MedPath

Darolutamide in Addition to ADT Versus ADT in Metastatic Hormone-sensitive Prostate Cancer

Phase 3
Active, not recruiting
Conditions
Prostatic Neoplasms
Interventions
Drug: Placebo
Other: Androgen deprivation therapy (ADT)
Registration Number
NCT04736199
Lead Sponsor
Bayer
Brief Summary

The purpose of the study is to assess the efficacy and safety of darolutamide in combination with standard androgen deprivation therapy (ADT) in patients with metastatic hormone sensitive prostate cancer.

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
Male
Target Recruitment
662
Inclusion Criteria
  • Histologically or cytologically confirmed adenocarcinoma of prostate
  • Metastatic disease
  • Started ADT (LHRH agonist/antagonist or orchiectomy) with or without first generation anti-androgen, but not earlier than 12 weeks before randomization
  • Eastern Cooperative Oncology Group (ECOG) Performance Status (PS) of 0, 1 or 2
  • Adequate bone marrow, liver and renal function
Exclusion Criteria
  • Prior treatment with: LHRH agonist/antagonists except neoadjuvant and /or adjuvant therapy; Second-generation androgen receptor (AR) inhibitors such as enzalutamide, darolutamide, apalutamide or other investigational AR inhibitors; Cytochrome P17 enzyme inhibitor such as abiraterone acetate or oral ketoconazole as anti-cancer treatment for prostate cancer; Chemotherapy including docetaxel or immunotherapy for prostate cancer; Use of systemic corticosteroid with dose greater than the equivalent 10 mg of prednisone/day within 28 days prior to randomization; Radiopharmaceuticals; Any other anti-cancer treatment for prostate cancer, excluding local therapies and ADT.
  • Treatment with radiotherapy within 2 weeks before randomization
  • Contraindication to iodinated CT and gadolinium chelate MRI intravenous contrast agent(s)
  • Had any of the following within 6 months before randomization: stroke, myocardial infarction, severe/unstable angina pectoris, coronary/peripheral artery bypass graft, congestive heart failure (New York Heart Association Class III or IV)
  • Uncontrolled hypertension as indicated by a resting systolic BP ≥ 160 mmHg or diastolic BP ≥ 100 mmHg despite medical management
  • A gastrointestinal (GI) disorder or procedure which is expected to interfere significantly with absorption of study drug
  • Any prior malignancy (other than adequately treated basal cell or squamous cell skin cancer, superficial bladder cancer, or any other cancer in situ currently in complete remission) within 5 years prior to randomization
  • Inability to swallow oral medications

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Darolutamide+ADTAndrogen deprivation therapy (ADT)Participants will receive darolutamide 600 mg (2 tablets of 300 mg) twice daily with food and ADT of investigator's choice as standard therapy
Placebo+ADTPlaceboParticipants will receive placebo twice daily with food and ADT of investigator's choice as standard therapy
Placebo+ADTAndrogen deprivation therapy (ADT)Participants will receive placebo twice daily with food and ADT of investigator's choice as standard therapy
Darolutamide+ADTDarolutamide (Nubeqa, BAY1841788)Participants will receive darolutamide 600 mg (2 tablets of 300 mg) twice daily with food and ADT of investigator's choice as standard therapy
Primary Outcome Measures
NameTimeMethod
Radiological progression-free survival (rPFS)36 months

Time from the date of randomization to the date of first documentation of radiological progressive disease or death due to any cause, whichever occurs first.

Secondary Outcome Measures
NameTimeMethod
Overall survival (OS)Up to 55 months

Time from the date of randomization to the date of death from any cause.

Time to castration-resistant prostate cancer (CRPC)Up to 55 months

Time from the date of randomization to the date of first castration resistant event (radiological progression, PSA progression or symptomatic skeletal events, whichever occurs first).

Time to initiation of subsequent anti-cancer therapyUp to 55 months

Time from the date of randomization to initiation of first subsequent anti-cancer therapy for prostate cancer.

Time to PSA progressionUp to 55 months

Time from the date of randomization to the date of first prostate-specific antigen (PSA) progression. PSA progression is defined as a ≥25% increase above the nadir (lowest Screening or baseline) value, which is confirmed by a second value 3 or more weeks later, and an increase in absolute value of ≥ 2 ng/mL above nadir, at least 12 weeks from baseline.

PSA undetectable rates (<0.2 ng/mL)Up to 55 months

The percentage of participants with detectable PSA values (≥0.2 ng/mL) at baseline which become undetectable (\<0.2 ng/mL) during the study treatment.

