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Safety and Efficacy of Solithromycin in the Treatment of Nonalcoholic Steatohepatitis Without Cirrhosis

Phase 2
Completed
Conditions
Nonalcoholic Steatohepatitis
Interventions
Registration Number
NCT02510599
Lead Sponsor
Melinta Therapeutics, Inc.
Brief Summary

The purpose of this study is to evaluate the effects of solithromycin on hepatic histology and biomarkers in patients with nonalcoholic steatohepatitis.

Detailed Description

Patients will be administered solithromycin for 13 weeks with regular safety visits and liver biopsies at baseline and after treatment.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
10
Inclusion Criteria
  • Histologic evidence of NASH based on liver biopsy obtained within 180 days
  • NAS> or = 5
  • Able to swallow capsules intact
Exclusion Criteria
  • Symptoms of acute liver disease
  • Cirrhosis on liver biopsy
  • Positive HIV or Hepatitis tests
  • Primary Biliary Cirrhosis
  • Poorly controlled diabetes with HgA1C >8.5%
  • ALT >4-fold upper limit of normal
  • QTcF >450 msec
  • CrCl <40 mL/min

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
SolithromycinsolithromycinSolithromycin 200 mg PO QD for 1 week, followed by 200 mg PO TIW for 12 weeks
Primary Outcome Measures
NameTimeMethod
To evaluate effects on hepatic histology in patients with NASH13 weeks

Using the Nonalcoholic fatty liver disease (NAFLD) Activity Score (NAS)

Secondary Outcome Measures
NameTimeMethod
Changes in inflammation on liver biopsy13 weeks

Graded from 0 to 3

Changes in hepatocellular ballooning score on liver biopsy13 weeks

Graded from 0 to 2

Changes in Steatosis on liver biopsy13 weeks

Graded from 0 to 3

Trial Locations

Locations (1)

Case Western University Hospitals

🇺🇸

Cleveland, Ohio, United States

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