MedPath

Safety and Efficacy Trial of BHV3000 (Rimegepant) 75 mg for the Acute Treatment of Migraine

Phase 3
Completed
Conditions
Acute Migraine
Interventions
Drug: Placebo
Registration Number
NCT04574362
Lead Sponsor
Pfizer
Brief Summary

This trial is to determine whether BHV3000 (rimegepant) 75mg is safe and effictive as a treatment for acute migraine in Chinese and Korean patients

Detailed Description

Biohaven Pharmaceuticals, Inc. is the agent for BioShin Limited, the sponsor of the studies in China and Korea.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
1648
Inclusion Criteria

Subject has at least 1 year history of migraines (with or without aura), consistent with a diagnosis according to the International Classification of Headache Disorder, 3rd Edition, Beta version including the following:

  1. Migraine attacks present for more than 1 year with the age of onset prior to 50 years of age
  2. Migraine attacks, on average, lasting about 4-72 hours if untreated
  3. Not more than 8 attacks of moderate to severe intensity per month within the last 3 months
  4. Consistent migraine headaches of at least 2 migraine headache attacks of moderate or severe intensity in each of the 3 months prior to the Screening Visit and maintains this requirement during the Screening period
  5. Less than 15 days with headache (migraine or non-migraine) per month in each of the 3 months prior to the Screening Visit and maintains this requirement during the Screening Period.
  6. Subjects on prophylactic migraine medication are permitted to remain on therapy provided they have been on a stable dose for at least 3 months prior to screening visit and the dose is not expected to change during the course of the study.
  7. Subjects with contraindications for use of triptans may be included provided they meet all other study entry criteria.

Key

Exclusion Criteria
  1. Subject with a history of HIV disease
  2. Subject history with current evidence of uncontrolled, unstable or recently diagnosed cardiovascular disease, such as ischemic heart disease, coronary artery vasospasm, and cerebral ischemia. subjects with Myocardial Infarction (MI), Acute Coronary Syndrome (ACS), Percutaneous Coronary Intervention (PCI), cardiac surgery, stroke or transient ischemic attack (TIA) during the 6 months prior to screening
  3. Uncontrolled hypertension (high blood pressure), or uncontrolled diabetes (however subjects can be included who have stable hypertension and/or diabetes for at least 3 months prior to being enrolled)
  4. Subject has a current diagnosis of major depression, other pain syndromes, psychiatric conditions (e.g., schizophrenia), dementia, or significant neurological disorders (other than migraine) that, in the Investigator's opinion might interfere with study assessments.
  5. Subject has a history of gastric, or small intestinal surgery (including Gastric Bypass, Gastric Banding, Gastric Sleeve, Gastric Balloon, etc.), or has disease that causes malabsorption
  6. The subject has a history of current or evidence of any significant and/ or unstable medical conditions (e.g., history of congenital heart disease or arrhythmia, known suspected infection, hepatitis B or C, or cancer) that, in the investigator's opinion, would expose them to undue risk of a significant adverse event (AE) or interfere with assessments of safety or efficacy during the course of the trial.
  7. History of, treatment for, or evidence of, alcohol or drug abuse within the past 12 months or subjects who have met DSM-V criteria for any significant substance use disorder within the past 12 months from the date of the screening visit.
  8. Subjects are excluded if they have previously participated in any study of rimegepant or other experimental CGRP-antagonist study, or have been prescribed CGRP-antibodies within the last 6 months
  9. Participation in any other investigational clinical trial while participating in this clinical trial

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlaceboMatching placebo
Rimegepant 75mgRimegepantOne 75mg oral disintegration tablet
Primary Outcome Measures
NameTimeMethod
Percentage of Participants Who Had Freedom From Most Bothersome Symptoms (MBS) at 2 Hours Post-dose2 hours post-dose

MBS included nausea, phonophobia or photophobia. MBS were measured using a binary scale as 0= absent, 1= present. Participants who had score of 0 (MBS absent) were considered to have freedom from MBS. Exact 95% CI was based on Clopper-Pearson method.