Time to pain progressionUp to 55 months

Time from the date of randomization to pain progression, where progression is defined as an increase of 2 or more points from baseline. Pain to be assessed with a patient reported questionaire.

Number of participants with adverse events as a measure of safetyUp to 55 months

Trial Locations

Locations (131)

National Cancer Institute

🇱🇹

Vilnius, Lithuania

Nantong tumor hospital

🇨🇳

Nantong, Jiangsu, China

The 2nd Affiliated Hospital of Soochow University

🇨🇳

Suzhou, Jiangsu, China

Christian Medical Center & Hospital

🇮🇳

Ludhiana, Punjab, India

Peking University Third Hospital

🇨🇳

Beijing, China

Post Graduate Institute of Medical Education and Research

🇮🇳

Chandigarh, India

Tata Medical Center

🇮🇳

Kolkata, India

Apex Wellness Hospital

🇮🇳

Nashik, India

Rajiv Gandhi Cancer Institute & Research Centre

🇮🇳

New Delhi, India

Daugavpils Regional Hospital

🇱🇻

Daugavpils, Latvia

RAKUS Hospital Gailezers

🇱🇻

Riga, Latvia

URO Ltd.

🇱🇻

Riga, Latvia

P. Stradins Clinical University Hospital

🇱🇻

Riga, Latvia

Vidzemes Hospital

🇱🇻

Valmiera, Latvia

The Hospital of Lithuanian University of Health SciencesLUHS

🇱🇹

Kaunas, Lithuania

PI Klaipedos University Hospital

🇱🇹

Klaipeda, Lithuania

Vilnius University Hospital Santaros Klinikos

🇱🇹

Vilnius, Lithuania

Canterbury Urology Research Trust

🇳🇿

Christchurch, Canterbury, New Zealand

Waikato Hospital

🇳🇿

Hamilton, New Zealand

Tauranga Urology Research Limited

🇳🇿

Tauranga, New Zealand

Aliada

🇵🇪

San Isidro, Lima, Peru

Hospital Guillermo Almenara Irigoyen

🇵🇪

Santiago de Surco, Lima, Peru

Hospital Militar Luis Arias Schreiber

🇵🇪

Lima, Peru

Clínica El Golf

🇵🇪

Lima, Peru

Arkhangelsk Clinical Oncology Dispensary

🇷🇺

Arkhangelsk, Russian Federation

Ltd "EVIMED"

🇷🇺

Chelyabinsk, Russian Federation

Chelyabinsk Regional Oncology Dispensary

🇷🇺

Chelyabinsk, Russian Federation

Ivanovo Regional Oncology Dispensary

🇷🇺

Ivanovo, Russian Federation

Republican Clinical Oncology Dispensary Kazan

🇷🇺

Kazan, Russian Federation

Research Centre of X-ray and Radiology

🇷🇺

Moscow, Russian Federation

Volga District Med Center FMBA

🇷🇺

Nizhny Novgorod, Russian Federation

LLC Reafan

🇷🇺

Novosibirsk, Russian Federation

Medical Center "Avicenna"

🇷🇺

Novosibirsk, Russian Federation

Clinical Oncological Dispensary of Omsk Region

🇷🇺

Omsk, Russian Federation

AV Medical Group

🇷🇺

St. Petersburg, Russian Federation

Russian Scientific Radiology and Surgery Technologies Center

🇷🇺

St. Petersburg, Russian Federation

Scientific Research Instutute of Oncology n.a. N.N. Petrov

🇷🇺

St. Petersburg, Russian Federation

Multi-Field Clinical Medical Center "Medical City"

