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A Study of the Safety of Oral Elsubrutinib Capsules and Oral Upadacitinib Tablets Given Alone or in Combination (ABBV-599) for Adult Participants With Moderately to Severely Active Systemic Lupus Erythematosus to Assess Change in Disease State

Phase 2
Completed
Conditions
Systemic Lupus Erythematosus (SLE)
Interventions
Registration Number
NCT04451772
Lead Sponsor
AbbVie
Brief Summary

Systemic Lupus Erythematosus (SLE) is an immune-mediated disease associated with inflammation of multiple organ systems. This study will evaluate how well elsubrutinib and upadacitinib given alone or as the ABBV-599 combination (elsubrutinib/upadacitinib) works within the body, in participants who completed study M19-130. This study will assess the change in disease symptoms.

ABBV-599 is an investigational drug being developed for the treatment of Systemic Lupus Erythematosus (SLE). This study is "double-blinded", which means that neither the trial participants nor the study doctors will know who will be given which study drug. Study doctors put the participants into 1 of 4 groups called treatment arms. Each group receives a different treatment. Adult participants with a diagnosis of SLE will be enrolled. Around 260 participants will be enrolled in the study in approximately 100 sites worldwide.

Participants will receive the following for up to 56 weeks:

Participants will receive oral elsubrutinib capsules and/or oral upadacitinib tablets once daily for up to 56 weeks. Participants who were receiving elsubrutinib and/or upadacitnib in M19-130 will continue to receive the same treatment in this study. Participants who were receiving placebo in M19-130 will be re-randomized to one of the 2 combination treatment arms in this study.

Arm 1: Elsubrutinib Dose A and Upadacitinib Dose A Arm 2: Elsubrutinib Dose A and Upadacitinib Dose B

