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A Study of Subcutaneous Blinatumomab Administration in Acute Lymphoblastic Leukemia (ALL) Patients

Phase 1
Active, not recruiting
Conditions
B Cell Precursor Acute Lymphoblastic Leukemia
Interventions
Registration Number
NCT04521231
Lead Sponsor
Amgen
Brief Summary

The study aims to evaluate the safety, efficacy, and tolerability of subcutaneous (SC) blinatumomab for treatment of Acute Lymphoblastic Leukemia (ALL), to determine the maximum tolerated dose (MTD), and recommended phase 2 dose(s) (RP2D) of SC administered blinatumomab. It will also conduct a clinical PK evaluation of SC1 and SC2 blinatumomab formulations.

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
125
Inclusion Criteria
  • Aged 18 years or older (or same or greater than legal age within the country if it is older than 18 years).

  • Participants with B-precursor ALL with any of the following:

    • Either refractory to primary induction therapy or refractory to at least 1 salvage therapy OR

    • In untreated first, second, third or greater relapse or refractory relapse

      • First Relapse is defined as achievement of first Complete Remission (CR) [CR1] during upfront therapy then relapse during or after continuation therapy
      • Primary Refractory disease is defined as the absence of CR after standard induction therapy
      • Refractory relapse is defined as lack of CR after salvage treatment
      • Second relapse or later relapse is defined as relapse after achieving a second CR (CR2) in first or later salvage
      • Refractory to salvage is defined as no attainment of CR after salvage
  • Relapsed or Refractory at any time after first salvage therapy.

  • Relapse at any time after allogenic hematopoietic stem cell transplant (HSCT).

  • Greater than or equal to 5% blasts in the Bone Marrow (Exception: Isolated Non-central nervous system (CNS) extramedullary disease [EMD]).

  • Eastern Cooperative Oncology Group (ECOG) Performance Status less than or equal to 2.

  • Participants with relapse or refractory B Cell ALL Ph+ disease and that are intolerant or refractory to prior tyrosine kinase inhibitors (TKIs) are eligible.

The above is a summary, other inclusion criteria details may apply.

Exclusion Criteria
  • Active ALL in the central nervous system (CNS). Presence of greater than 5 white blood cells per cubic millimeter in cerebrospinal fluid (CSF) with lymphoblasts present and/or clinical signs of CNS leukemia.
  • History or presence of clinically relevant CNS pathology such as epilepsy, childhood or adult seizure, paresis, aphasia, stroke, severe brain injuries, dementia, Parkinson's disease, cerebellar disease, organic brain syndrome, psychosis or severe (≥ grade 3) CNS events including immune effector cell-associated neurotoxicity syndrome (ICANS) from prior chimeric antigen receptor T-cell (CAR T) or other T cell engager therapies.
  • Isolated Extramedullary (EM) Disease
  • Symptoms and/or signs that indicate an acute or uncontrolled chronic infection, any other disease or condition that could be exacerbated by the treatment or would complicate protocol compliance.
  • Testicular leukemia
  • History of malignancy (with certain exceptions) other than ALL within 3 years prior to start of protocol-specified therapy.
  • Allogeneic HSCT within 12 weeks before the start of protocol-specified therapy.
  • Cancer chemotherapy within 2 weeks before the start of protocol-specified therapy (with certain exceptions).
  • Immunotherapy within 4 weeks before start of protocol-specified therapy. Prior failed cluster of differentiation (CD19) directed therapy such as prior blinatumomab or CD19 CAR T cells will be allowed, if treatment ended more than 4 weeks prior to start of protocol therapy therapy and no prior CNS complications.
  • Currently receiving treatment in or less than 30 days or 5 half lives since ending treatment on another investigational study(ies).
  • Abnormal screening laboratory parameters.
  • Female participant: Expected to breastfeed during treatment and for 96 hours after the last dose of investigational product (SC blinatumomab).

