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Relative Bioavailability of BI 10773 and Glimepiride in Healthy Male Volunteers

Phase 1
Completed
Conditions
Healthy
Interventions
Registration Number
NCT02172261
Lead Sponsor
Boehringer Ingelheim
Brief Summary

The objective was to investigate whether there was a drug-drug interaction between BI 10773 and glimepiride when co-administered. Therefore, the relative bioavailabilities of BI 10773 and glimepiride were determined when both drugs were given in combination compared to multiple oral doses of BI 10773 once daily alone and a single oral dose of glimepiride given alone.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
16
Inclusion Criteria
  • Healthy male volunteers according to the following criteria: Based upon a complete medical history, including the physical examination, vital signs (BP, PR), 12-lead ECG, clinical laboratory tests
  • Age 18 to 50 years (incl.)
  • BMI (Body Mass Index) 18.5 to 29.9 kg/m2 (incl.)
  • Signed and dated written informed consent prior to admission to the study in accordance with GCP (Good Clinical Practice) and the local legislation
Exclusion Criteria
  • Any finding of the medical examination (including BP (Blood Pressure, PR (Pulse Rate) and ECG (Electrocardiogram)) deviating from normal and of clinical relevance
  • Any evidence of a clinically relevant concomitant disease
  • Gastrointestinal, hepatic, renal, respiratory, cardiovascular, metabolic, immunological or hormonal disorders
  • Surgery of the gastrointestinal tract (except appendectomy)
  • Diseases of the central nervous system (such as epilepsy) or psychiatric disorders or neurological disorders
  • History of relevant orthostatic hypotension, fainting spells or blackouts
  • Chronic or relevant acute infections
  • History of relevant allergy/hypersensitivity (including allergy to drug or its excipients)
  • Intake of drugs with a long half-life (> 24 hours) within at least one month or less than 10 half-lives of the respective drug prior to administration or during the trial
  • Participation in another trial with an investigational drug within two months prior to administration or during the trial
  • Smoker (> 10 cigarettes or > 3 cigars or > 3 pipes/day)
  • Inability to refrain from smoking on trial days
  • Alcohol abuse (more than 30 g/day)
  • Drug abuse
  • Blood donation (more than 100 mL within four weeks prior to administration or during the trial)
  • Excessive physical activities (within one week prior to administration or during the trial)
  • Any laboratory value outside the reference range that is of clinical relevance
  • Inability to comply with dietary regimen of trial site
  • Glucose-6-phosphate dehydrogenase deficiency

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Sequence ABCBI 107731. Treatment A: BI 10773 once daily from day 1 to 5 2. Treatment B: BI 10773 and glimepiride once on day 1 3. Treatment C: Glimepiride once on day 1
Sequence ABCGlimepiride1. Treatment A: BI 10773 once daily from day 1 to 5 2. Treatment B: BI 10773 and glimepiride once on day 1 3. Treatment C: Glimepiride once on day 1
Sequence CABBI 107731. Treatment C: Glimepiride once on day 1 2. Treatment A: BI 10773 once daily from day 1 to 5 3. Treatment B: BI 10773 and glimepiride once on day 1
Sequence CABGlimepiride1. Treatment C: Glimepiride once on day 1 2. Treatment A: BI 10773 once daily from day 1 to 5 3. Treatment B: BI 10773 and glimepiride once on day 1
Primary Outcome Measures
NameTimeMethod
AUCτ,ss (area under the concentration-time curve of the analyte in plasma at steady state over a uniform dosing interval τ) of BI 10773up to 5 days
Cmax,ss (maximum measured concentration of the analyte in plasma at steady state over a uniform dosing interval τ) of BI 10773up to 5 days
AUC0-∞ (area under the concentration-time curve of the analyte in plasma over the time interval from 0 extrapolated to infinity) of glimepirideup to 4 days
Cmax (maximum measured concentration of the analyte in plasma) of glimepirideup to 4 days
Secondary Outcome Measures
NameTimeMethod
λz (terminal rate constant in plasma) of glimepirideup to 4 days
AUC0-tz (area under the concentration-time curve of the analyte in plasma over the time interval from 0 to the time of the last quantifiable data point) of glimepirideup to 4 days
tmax (time from dosing to the maximum concentration of the analyte in plasma) of glimepirideup to 4 days
t½ (terminal half-life of the analyte in plasma) of glimepirideup to 4 days
MRTpo (mean residence time of the analyte in the body after po administration) of glimepirideup to 4 days
CL/F (apparent clearance of the analyte in the plasma after extravascular administration) of glimepirideup to 4 days
Vz/F (apparent volume of distribution during the terminal phase λz following an extravascular dose) of glimepirideup to 4 days
MRTpo,ss (mean residence time of the analyte in the body at steady state after oral administration) of BI 10773up to 5 days
CL/F,ss (apparent clearance of the analyte in the plasma after extravascular administration at steady state) of BI 10773up to 5 days
Vz/F,ss (apparent volume of distribution during the terminal phase λz at steady state following extravascular administration) of BI 10773up to 5 days
Aet1-t2,ss (amount of analyte eliminated in urine at steady state over a uniform dosing interval τ) of BI 107731 hour pre-dose and 0-2, 2-4, 4-8, 8-12, 12-24 after administration on day 1 and 5
fet1-t2,ss (fraction of analyte excreted unchanged in urine at steady state over a uniform dosing interval τ) of BI 107731 hour pre-dose and 0-2, 2-4, 4-8, 8-12, 12-24 after administration on day 1 and 5
CLR,ss (renal clearance of the analyte at steady state) of BI 107731 hour pre-dose and 0-2, 2-4, 4-8, 8-12, 12-24 after administration on day 1 and 5
UGE0-24 (Urinary glucose excretion of the analyte in urine over the time interval from time zero to 24 h)1 hour pre-dose and 0-2, 2-4, 4-8, 8-12, 12-24 after administration on days 1 and 5
Number of patients with abnormal findings in physical examinationBaseline and within 3-14 days after last glimepiride administration
Number of patients with clinically significant changes in vital signs (blood pressure, pulse rate)Baseline, day 1 and within 3-14 days after last glimepiride administration
Number of patients with abnormal findings in 12-lead ECG (electrocardiogram)Baseline, day 1 and within 3-14 days after last glimepiride administration
Number of patients with abnormal findings in clinical laboratory testsBaseline, day 1,4 and within 3-14 days after last glimepiride administration
Number of patients with adverse eventsUp to 34 days
Assessment of tolerability by investigator on a 4-point scaleWithin 3-14 days after last glimepiride administration
Number of patients with abnormal findings in glucose bedside testsPre-dose and 1, 2, 4, 7, 10, 14, 24 hours after glimepiride administration on day 1
tmax,ss (time from last dosing to maximum concentration of the analyte in plasma at steady state over a uniform dosing interval τ) of BI 10773up to 5 days
Aet1-t2 (amount of analyte eliminated in urine over the time interval from t1 to t2) of glimepiride1 hour pre-dose and 0-2, 2-4, 4-8, 8-12, 12-24 after administration on day 1
fet1-t2 (fraction of analyte excreted unchanged in urine over the time interval from t1 to t2) of glimepiride1 hour pre-dose and 0-2, 2-4, 4-8, 8-12, 12-24 after administration on day 1
CLR (renal clearance of the analyte) of glimepiride1 hour pre-dose and 0-2, 2-4, 4-8, 8-12, 12-24 after administration on day 1
λz,ss (terminal rate constant of analyte in plasma at steady-state) of BI 10773up to 5 days
t½,ss (terminal half-life of analyte in plasma at steady-state) of BI 10773up to 5 days
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