There may be higher burden for participants in this trial compared to their standard of care. Participants will attend monthly visits during the course of the study at a hospital or clinic. The effect of the treatment will be checked by medical assessments, blood tests, checking for side effects and completing questionnaires.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
185
Inclusion Criteria
  • Completed Study M19-130 (i.e., the randomized controlled trial of elsubrutinib, upadacitinib, and ABBV-599 [elsubrutinib/upadacitinib] combination or matching placebo) and will not have developed any laboratory or clinical discontinuation criteria as defined in that study.
  • On stable background treatment for SLE throughout the study.
Exclusion Criteria
  • Active, chronic, or recurrent viral, or bacterial infection.
  • Active tuberculosis (TB)
  • History of gastrointestinal (GI) perforation, diverticulitis, or a significantly increased risk for GI perforation per investigator assessment.
  • Participant require vaccination with live vaccine during study participation.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
ABBV-599 High Dose (Elsubrutinib 60 mg/upadacitinib 30 mg) -> ABBV-599 High DoseElsubrutinibParticipants received elsubrutinib 60 mg capsules once a day by mouth and upadacitinib 30 mg film-coated tablets once a day by mouth for 48 weeks in Study M19-130. Participants continued on this regimen in the current study (M20-186) for up to 56 weeks.
Elsubrutinib placebo/upadacitinib 30 mg -> Elsubrutinib placebo/upadacitinib 30 mgPlacebo for ElsubrutinibParticipants received placebo capsules for elsubrutinib once a day by mouth and upadacitinib 30 mg film-coated tablets once a day by mouth for 48 weeks in Study M19-130. Participants continued on this regimen in the current study (M20-186) for up to 56 weeks.
ABBV-599 Low Dose (Elsubrutinib 60 mg/upadacitinib 15 mg) -> ABBV-599 Low DoseUpadacitinibParticipants received elsubrutinib 60 mg capsules once a day by mouth and upadacitinib 15 mg film-coated tablets once a day by mouth for 48 weeks in Study M19-130. Participants continued on this regimen in the current study (M20-186) for up to 56 weeks.
ABBV-599 High Dose (Elsubrutinib 60 mg/upadacitinib 30 mg) -> ABBV-599 High DoseUpadacitinibParticipants received elsubrutinib 60 mg capsules once a day by mouth and upadacitinib 30 mg film-coated tablets once a day by mouth for 48 weeks in Study M19-130. Participants continued on this regimen in the current study (M20-186) for up to 56 weeks.
Elsubrutinib placebo/upadacitinib 30 mg -> Elsubrutinib placebo/upadacitinib 30 mgUpadacitinibParticipants received placebo capsules for elsubrutinib once a day by mouth and upadacitinib 30 mg film-coated tablets once a day by mouth for 48 weeks in Study M19-130. Participants continued on this regimen in the current study (M20-186) for up to 56 weeks.
Elsubrutinib placebo/upadacitinib placebo -> ABBV-599 High DoseUpadacitinibParticipants received placebo capsules for elsubrutinib once a day by mouth and placebo film-coated tablets for upadacitinib once a day by mouth for 48 weeks in Study M19-130. Participants received elsubrutinib 60 mg capsules once a day by mouth and upadacitinib 30 mg film-coated tablets once a day in the current study (M20-186) for up to 56 weeks.
Elsubrutinib 60 mg/upadacitinib placebo -> Elsubrutinib 60 mg/upadacitinib placeboPlacebo for UpadacitinibParticipants received elsubrutinib 60 mg capsules once a day by mouth and placebo film-coated tablets for upadacitinib once a day by mouth for 48 weeks in Study M19-130. Participants continued on this regimen in the current study (M20-186) for up to 56 weeks.
Elsubrutinib placebo/upadacitinib placebo -> ABBV-599 Low DoseUpadacitinibParticipants received placebo capsules for elsubrutinib once a day by mouth and placebo film-coated tablets for upadacitinib once a day by mouth for 48 weeks in Study M19-130. Participants received elsubrutinib 60 mg capsules once a day by mouth and upadacitinib 15 mg film-coated tablets once a day by mouth for 48 weeks in the current study (M20-186) for up to 56 weeks.
Elsubrutinib placebo/upadacitinib placebo -> ABBV-599 High DoseElsubrutinibParticipants received placebo capsules for elsubrutinib once a day by mouth and placebo film-coated tablets for upadacitinib once a day by mouth for 48 weeks in Study M19-130. Participants received elsubrutinib 60 mg capsules once a day by mouth and upadacitinib 30 mg film-coated tablets once a day in the current study (M20-186) for up to 56 weeks.
ABBV-599 Low Dose (Elsubrutinib 60 mg/upadacitinib 15 mg) -> ABBV-599 Low DoseElsubrutinibParticipants received elsubrutinib 60 mg capsules once a day by mouth and upadacitinib 15 mg film-coated tablets once a day by mouth for 48 weeks in Study M19-130. Participants continued on this regimen in the current study (M20-186) for up to 56 weeks.
Elsubrutinib 60 mg/upadacitinib placebo -> Elsubrutinib 60 mg/upadacitinib placeboElsubrutinibParticipants received elsubrutinib 60 mg capsules once a day by mouth and placebo film-coated tablets for upadacitinib once a day by mouth for 48 weeks in Study M19-130. Participants continued on this regimen in the current study (M20-186) for up to 56 weeks.
Elsubrutinib placebo/upadacitinib placebo -> ABBV-599 Low DoseElsubrutinibParticipants received placebo capsules for elsubrutinib once a day by mouth and placebo film-coated tablets for upadacitinib once a day by mouth for 48 weeks in Study M19-130. Participants received elsubrutinib 60 mg capsules once a day by mouth and upadacitinib 15 mg film-coated tablets once a day by mouth for 48 weeks in the current study (M20-186) for up to 56 weeks.
Primary Outcome Measures
NameTimeMethod
Number of Participants With Treatment-Emergent Adverse EventsFrom the first dose of study drug in Study M20-186 up to 30 days after the last dose of study drug, up to 442 days

An adverse event (AE) is defined as any untoward medical occurrence in a patient or clinical investigation participant administered a pharmaceutical product and which does not necessarily have a causal relationship with this treatment. A serious adverse event (SAE) is an event that results in death, is life-threatening, requires or prolongs hospitalization, results in a congenital anomaly, persistent or significant disability/incapacity or is an important medical event that, based on medical judgment, may jeopardize the participant and may require medical or surgical intervention to prevent any of the outcomes listed above. Treatment-emergent events (TEAEs) are defined as an adverse event with an onset date that is on or after the first dose of study drug from Study M20-186, and no more than 30 days after the last dose of study drug from Study M20-186. For more details on adverse events please see the Adverse Event section.

