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STC-15 as a Part of Combination Therapy With Toripalimab in Selected Advanced Cancers

Phase 1
Recruiting
Conditions
Metastatic Non-small Cell Lung Cancer
Metastatic Melanoma
Metastatic Endometrial Cancer
Metastatic Head-and-neck Squamous-cell Carcinoma
Solid Tumor
Registration Number
NCT06975293
Lead Sponsor
STORM Therapeutics LTD
Brief Summary

This early phase oncology trial will be conducted at various study centers to investigate the safety, tolerability, and antitumor activity of STC-15 (a METTL3 inhibitor) in combination with toripalimab (anti- programmed cell death 1 \[PD-1\]) in four different locally advanced unresectable or metastatic tumors such as indications: (1) in combination with toripalimab (anti- programmed cell death 1 \[PD-1\]) in locally advanced and unresectable or metastatic non-small cell lung cancer (NSCLC), (2) in combination with toripalimab in locally advanced unresectable or metastatic melanoma, (3) in combination with toripalimab in locally advanced unresectable or metastatic endometrial cancers, and (4) in combination with toripalimab in locally advanced or metastatic head and neck squamous cell carcinoma (HNSCC).

This study comprises of 2 parts: a combination dose escalation part (Phase 1b) followed by an assessment of the combination treatment's antitumor activity (Phase 2). This study will be conducted in adult participants with advanced malignancies to characterize the safety, tolerability, PK, and clinical activity of STC-15 in combination with toripalimab.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
188
Inclusion Criteria
  • Estimated life expectancy ≥ 3 months.
  • ECOG performance status 0 or 1.
  • Measurable disease according to RECIST v1.1 as assessed by the local site investigator/radiology.
  • Documented radiologic assessment of progression on the prior therapy before study entry.
  • Have the ability to swallow, retain, and absorb oral medication.

Inclusion Criteria (Expansion):

  • NSCLC (when applicable): Participants with AGAs (actionable genetic alterations) must have received targeted therapy unless contraindicated. Participants must not have received more than three previous lines of systemic treatment for unresectable locally advanced or metastatic disease. This must include at least a prior anti-PD-1/L1 alone or in combination with chemotherapy. Participants must have disease progression on prior anti-PD-1/L1.
  • HNSCC (when applicable): Participants must have progressed on following prior lines: 2L or 3L recurrent/metastatic disease; regardless of PD-L1 score. Participants must not have received more than three previous lines of systemic treatment for unresectable locally advanced or metastatic disease. This must include at least a prior anti-PD-1/L1 alone or in combination with chemotherapy.
  • Endometrial (when applicable): Participants must not have received more than three previous lines of systemic treatment for unresectable locally advanced or metastatic disease. This must include at least a prior anti-PD-1/L1 alone or in combination with chemotherapy. Participants must have disease progression on prior anti-PD-1/L1
  • Melanoma (when applicable): Participants must not have received more than three previous lines of systemic treatment for unresectable locally advanced or metastatic disease. This must include at least a prior anti-PD-1/L1 alone or in combination with chemotherapy. Participants must have disease progression on prior anti-PD-1/L1.

Key

Exclusion Criteria
  • Pregnant and lactating women.
  • Received prior systemic anticancer therapy including investigational agents within 4 weeks prior to first IMP administration.
  • Participants who have not recovered from all AEs due to previous therapies to Grade ≤ 1 or baseline, according to NCI-CTCAE v5.0. Exceptions include: alopecia, Grade ≤ 2 neuropathy, and endocrine-related AEs Grade ≤ 2 who are stable on treatment or hormone replacement.
  • Major surgery less than 4 weeks prior to the first IMP administration or participants who have not recovered from the side effects of the surgery.
  • History of (non-infectious) pneumonitis/interstitial lung disease that required steroids or the presence of ongoing pneumonitis/interstitial lung disease).
  • Clinically significant cardiovascular disease or condition.
  • Known active CNS metastases and/or leptomeningeal disease.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Primary Outcome Measures
NameTimeMethod
Safety and tolerability of STC-15 in combination with toripalimab6 months

Incidence of adverse events graded according to CTCAE v5.0

Secondary Outcome Measures
NameTimeMethod
Anti-tumor activity6 months

To evaluate the antitumor activity of STC-15 in combination with toripalimab as per Response Evaluation Criteria in Solid Tumors (RECIST) v1.1 and immune RECIST (iRECIST) criteria

Maximum observed plasma concentration of STC-15 (Cmax)22 days
Recommended Phase 2 Dose6 months

Identification of a tolerable and safe dose for expansion cohorts based on dose limiting toxicities

Calculated time to reach maximum observed plasma concentration (Tmax)22 days
Calculated area under the plasma concentration-time curve of STC-15 (AUC0-t)22 days

Trial Locations

Locations (2)

The START Center

🇺🇸

San Antonio, Texas, United States

NEXT Oncology

🇺🇸

Fairfax, Virginia, United States

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