🇷🇺

Tyumen, Russian Federation

Republican Clinical Oncology Dispensary

🇷🇺

Ufa, Russian Federation

Vologda Regional Hospital

🇷🇺

Vologda, Russian Federation

Sverdlovsk Regional Clinical Hospital #1

🇷🇺

Yekaterinburg, Russian Federation

Cancercare Langenhoven

🇿🇦

Port Elizabeth, Eastern Cape, South Africa

East Rand Medical Research Unit

🇿🇦

Johannesburg, Gauteng, South Africa

University of Pretoria, Clinical Research Unit

🇿🇦

Pretoria, Gauteng, South Africa

Cape Town Oncology Trials

🇿🇦

Cape Town, South Africa

Corporació Sanitària Parc Taulí

🇪🇸

Sabadell, Barcelona, Spain

Fundación Hospital Alcorcón

🇪🇸

Alcorcón, Madrid, Spain

Hospital Fundació Puigvert

🇪🇸

Barcelona, Spain

Hospital San Pedro de Alcántara

🇪🇸

Cáceres, Spain

Hospital Universitario Virgen de la Victoria | Cardiology Department

🇪🇸

Málaga, Spain

H Virgen del Rocio |Cardiology|AF|Stroke prevention

🇪🇸

Sevilla, Spain

Kaohsiung Medical University Chung-Ho Memorial Hospital

🇨🇳

Kaohsiung City, Kaohsiung, Taiwan

Changhua Christian Hospital

🇨🇳

Changhua, Taiwan

Taichung Veterans General Hospital

🇨🇳

Taichung, Taiwan

National Cheng Kung University Hospital

🇨🇳

Tainan, Taiwan

Taipei Veterans General Hospital

🇨🇳

Taipei, Taiwan

CNE "Clinical Center of Oncology, Hematology, Transplantology and Palliative Care of the Cherkasy Regional Council"

🇺🇦

Cherkasy, Ukraine

City Dnipropetrovsk Multi- field Clinical Hosp. 4 DSMA

🇺🇦

Dnipro, Ukraine

Kyiv City Hospital #3 - Department of Urology

🇺🇦

Kyiv, Ukraine

Kyiv Regional Oncological Dispensary

🇺🇦

Kyiv, Ukraine

Nepean Hospital

🇦🇺

Kingswood, New South Wales, Australia

Northern Cancer Institute

🇦🇺

St Leonards, New South Wales, Australia

Macquarie University Hospital

🇦🇺

Sydney, New South Wales, Australia

Cancer Research South Australia

🇦🇺

Adelaide, South Australia, Australia

Peninsula Oncology Centre

🇦🇺

Frankston, Victoria, Australia

Austin Health

🇦🇺

Heidelberg, Victoria, Australia

Assistência Multidisciplinar em Oncologia (AMO)

🇧🇷

Salvador, Bahia, Brazil

Hosp. Araujo Jorge da Associação de Combate ao Câncer

🇧🇷

Goiânia, Goiás, Brazil

Hospital da Universidade Federal de Minas Gerais

🇧🇷

Belo Horizonte, Minas Gerais, Brazil

Cetus Oncologia Hospital Dia

🇧🇷

Belo Horizonte, Minas Gerais, Brazil

Liga Paranaense de Combate ao Cancer-Hosp Erasto Gaertner

🇧🇷

Curitiba, Parana, Brazil

Liga Norte Riograndense Contra o Cancer | Centro de Pesquisa Clínica

🇧🇷

Natal, Rio Grande Do Norte, Brazil

Unidade de Pesquisas Clinicas em Oncologia

🇧🇷

Pelotas, Rio Grande Do Sul, Brazil

Irmandade da Santa Casa de Misericordia de Porto Alegre | Hospital Sao Francisco - Centro Medico Pesquisa Clinica Cardiologia

🇧🇷

Porto Alegre, Rio Grande Do Sul, Brazil

Hospital Mae de Deus

🇧🇷

Porto Alegre, Rio Grande Do Sul, Brazil

FZ Pesquisa e Servicos em Cardiologia | Porto Alegre, Brazil

🇧🇷

Porto Alegre, Rio Grande Do Sul, Brazil

Fundacao Pio XII - Hospital de Cancer de Barretos

🇧🇷

Barretos/SP, Sao Paulo, Brazil

Hospital de Base | Integrated Research Center

🇧🇷

São José do Rio Preto, Sao Paulo, Brazil

Urobrasil

🇧🇷

São Paulo, Sao Paulo, Brazil

IBCC - Instituto Brasileiro de Controle do Cancer

🇧🇷

São Paulo, Sao Paulo, Brazil

Inst. de Assistência Médica ao Sérvidor Público Estadual

🇧🇷

São Paulo, Sao Paulo, Brazil

Instituto COI de Educação e Pesquisa

🇧🇷

Rio de Janeiro, Brazil

G. Kenneth Jansz Medicine Professional Corporation

🇨🇦

Burlington, Ontario, Canada

Centre de Recherche du Centre Hospitalier de l'Universite de Montreal (CRCHUM)