Secondary Outcome Measures
NameTimeMethod
Percentage of Participants Achieving Systemic Lupus Erythematosus (SLE) Responder Index (SRI)-4Baseline of Study M19-130 (Week 0), Weeks 56, 64, 72, 80, 88, 96, 104

SLE Responder Index (SRI)-4 is defined as follows with all criteria compared to Baseline in Study M19-130:

* ≥4-point reduction in Systemic Lupus Erythematosus Disease Activity Index 2000 (SLEDAI-2K) score

* No worsening of the overall condition (\< 0.3 point increase in Physician's Global Assessment \[PhGA\])

* No new British Isles Lupus Assessment Group (BILAG) A or more than 1 new BILAG B disease activity scores (i.e., no organ system changes from baseline B/C/D/E to A and no more than 1 organ system changes from baseline C/D/E to B). A letter score is assigned to each organ system with following indications: A = severe, B = moderate, C = mild, D = inactive with prior history, and E = inactive with no history.

Percentage of Participants Achieving British Isles Lupus Assessment Group (BILAG)-Based Combined Lupus Assessment (BICLA) ResponseBaseline of Study M19-130 (Week 0), Weeks 56, 64, 72, 80, 88, 96, 104

BICLA is a composite responder index. Achievement of BICLA response is defined as improvement in all initial A and B BILAG scores, with no more than one new BILAG B score without worsening of the overall condition (no worsening in Physician's Global Assessment \[PhGA\], \< 0.3 point increase) and no worsening of the Systemic Lupus Erythematosus Disease Activity Index 2000 (SLEDAI-2K) score.

Change From Baseline in Daily Prednisone Dose Over TimeBaseline of M19-130 (Week 0), Weeks 56, 64, 72, 80, 88, 96, 104

Participants'current use of steroid therapy was assessed at each study visit, and the amount of daily prednisone was documented.

Number of Flares Per Patient-year by Safety of Estrogens in Lupus Erythematosus National Assessment (SELENA) SLE Disease Activity Index (SLEDAI) Flare Index Through Week 104From Week 56 through Week 104

The SELENA SLEDAI flare index defines mild/moderate or severe SLE flares using the SLEDAI score, definitions of worsening signs and symptoms, treatment changes, and Physician's Global Assessment of Disease Activity.

Trial Locations

Locations (87)

Duplicate_AZ Arthritis and Rheumotology Research, PLLC /ID# 227833

🇺🇸

Phoenix, Arizona, United States

Duplicate_NYU Langone Health/NYU School of Medicine /ID# 245088

🇺🇸

New York, New York, United States

Duplicate_Peking Union Medical College Hospital /ID# 222950

🇨🇳

Beijing, Beijing, China

Duplicate_Arthritis & Rheumatic Disease Specialties /ID# 227828

🇺🇸

Aventura, Florida, United States

Duplicate_Centro de Investigacion en Reumatologia y Especialidades Medicas- CIRE /ID# 221884

🇨🇴

Bogota, Cundinamarca, Colombia

Healthy Medical Center S.A.S /ID# 221882

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Zipaquirá, Cundinamarca, Colombia

Duplicate_Centro Integral de Reumatologia del Caribe Circaribe SAS /ID# 221879

🇨🇴

Barranquilla, Atlantico, Colombia

Centro de Investigaciones Medicas Tucuman /ID# 221888

🇦🇷

San Miguel de Tucuman, Tucuman, Argentina

Investigaciones Clinicas Tucuman /ID# 221889

🇦🇷

San Miguel de Tucuman, Tucuman, Argentina

Rheumatology Research Unit Sunshine Coast /ID# 221816

🇦🇺

Maroochydore, Queensland, Australia

Emeritus Research /ID# 223027

🇦🇺

Camberwell, Victoria, Australia

Monash Medical Centre /ID# 221814

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Clayton, Victoria, Australia

UMHAT Sveti Ivan Rilski /ID# 223358

🇧🇬

Sofia, Bulgaria

Duplicate_Charite Universitaetsmedizin Berlin - Campus Mitte /ID# 222963

🇩🇪

Berlin, Germany

Duplicate_Debreceni Egyetem Klinikai Kozpont /ID# 222480

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Debrecen, Hajdu-Bihar, Hungary