Percentage of Participants Who Had Freedom From Pain at 2 Hours Post-dose2 hours post-dose

Pain was measured on a 4-point Likert scale, with following scores: 0= none, 1= mild, 2= moderate, 3= severe. Participants with score of 0 (no pain) were considered to have freedom from pain. Exact 95 percent (%) confidence interval (CI) was based on Clopper-Pearson method.

Secondary Outcome Measures
NameTimeMethod
Percentage of Participants Who Sustained Pain Freedom From 2 to 48 Hours Post-dose2 to 48 hours post-dose

Pain was measured on a 4-point Likert scale, with following scores: 0= none, 1= mild, 2= moderate, 3= severe. Participants with score of 0 (with no pain) through 2 to 48 hours post-dose were considered to have sustained pain freedom. Exact 95% CI was based on Clopper-Pearson method.

Percentage of Participants Who Had Freedom From Pain at 15, 30, 45, 60 and 90 Minutes Post-dose15, 30, 45, 60 and 90 minutes post-dose

Pain was measured on a 4-point Likert scale, with following scores: 0= none, 1= mild, 2= moderate, 3= severe. Percentage of participants who reported a pain level of moderate or severe just before taking study treatment and then reported a pain level of none at the specified timepoints. Exact 95% CI was based on Clopper-Pearson method.

Percentage of Participants Who Had Freedom From MBS at 15, 30, 45, 60 and 90 Minutes Post-dose15, 30, 45, 60 and 90 minutes post-dose

MBS included nausea, phonophobia or photophobia. MBS were measured using a binary scale as 0= absent, 1= present. Participants who had score of 0 (MBS absent) were considered to have freedom from MBS at the specified timepoints. Exact 95% CI was based on Clopper-Pearson method.

Percentage of Participants With Pain Relief at 2 Hours Post-dose2 hours post-dose

Pain was measured on a 4-point Likert scale, with following scores: 0= none, 1= mild, 2= moderate, 3= severe. Participants who reported a pain level of moderate or severe at baseline and then reported a pain level of none or mild at 2 hours post-dose, were considered to have pain relief. Exact 95% CI was based on Clopper-Pearson method.

Percentage of Participants Who Functioned Normally at 2 Hours Post-dose2 hours post-dose

Participants rated the level of disability they perceived as a result of their migraine in performing normal actions using following level of severity: normal function, mild impairment, severe impairment, or required bedrest. This outcome measure was analyzed only among those participants who reported any impairment at baseline. Percentage of participants with a response of "normal function" at the 2 hours post-dose were reported in this outcome measure.

Percentage of Participants Who Used Rescue Medication Within 24 Hours Post-dose24 hours post-dose

Percentage of participants who used rescue medications within 24 hours of administration of study drug were reported in this outcome measure. Exact 95% CI was based on Clopper-Pearson method.

Percentage of Participants Who Sustained Pain Freedom From 2 to 24 Hours Post-dose2 to 24 hours post-dose

Pain was measured on a 4-point Likert scale, with following scores: 0= none, 1= mild, 2= moderate, 3= severe. Participants with score of 0 (with no pain) through 2 to 24 hours post-dose were considered to have sustained pain freedom. Exact 95% CI was based on Clopper-Pearson method.

Percentage of Participants With Pain Relapse2 Hours to 48 Hours Post-dose

Pain was measured on a 4-point Likert scale, with following scores: 0= none, 1= mild, 2= moderate, 3= severe. This outcome measure was analyzed only in those participants who were pain free at 2 hours post-dose. Percentage of participants who were pain free at 2 hours post-dose and then had a migraine of any pain severity (score 2 or 3 on the 4-point scale) within 48 hours after administration of study drug were considered to have pain relapse. Exact 95% CI was based on Clopper-Pearson method.