🇨🇦

Montreal, Quebec, Canada

Centro de Investigación Clínica del Sur

🇨🇱

Temuco, Araucanía, Chile

Centro de Estudios Clínicos SAGA SpA

🇨🇱

Providencia, Santiago, Chile

OncoCentro

🇨🇱

Viña del Mar, Valparaíso, Chile

Fundación Arturo López Perez

🇨🇱

Santiago, Chile

Oncovida

🇨🇱

Santiago, Chile

Hospital Clínico de la Pontificia Univ. Católica de Chile

🇨🇱

Santiago, Chile

UROMED

🇨🇱

Santiago, Chile

Anhui Provincial Hospital

🇨🇳

Hefei City, Anhui Province, Anhui, China

Beijing Hospital

🇨🇳

Beijing, Beijing, China

Sun Yat-sen University Cancer Center

🇨🇳

Guangzhou, Guangdong, China

Guangzhou First People Hospital

🇨🇳

Guangzhou, Guangdong, China

Cancer Hospital Chinese Academy of Medical Sciences, Shenzhen Center

🇨🇳

Shenzhen, Guangdong, China

Tongji Hosp. of Tongji Med Coll, Huazhong Uni of Sci & Tech.

🇨🇳

Wuhan, Hubei, China

Zhongnan hospital ,Wuhan University

🇨🇳

Wuhan, Hubei, China

Hubei Cancer Hospital

🇨🇳

Wuhan, Hubei, China

Hunan Cancer Hospital

🇨🇳

Changsha, Hunan, China

NJ Drum Tower Hospital, the Affil Hos of NJ Univ Med School

🇨🇳

Nanjing, Jiangsu, China

1st Hospital of Jilin University

🇨🇳

Changchun, Jilin, China

Liaoning Cancer Hospital and Institute

🇨🇳

Shengyang, Liaoning, China

Yantai Yuhuangding Hospital

🇨🇳

Yantai, Shandong, China

The First Affiliated Hospital of Xi'an Jiaotong University

🇨🇳

Xi'an, Shanxi, China

SichuanAcademyofMedicalSciences&SichuanProvincialPeople'sHos

🇨🇳

Chengdu, Sichuan, China

Sichuan University West China Hospital

🇨🇳

Chengdu, Sichuan, China

The 1st Affiliated Hospital of Zhejiang University

🇨🇳

Hangzhou, Zhejiang, China

ZheJiang Provincial People's Hospital

🇨🇳

Hangzhou, Zhejiang, China

Ningbo First Hospital

🇨🇳

Ningbo, Zhejiang, China

The First Affiliated Hospital of Wenzhou Medical University

🇨🇳

Wenzhou, Zhejiang, China

Cancer Hospital, Chinese Academy of Medical Sciences

🇨🇳

Beijing, China

Beijing Cancer Hospital

🇨🇳

Beijing, China

Mahatma Gandhi Cancer Hospital & Research Institute

🇮🇳

Vishakapatnam, Andhra Pradesh, India

The Gujarat Cancer & Research Institute

🇮🇳

Ahmedabad, Gujarat, India

HCG Cancer Centre - Ahmedabad

🇮🇳

Ahmedabad, Gujarat, India

Cancer Care Clinic - Vadodara

🇮🇳

Vadodara, Gujarat, India

K.L.E.S. Dr. Prabhakar Kore Hospital & Medical Research Centre

🇮🇳

Belgaum, Karnataka, India

Healthcare Global Enterprises Ltd

🇮🇳

Bengaluru, Karnataka, India

Amrita Institute of Medical Sciences

🇮🇳

Kochi, Kerala, India

Regional Cancer Centre - Thiruvananthapuram

🇮🇳

Thiruvananthapuram, Kerala, India

Marathwada Regional Cancer Centre and Research Institute

🇮🇳

Aurangabad, Maharashtra, India

Jaslok Hospital and Research Centre

🇮🇳

Mumbai, Maharashtra, India

Curie Manavata Cancer Centre

🇮🇳

Nashik, Maharashtra, India

Jehangir Hospital

🇮🇳

Pune, Maharashtra, India

All India Institute of Medical Sciences

🇮🇳

Bhubaneswar, Odisha, India

Sparsh Hospital & Critical Care

🇮🇳

Bhubaneswar, Orissa, India

Jawaharlal Institute Of Postgraduate Medical Education and R

🇮🇳

Gorimedu, Pondicherry, India

Sawami Man Singh (SMS) Medical College & Attached Hospitals

🇮🇳

Jaipur, Rajasthan, India

Apollo Speciality Hospitals

🇮🇳

Madurai, Tamil Nadu, India

Meenakshi Mission Hospital & Research Centre

🇮🇳

Madurai, Tamil Nadu, India

© Copyright 2025. All Rights Reserved by MedPath