Duplicate_Azienda Ospedaliero-Universitaria di Ferrara-Arcispedale Sant Anna /ID# 221919

🇮🇹

Cona, Ferrara, Italy

Duplicate_Hospital Universitario A Coruna - CHUAC /ID# 221993

🇪🇸

A Coruna, Spain

Duplicate_Manchester University NHS Foundation Trust /ID# 221861

🇬🇧

Manchester, United Kingdom

Wallace Rheumatic Studies Center, LLC /ID# 224374

🇺🇸

Beverly Hills, California, United States

Valerius Medical Group & Research Center /ID# 223922

🇺🇸

Los Alamitos, California, United States

East Bay Rheumatology Medical /ID# 225493

🇺🇸

San Leandro, California, United States

University of Colorado Hospital /ID# 245087

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Aurora, Colorado, United States

Millennium Research /ID# 233192

🇺🇸

Ormond Beach, Florida, United States

IRIS Research and Development, LLC /ID# 227814

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Plantation, Florida, United States

Deerbrook Medical Associates /ID# 227330

🇺🇸

Libertyville, Illinois, United States

Qualmedica Research, LLC /ID# 227817

🇺🇸

Evansville, Indiana, United States

The Center for Rheumatology and Bone Research /ID# 225479

🇺🇸

Wheaton, Maryland, United States

Beth Israel Deaconess Medical Center /ID# 222505

🇺🇸

Boston, Massachusetts, United States

June DO, PC /ID# 221841

🇺🇸

Lansing, Michigan, United States

STAT Research, Inc. /ID# 221840

🇺🇸

Vandalia, Ohio, United States

Allegheny Health Network Research Institute /ID# 245086

🇺🇸

Pittsburgh, Pennsylvania, United States

Dr. Ramesh Gupta /ID# 225524

🇺🇸

Memphis, Tennessee, United States

Tekton Research, Inc. /ID# 224411

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Austin, Texas, United States

Accurate Clinical Management /ID# 225509

🇺🇸

Houston, Texas, United States

SW Rheumatology Res. LLC /ID# 225485

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Mesquite, Texas, United States

Carilion Clinic /ID# 227832

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Roanoke, Virginia, United States

Hospital Militar Central Cirujano Mayor Dr. Cosme Argerich /ID# 222569

🇦🇷

Ciudad Autonoma Buenos Aires, Buenos Aires, Argentina

Hospital Interzonal General de Agudos General Jose de San Martin /ID# 221893

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La Plata, Buenos Aires, Argentina

CER Instituto Medico /ID# 223175

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Quilmes, Buenos Aires, Argentina

Aprillus Asistencia e Investigacion /ID# 221890

🇦🇷

Ciudad Autonoma de Buenos Aire, Ciudad Autonoma De Buenos Aires, Argentina

Instituto CAICI S.R.L /ID# 221892

🇦🇷

Rosario, Santa Fe, Argentina

UMHAT Sveti Ivan Rilski /ID# 223359

🇧🇬

Sofia, Bulgaria

Guangdong Provincial People's Hospital /ID# 222851

🇨🇳

Guangzhou, Guangdong, China

People's Hospital of Xinjiang /ID# 222928

🇨🇳

Urumqi, Guizhou, China

Huashan Hospital, Fudan University /ID# 222929

🇨🇳

Shanghai, Shanghai, China

Preventive Care Sas /Id# 221881

🇨🇴

Chia, Cundinamarca, Colombia

Clinica Universitaria Bolivari /ID# 221880

🇨🇴

Medellin, Valle Del Cauca, Colombia

Universitaetsklinikum Carl Gustav Carus an der TU Dresden /ID# 222964

🇩🇪

Dresden, Germany

Vital Medicina Kft /ID# 222479

🇭🇺

Veszprém, Veszprem, Hungary

Chukyo Hospital /ID# 223398

🇯🇵

Nagoya-shi, Aichi, Japan

NHO Nagoya Medical Center /ID# 222397

🇯🇵

Nagoya-shi, Aichi, Japan

Hospital of the University of Occupational and Environmental Health, Japan /ID# 222499