Trial Locations

Locations (90)

1st Hospital of Jilin University

🇨🇳

Changchun, Jilin, China

Shandong Provincial Qianfoshan Hospital

🇨🇳

Jinan, Shandong, China

Kangdong Sacred Heart Hospital

🇰🇷

Seoul, Korea, Republic of

Severance Hospital

🇰🇷

Seoul, Korea, Republic of

Kangbuk Samsung Hospital

🇰🇷

Seoul, Korea, Republic of

Samsung Medical Center

🇰🇷

Seoul, Korea, Republic of

Chungnam National University Hospital

🇰🇷

Daejeon, Korea, Republic of

Ewha Womans University Medical Center

🇰🇷

Seoul, Korea, Republic of

Seoul National University Bundang Hospital

🇰🇷

Seongnam-si, Gyeonggi-do, Korea, Republic of

Nowon Eulji Medical Center

🇰🇷

Seoul, Korea, Republic of

Korea University Guro Hospital

🇰🇷

Seoul, Korea, Republic of

Dongtan Sacred Heart Hospital

🇰🇷

Hwaseong-si, Gyeonggi-do, Korea, Republic of

Baoji Central Hospital

🇨🇳

Baoji, Shaanxi, China

The First Affiliated Hospital of Bengbu Medical College

🇨🇳

Bengbu, Anhui, China

Anhui provincal Hospital

🇨🇳

Hefei, Anhui, China

Lu'An People's Hospital

🇨🇳

Lu'an, Anhui, China

Wuhan Third Hospital

🇨🇳

Wuhan, Hubei, China

The People's Hospital of Xuancheng City

🇨🇳

Xuancheng, Anhui, China

Chinese PLA General Hospital

🇨🇳

Beijing, Beijing, China

Chongqing Emergency Medical Center

🇨🇳

Chongqing, Chongqing, China

The First Affiliated Hospital of Chongqing Medical University

🇨🇳

Chongqing, Chongqing, China

Chonggang General Hospital

🇨🇳

Chongqing, Chongqing, China

Chongqing Three Gorges Central Hospital

🇨🇳

Chongqing, Chongqing, China

Fujian medical University Union Hospital

🇨🇳

Fuzhou, Fujian, China

The 900th Hospital of Joint Logistics Support Force, PLA

🇨🇳

Fuzhou, Fujian, China

Sun Yat-Sen Memorial Hospital of Zhongshan University

🇨🇳

Guangzhou, Guangdong, China

Lanzhou University Second Hospital

🇨🇳

Lanzhou, Gansu, China

The First Affiliated Hospital of Hainan Medical College

🇨🇳

Haikou, Hainan, China

Henan University of Science and Technology First Affiliated Hospital

🇨🇳

Luoyang, Henan, China

Henan Provincial People's Hospital

🇨🇳

Zhengzhou, Henan, China

Zhengzhou People's Hospital

🇨🇳

Zhengzhou, Henan, China

The First Affiliated Hospital of Zhengzhou University

🇨🇳

Zhengzhou, Henan, China

Wuhan Fourth hospital

🇨🇳

Wuhan, Hubei, China

Renmin Hospital Of Wuhan University

🇨🇳

Wuhan, Hubei, China

Huanggang Central Hospital

🇨🇳

Huanggang, Hubei, China

Changsha Central Hospital

🇨🇳

Changsha, Hunan, China

The Second Xiangya Hospital Of Central South University

🇨🇳

Changsha, Hunan, China

The Central Hospital of Shaoyang

🇨🇳

Shaoyang, Hunan, China

The First People's Hospital of Yueyang

🇨🇳

Yueyang, Hunan, China

Zhuzhou Central Hospital

🇨🇳

Zhuzhou, Hunan, China

Zigong First People's Hospital

🇨🇳

Sichuan, Igong, China

The first affiliated hospital of Baotou medical college of Inner Mongolia university of science and technology

