achieved at Least a 50% Decrease From Baseline in the Average NPRS Score at Week 12Week 12

The NPRS of pain intensity is a numeric scale, ranging from 0 (representing no pain at all) to 10 (representing the worst pain imaginable). The participant will select a whole number (0 to 10) that best indicates the intensity of his/her pain in the past 24 hours. Lower scores indicate less pain.

Duration of Rescue Medications Used During the Treatment PeriodUp to Week 12
Number of Participants who Achieved at Least a 30% Decrease From Baseline in the Average NPRS Score at Week 12Week 12

The NPRS of pain intensity is a numeric scale, ranging from 0 (representing no pain at all) to 10 (representing the worst pain imaginable). The participant selects a whole number (0 to 10) that best indicates the intensity of his/her pain in the past 24 hours. Lower scores indicate less pain.

Number of Participants Using Rescue Medications During the Treatment PeriodUp to Week 12
Amount of Rescue Medications Used During the Treatment PeriodUp to Week 12
Change From Baseline in the Average Daily Sleep Interference Scale (DSIS) score at Week 12Baseline, Week 12

DSIS is a participant reported outcome that was developed to quantify sleep interference due to pain. The DSIS will be completed daily by participants upon waking (3-minute self-administered questionnaire), preferably in the morning, to accurately capture variability in sleep interference due to pain, thus minimizing recall bias. Using the e-diary, participants will assess how pain has interfered with their sleep during the past 24 hours. This score ranges from 0 to 10; 0 representing no interference with sleep to 10 representing complete inability to sleep. Lower score indicates less pain interference during sleep.

Trial Locations

Locations (68)

Centricity Research Phoenix Multispecialty

🇺🇸

Mesa, Arizona, United States

Arizona Research Center

🇺🇸

Phoenix, Arizona, United States

Hope Clinical Research, Inc.

🇺🇸

Canoga Park, California, United States

Valley Research - Trials

🇺🇸

Fresno, California, United States

Clinical Research Institute

🇺🇸

Los Angeles, California, United States

Acclaim Clinical Research

🇺🇸

San Diego, California, United States

Optimus Medical Group

🇺🇸

San Francisco, California, United States

PIH Health Whittier Hospital

🇺🇸

Whittier, California, United States

Denver Endocrinology Diabetes and Thyroid Center PC

🇺🇸

Englewood, Colorado, United States

Paradigm Clinical Research

🇺🇸

Wheat Ridge, Colorado, United States

Innovative Research of West Florida, Inc.

🇺🇸

Clearwater, Florida, United States

Clinical Research of West Florida Inc

🇺🇸

Clearwater, Florida, United States

East Coast Institute for Research, LLC

🇺🇸

Macon, Georgia, United States

Multi Specialty Research Associates, LLC

🇺🇸

Lake City, Florida, United States

3 Sync LLC

🇺🇸

Kingwood, Texas, United States

Floridian Clinical Research

🇺🇸

Miami Lakes, Florida, United States

Finlay Medical Research

🇺🇸

Miami, Florida, United States

New Horizon Research Center

🇺🇸

Miami, Florida, United States

IMA Clinical Research, PC

🇺🇸

Saint Petersburg, Florida, United States

Genesis Clinical Research

🇺🇸

Tampa, Florida, United States

Clinical Research of West Florida, Inc.

🇺🇸

Tampa, Florida, United States

Baycare Clinical Research

🇺🇸

Tampa, Florida, United States

VICIS Clinical Research

🇺🇸

Tampa, Florida, United States

Clinical Site Partners, Orlando

🇺🇸

Winter Park, Florida, United States

Conquest Research, LLC

🇺🇸

Winter Park, Florida, United States

Agile Clinical Research Trials, LLC

🇺🇸

Atlanta, Georgia, United States

Centricity Research Columbus Endocrinology

🇺🇸

Columbus, Georgia, United States

Methodist Medical Center of Illinois

🇺🇸

Peoria, Illinois, United States

MediSphere Medical Research Center, LLC

🇺🇸

Evansville, Indiana, United States

Integrated Clinical Trial Services, Inc.

🇺🇸

West Des Moines, Iowa, United States

Tandem Clinical Research

🇺🇸

Metairie, Louisiana, United States

Boston Clinical Trials, LLC

🇺🇸

Boston, Massachusetts, United States

Brigham and Women's Hospital

🇺🇸

Boston, Massachusetts, United States

ActivMed Practices & Research, LLC

🇺🇸

Portsmouth, New Hampshire, United States

Revival Research Institute, LLC.

🇺🇸

Sterling Heights, Michigan, United States

Clinical Research Consultants, LLC

🇺🇸

Kansas City, Missouri, United States

StudyMetrix Research

🇺🇸

Saint Peters, Missouri, United States

Velocity Clinical Research, Inc.

🇺🇸

Norfolk, Nebraska, United States

Las Vegas Endocrinology

🇺🇸

Henderson, Nevada, United States

Jubilee Clinical Research Inc

🇺🇸

Las Vegas, Nevada, United States

Excel Clinical Research

🇺🇸

Las Vegas, Nevada, United States

Columbia University

🇺🇸

New York, New York, United States

Richmond Behavioral Associates

🇺🇸

Staten Island, New York, United States

Carolina Institute for Clinical Research, LLC

🇺🇸

Fayetteville, North Carolina, United States

Diabetes & Endocrinology Associates of Stark County, Inc.

🇺🇸

Canton, Ohio, United States

Velocity Clinical Research, Cincinnati

🇺🇸

Cincinnati, Ohio, United States

Cleveland Clinic

🇺🇸

Cleveland, Ohio, United States

Remington-Davis, Inc.

🇺🇸

Columbus, Ohio, United States

Meta Medical Research Institute

🇺🇸

Dayton, Ohio, United States

Velocity Clinical Research, Providence

🇺🇸

East Greenwich, Rhode Island, United States

Notus Clinical Research

🇺🇸

Charleston, South Carolina, United States

WR-ClinSearch, LLC

🇺🇸

Chattanooga, Tennessee, United States

Trinity Clinical Research LLC

🇺🇸

Tullahoma, Tennessee, United States

FutureSearch Trials of Neurology

🇺🇸

Austin, Texas, United States

REX Clinical Trials, LLC

🇺🇸

Beaumont, Texas, United States

Zenos Clinical Research

🇺🇸

Dallas, Texas, United States

Care United Research, LLC

🇺🇸

Forney, Texas, United States

Diabetes and Thyroid Center of Fort Worth

🇺🇸

Fort Worth, Texas, United States

Nerve and Muscle Center of Texas

🇺🇸

Houston, Texas, United States

Biopharma Informatic, LLC

🇺🇸

Houston, Texas, United States

Endocrine IPS, PLLC

🇺🇸

Houston, Texas, United States

Amir A Hassan, MD, PA

🇺🇸

Houston, Texas, United States

Epic Clinical Research

🇺🇸

Lewisville, Texas, United States

Shadow Creek Medical Clinic

🇺🇸

Pearland, Texas, United States

Diabetes & Glandular Disease Clinic, P.A.

🇺🇸

San Antonio, Texas, United States

VIP Trials

🇺🇸

San Antonio, Texas, United States

Velocity Clinical Research, Salt Lake City

🇺🇸

West Jordan, Utah, United States

Rainier Clinical Research Center

🇺🇸

Renton, Washington, United States

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