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Kitakyushu-shi, Fukuoka, Japan

Hiroshima Red Cross Hospital & Atomic-bomb Survivors Hospital /ID# 222393

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Hiroshima-shi, Hiroshima, Japan

National Hospital Organization Asahikawa Medical Center /ID# 222394

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Asahikawa-shi, Hokkaido, Japan

EIRAKU Internal Medicine Clinic /ID# 222385

🇯🇵

Kagoshima-shi, Kagoshima, Japan

Tohoku University Hospital /ID# 222392

🇯🇵

Sendai-shi, Miyagi, Japan

Shinshu University Hospital /ID# 222395

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Matsumoto-shi, Nagano, Japan

Saitama Medical Center /ID# 222389

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Kawagoe-shi, Saitama, Japan

Keio University Hospital /ID# 222498

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Shinjuku-ku, Tokyo, Japan

Seoul National University Hospital /ID# 221897

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Seoul, Seoul Teugbyeolsi, Korea, Republic of

RM Pharma Specialists S.A de C.V. /ID# 221915

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Mexico City, Ciudad De Mexico, Mexico

CINTRE, Centro de Investigación y Tratamiento Reumatológico SC /ID# 221913

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Mexico City, Ciudad De Mexico, Mexico

Morales Vargas Centro de Investigacion S.C. /ID# 221912

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Leon, Guanajuato, Mexico

Centro Integral en Reumatologia S.A de C.V /ID# 221914

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Guadalajara, Jalisco, Mexico

Centro de Estudios de Investigación Básica y Clínica, S.C. /ID# 221910

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Guadalajara, Jalisco, Mexico

Medical Care & Research SA de CV /ID# 221911

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Mérida, Yucatan, Mexico

North Shore Hospital /ID# 221850

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Takapuna, Auckland, New Zealand

WroMedica I. Bielicka, A. Strzalkowska s.c. /ID# 221860

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Wroclaw, Dolnoslaskie, Poland

Centrum Nowoczesnych Terapii Dobry Lekarz Sp. z o.o. /ID# 224430

🇵🇱

Krakow, Malopolskie, Poland

MTZ Clinical Research Powered by Pratia /ID# 224431

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Warszawa, Mazowieckie, Poland

Ortopedyczno-Rehabilitacyjny Szpital Kliniczny im. Wiktora Degi /ID# 221859

🇵🇱

Poznan, Wielkopolskie, Poland

GCM Medical Group PSC /ID# 224394

🇵🇷

San Juan, Puerto Rico

Mindful Medical Research /ID# 222513

🇵🇷

San Juan, Puerto Rico

HUA - Txagorritxu /ID# 221992

🇪🇸

Vitoria, Alava, Spain

Consorci Corporacio Sanitaria Parc Tauli Sabadell /ID# 221995

🇪🇸

Sabadell, Barcelona, Spain

Hospital Universitario Basurto /ID# 221999

🇪🇸

Bilbao, Vizcaya, Spain

Hospital Universitario de Galdakao /ID# 221996

🇪🇸

Galdakao, Vizcaya, Spain

Hospital Universitario 12 de Octubre /ID# 221994

🇪🇸

Madrid, Spain

Hospital Universitario Virgen de Valme /ID# 221997

🇪🇸

Sevilla, Spain

Hospital Universitario y Politecnico La Fe /ID# 221998

🇪🇸

Valencia, Spain

Taichung Veterans General Hospital /ID# 221748

🇨🇳

Taichung, Keelung, Taiwan

Taipei Veterans General Hosp /ID# 221746

🇨🇳

Taipei, Keelung, Taiwan

National Taiwan University Hospital /ID# 221745

🇨🇳

Taipei City, Taipei, Taiwan

China Medical University Hospital /ID# 221747

🇨🇳

Taichung, Taiwan

Taipei Medical University Hospital /ID# 227653

🇨🇳

Taipei City, Taiwan

Linkou Chang Gung Memorial Hospital /ID# 222469

🇨🇳

Taoyuan City, Taiwan

Guys and St Thomas NHS Foundation Trust /ID# 221863

🇬🇧

London, London, City Of, United Kingdom

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