🇨🇳

Baotou, Inner Mongolia, China

Affiliated Hospital of Chifeng University

🇨🇳

Chifeng, Inner Mongolia, China

Inner Mongolia People's Hospital

🇨🇳

Hohhot, Inner Mongolia, China

The Second People's Hospital of Lianyungang

🇨🇳

Lianyungang, Jiangsu, China

Nanjing Drum Tower Hospital

🇨🇳

Nanjing, Jiangsu, China

Zhongda Hospital Southeast University

🇨🇳

Nanjing, Jiangsu, China

Wuxi people's Hospital

🇨🇳

Wuxi, Jiangsu, China

The Affiliated Hospital of Jiangsu University

🇨🇳

Zhenjiang, Jiangsu, China

The Second Affiliated Hospital of Nanjing Medical University

🇨🇳

Nanjing, Jiangsu, China

Sir Run Run Hospital, Nanjing Medical University

🇨🇳

Nanjing, Jiangsu, China

The Second Hospital of Jilin University

🇨🇳

Changchun, Jilin, China

General Hospital of Ningxia Medical Hospital

🇨🇳

Yinchuan, Ning Xia, China

The First People's Hospital of Yinchuan

🇨🇳

Yinchuan, Ningxia, China

General Hospital of Northern Theater Command

🇨🇳

Shenyang, Liaoning, China

Yan'an University Xianyang Hospital Co., Ltd

🇨🇳

Xianyang, Shaanxi, China

Affiliated Hospital of Jining Medical University

🇨🇳

Jining, Shandong, China

Qingdao Central Hospital

🇨🇳

Qingdao, Shandong, China

Zaozhuang Municipal Hospital

🇨🇳

Zaozhuang, Shandong, China

Xi'an Gaoxin Hospital Co., Ltd

🇨🇳

Xi'an, Shaanxi, China

The First Affiliated Hospital of Xi'an Medical University

🇨🇳

Xi'an, Shaanxi, China

Heping Hospital Affiliated to Changzhi Medical College

🇨🇳

Changzhi, Shanxi, China

The Second Hospital of Shanxi Medical University

🇨🇳

Taiyuan, Shanxi, China

Shanghai East Hospital

🇨🇳

Shanghai, Shanghai, China

West China Hospital of Sichuan University

🇨🇳

Chengdu, Sichuan, China

Nankai University, Tianjin Union Medical Center

🇨🇳

Tianjin, Tianjin, China

Tianjin Huanhu Hospital

🇨🇳

Tianjin, Tianjin, China

The Fifth Affiliated Hospital of Xinjiang Medical University

🇨🇳

Xinjiang, Uramqi, China

People's Hospital of Xinjiang Uygur Autonomous Region

🇨🇳

Xinjiang, Wulumuqi, China

The Second Affiliated Hospital of Xinjiang Medical University

🇨🇳

Xinjiang, Wulumuqi, China

Ruian People's Hospital

🇨🇳

Rui'an, Zhejiang, China

The Second Hospital of Anhui Medical University

🇨🇳

Hefei, Anhui, China

Peking University People's Hospital

🇨🇳

Beijing, Beijing, China

Beijing Friendship Hospital,Capital Medical University

🇨🇳

Beijing, Beijing, China

Cangzhou Central Hospital

🇨🇳

Cangzhou, Hebei, China

Hainan General Hospital

🇨🇳

Haikou, Hainan, China

Taihe Hospital

🇨🇳

Shiyan, Hubei, China

Jingzhou Central Hospital

🇨🇳

Jingzhou, Hubei, China

The Third Xiangya Hospital Of Central South University

🇨🇳

Changsha, Hunan, China

Nanjing Brain Hospital

🇨🇳

Nanjing, Jiangsu, China

Wuxi Integrated Traditional Chinese and Western Medicine Hospital

🇨🇳

Wuxi, Jiangsu, China

The First Affiliated Hospital With Nanjing Medical University

🇨🇳

Nanjing, Jiangsu, China

The Second Affiliated Hospital of Xi'an Jiaotong University

🇨🇳

Xi'an, Shaanxi, China

Shaanxi Provincial People' Hospital

🇨🇳

Xi'an, Shaanxi, China

Liaocheng People's Hospital

🇨🇳

Liaocheng, Shandong, China

Chuncheon Sacred Heart Hospital

🇰🇷

Chuncheon, Gangwon, Korea, Republic of

Inje University Ilsan Paik Hospital

🇰🇷

Goyang-si, Gyeonggi-do, Korea, Republic of

The Second Affiliated hospital of Kunming Medical University

🇨🇳

Kunming, Yunnan, China

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

First Hospital of Shanxi Medical University

🇨🇳

Taiyuan, Shanxi, China

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