The above is a summary, other exclusion criteria details may apply.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Dose Expansion Phase: Blinatumomab SC1BlinatumomabUp to 4 cohorts of participants with R/R B-ALL will be enrolled to the preliminary recommended phase 2 dose (RP2D) and schedule determined from dose escalation phase. Each cohort will aim to further assess safety, pharmacokinetics (PK), pharmacodynamics (PD), and efficacy.
Dose Escalation Phase: Blinatumomab Subcutaneous Formulation 1 (SC1)BlinatumomabCohorts of at least 3 participants each will be treated with escalating doses of bilinatumomab to determine the maximum tolerated dose (MTD). The MTD will be defined as the dose for which the estimate of the toxicity rate from an isotonic regression (Yan et al, 2017) is closest to the target toxicity rate. Safety, pharmacokinetics (PK), pharmacodynamics (PD) and efficacy will be assessed.
Ph-IIC: Clinical PK Evaluation of SC Blinatumomab FormulationsBlinatumomab1 cohort of participants will be enrolled into the Ph-IIC arm. The clinical PK evaluation cohort (Ph-IIC) will be conducted to compare the PK of SC1 and SC2 formulations at the RP2D determined from the dose expansion phase, in participants with R/R B-ALL.
Primary Outcome Measures
NameTimeMethod
Dose Escalation Phase: Number of participants who experience dose limiting toxicities (DLTs)Up to 29 days
Dose Escalation Phase: Number of participants who experience one or more treatment-emergent adverse events (TEAEs)Up to approximately 28 weeks
Dose Escalation Phase: Number of participants who experience one or more serious TEAEsUp to approximately 28 weeks
Dose Escalation Phase: Number of participants who experience one or more treatment-related treatment-emergent adverse eventsUp to approximately 28 weeks
Dose Escalation Phase: Number of participants who experience one or more adverse events (AEs) of Interest (AEIs)Up to approximately 28 weeks
Dose Expansion Phase (R/R B-ALL): Number of participants who achieve complete remission (CR)Up to 68 days
Dose Expansion Phase (R/R B-ALL): Number of participants who achieve complete remission with partial hematological recovery (CRh)Up to 68 days
Phase 2 Ph-IIC: Maximum concentration (Cmax) of blinatumomab SC1 and SC2Up to approximately 4 weeks
Phase 2 Ph-IIC: Average concentration (Cavg) of blinatumomab SC1 and SC2Up to approximately 4 weeks
Phase 2 Ph-IIC: Time to reach maximum concentration (Tmax) of blinatumomab SC1 and SC2Up to approximately 4 weeks
Phase 2 Ph-IIC: Area under the concentration-time curve (AUC) of blinatumomab SC1 and SC2Up to approximately 4 weeks
Secondary Outcome Measures
NameTimeMethod
Dose Expansion Phase and Phase 2 (Ph-IIC cohort): Number of participants who experience one or more treatment-related treatment-emergent adverse eventsUp to approximately 28 weeks
Dose Expansion Phase and Phase 2 (Ph-IIC cohort): Number of participants who experience one or more AEIsUp to approximately 28 weeks
Dose Expansion Phase and Phase 2 (Ph-IIC cohort): Summary scores of quality of life at each assessment as assessed by the European Organization for Research and Treatment of Cancer (EORTC) Quality of Life Questionnaire (QLQ-C30)Baseline (Day 1) up to approximately 28 weeks
Dose Expansion Phase and Phase 2 (Ph-IIC cohort): Change from baseline of quality of life as assessed by the EORTC QLQ-C30Baseline (Day 1) up to approximately 28 weeks
Dose Expansion Phase and Phase 2 (Ph-IIC cohort): Relapse-Free Survival in participants who achieve CR/CRh within the first 2 cycles(R/R B-ALL)Up to 68 days
Dose Expansion Phase and Phase 2 (Ph-IIC cohort): Overall survival (OS)Up to approximately 28 weeks
Dose Expansion Phase and Phase 2 (Ph-IIC cohort): Duration of complete responseUp to approximately 28 weeks
Dose Expansion Phase and Phase 2 (Ph-IIC cohort): Number of participants who experience one or more TEAEsUp to approximately 28 weeks
Dose Expansion Phase and Phase 2 (Ph-IIC cohort): Number of participants who experience one or more serious treatment-emergent adverse eventUp to approximately 28 weeks
Dose Escalation Phase: Minimum concentration over the dosing interval (Cmin) of blinatumomabUp to approximately 28 weeks
Dose Escalation Phase: Cmax of blinatumomabUp to approximately 28 weeks
Dose Escalation Phase: Tmax of blinatumomabUp to approximately 28 weeks
Dose Escalation Phase: AUC of blinatumomabUp to approximately 28 weeks
Dose Escalation Phase and Phase 2 (Ph-IIC cohort): Number of participants who achieve CR/CRhUp to 68 days
Dose Escalation, Dose Expansion, and Ph-IIC: Number of participants with incidence of anti-blinatumomab antibody formationUp to approximately 28 weeks
Dose Expansion Phase: Cmin of blinatumomabUp to approximately 28 weeks
Dose Expansion Phase: Cmax of blinatumomabUp to approximately 28 weeks
Dose Expansion Phase: Tmax of blinatumomabUp to approximately 28 weeks
Dose Expansion Phase: AUC of blinatumomabUp to approximately 28 weeks

Trial Locations

Locations (43)

City of Hope National Medical Center

🇺🇸

Duarte, California, United States

University of Texas MD Anderson Cancer Center

🇺🇸

Houston, Texas, United States

Fred Hutchinson Cancer Center

🇺🇸

Seattle, Washington, United States

Westmead Hospital

🇦🇺

Westmead, New South Wales, Australia

Royal Adelaide Hospital

🇦🇺

Adelaide, South Australia, Australia

The Alfred Hospital

🇦🇺

Melbourne, Victoria, Australia

Erasmus Medisch Centrum

🇳🇱

Rotterdam, Netherlands

Hospital Universitario Virgen del Rocio

🇪🇸

Sevilla, Andalucía, Spain

Complejo Asistencial Universitario de Salamanca Hospital Universitario de Salamanca

🇪🇸

Salamanca, Castilla León, Spain

Institut Catala d Oncologia Badalona Hospital Universitari Germans Trias i Pujol

🇪🇸

Badalona, Cataluña, Spain

Hospital Clinico Universitario de Valencia

🇪🇸

Valencia, Comunidad Valenciana, Spain

Clinica Universidad de Navarra

🇪🇸

Pamplona, Navarra, Spain

Hospital Universitario 12 de Octubre

🇪🇸

Madrid, Spain

Bagcilar Medipol Mega Universite Hastanesi

🇹🇷

Istanbul, Turkey

Izmir Ekonomi Universitesi Medical Point Hastanesi

🇹🇷

Izmir, Turkey

New York University Grossman School of Medicine and New York University Langone Hospitals

🇺🇸

New York, New York, United States

Monash Medical Centre

🇦🇺

Clayton, Victoria, Australia

Arthur J E Child Comprehensive Cancer Centre

🇨🇦

Calgary, Alberta, Canada

University of Alberta

🇨🇦

Edmonton, Alberta, Canada

Vancouver General Hospital, Gordon and Leslie Diamond Health Care Centre

🇨🇦

Vancouver, British Columbia, Canada

Universitaetsklinikum Augsburg

🇩🇪

Augsburg, Germany

Charite - Universitaetsmedizin Berlin, Campus Benjamin Franklin

🇩🇪

Berlin, Germany

Universitaetsklinikum Jena

🇩🇪

Jena, Germany

Universitaetsklinikum Koeln

🇩🇪

Koeln, Germany

Universitaetsklinikum Leipzig

🇩🇪

Leipzig, Germany

Universitaetsklinikum Tuebingen

🇩🇪

Tuebingen, Germany

Universitatsklinikum Ulm

🇩🇪

Ulm, Germany

Azienda Socio Sanitaria Territoriale Papa Giovanni xxiii

🇮🇹

Bergamo, Italy

IRCCS Azienda Ospedaliero Universitaria di Bologna Policlinico di Sant Orsola

🇮🇹

Bologna, Italy

Azienda Socio Sanitaria Territoriale degli Spedali Civili di Brescia

🇮🇹

Brescia, Italy

IRCCS Ospedale San Raffaele

🇮🇹

Milano, Italy

Azienda Ospedaliera Policlinico Umberto I

🇮🇹

Roma, Italy

Akita University Hospital

🇯🇵

Akita-shi, Akita, Japan

National Cancer Center Hospital East

🇯🇵

Kashiwa-shi, Chiba, Japan

Austin Health, Austin Hospital

🇦🇺

Heidelberg, Victoria, Australia

Universitaetsklinikum Allgemeines Krankenhaus Wien

🇦🇹

Wien, Austria

Princess Margaret Cancer Centre

🇨🇦

Toronto, Ontario, Canada

Centre Hospitalier Regional Universitaire de Lille - Hopital Claude Huriez

🇫🇷

Lille, France

Centre Hospitalier Universitaire de Nice

🇫🇷

Nice cedex 3, France

Hopital Saint Antoine

🇫🇷

Paris, France

Institut Universitaire du Cancer Toulouse Oncopole

🇫🇷

Toulouse cedex 9, France

Fukushima Medical University Hospital

🇯🇵

Fukushima-shi, Fukushima, Japan

Yokohama City University Medical Center

🇯🇵

Yokohama-shi, Kanagawa, Japan

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