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Trial of Magrolimab (Hu5F9-G4) in Combination With Rituximab or Rituximab + Chemotherapy in Participants With Relapsed/Refractory B-cell Non-Hodgkin's Lymphoma

Phase 1
Terminated
Conditions
Non Hodgkin Lymphoma
Interventions
Registration Number
NCT02953509
Lead Sponsor
Gilead Sciences
Brief Summary

The primary objectives of this study are:

* To investigate the safety and tolerability, and to define the recommended Phase 2 dose and schedule (RP2DS) for magrolimab in combination with rituximab and for magrolimab in combination with rituximab, gemcitabine, and oxaliplatin (R-GemOx).

* To evaluate the efficacy of magrolimab in combination with rituximab in participants with indolent lymphoma and diffuse large B-cell lymphoma (DLBCL) and to evaluate the efficacy of magrolimab in combination with R-GemOx in autologous stem cell transplant (ASCT) ineligible DLBCL participants.

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
178
Inclusion Criteria
  • Phase 1b only: B-cell non-Hodgkin's lymphoma (NHL), relapsed or refractory to standard approved therapies
  • DLBCL Phase 2 cohort: De novo or transformed diffuse large B-cell lymphoma (DLBCL) expressing CD 20, relapsed or refractory to at least 2 prior lines treatment containing anti-CD20 therapy
  • Indolent lymphoma Phase 2 cohort: Marginal zone or follicular lymphoma, relapsed or refractory to standard approved therapies
  • DLBCL chemotherapy combination cohort: De novo or transformed diffuse large B-cell lymphoma (DLBCL), relapsed or refractory to 1-3 prior lines of treatment
  • Adequate performance status and hematological, liver and kidney functions
  • Willing to consent to 1 mandatory pre-treatment and 1 on-treatment tumor biopsy

Key

Exclusion Criteria
  • Active brain metastases
  • Prior allogeneic hematopoietic cell transplantation
  • Prior treatment with CD47 or signal regulatory protein alpha (SIRPα) targeting agents
  • Second malignancy within the last 3 years
  • Known active or chronic hepatitis B or C infection or HIV
  • Pregnancy or active breastfeeding
  • Prior chimeric antigen receptor (CAR-T) therapy

Note: Other protocol defined Inclusion/Exclusion criteria may apply.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Magrolimab + Rituximab, Phase 1b Dose EscalationMagrolimabParticipants with B-cell non-Hodgkin's lymphoma will receive 1 mg/kg magrolimab priming dose on Day 1 of Cycle 1 followed by weekly maintenance doses of 10, 20, 30, or 45 mg/kg on Days 8, 15, 22 for Cycle 1 and Days 1, 8, 15, and 22 for each cycle to determine the maximum tolerated dose (MTD) and recommended Phase 2 dose and schedule (RP2DS) in combination with rituxumab 375 mg/m\^2. Cycle length is 28 days.
Magrolimab + Rituximab, Phase 1b Dose EscalationRituximabParticipants with B-cell non-Hodgkin's lymphoma will receive 1 mg/kg magrolimab priming dose on Day 1 of Cycle 1 followed by weekly maintenance doses of 10, 20, 30, or 45 mg/kg on Days 8, 15, 22 for Cycle 1 and Days 1, 8, 15, and 22 for each cycle to determine the maximum tolerated dose (MTD) and recommended Phase 2 dose and schedule (RP2DS) in combination with rituxumab 375 mg/m\^2. Cycle length is 28 days.
Magrolimab + Rituximab, Phase 2 Indolent LymphomaMagrolimabParticipants with indolent lymphoma will receive magrolimab based on RP2DS from Phase 1b portion of the study in combination with rituxumab 375 mg/m\^2.
Magrolimab + Rituximab, Phase 2 Indolent LymphomaRituximabParticipants with indolent lymphoma will receive magrolimab based on RP2DS from Phase 1b portion of the study in combination with rituxumab 375 mg/m\^2.
Magrolimab + R-GemOx, Phase 1b Dose Expansion PhaseMagrolimabAutologous stem cell transplant (or transplantation) ineligible DLBCL participants will receive magrolimab at a dose determined from Phase 1b Safety Dose-Escalation Phase in combination with rituxumab 375 mg/m\^2 + gemcitabine 1000 mg/m\^2 + oxaliplatin 100 mg/m\^2.
Magrolimab + R-GemOx, Phase 1b Safety Dose Escalation PhaseGemcitabineAutologous stem cell transplant (or transplantation) ineligible DLBCL participants will receive 1 mg/kg magrolimab priming dose on Day 1 for Cyle 1 followed by maintenance doses of 30 or 45 mg/kg on Days 8, 11, 15, 22, and 29 for Cycle 1, every week for Cycle 2, and every 2 weeks for each cycle to determine maximum tolerated dose (MTD) + rituxumab 375 mg/m\^2 + gemcitabine 1000 mg/m\^2 + oxaliplatin 100 mg/m\^2. Cycle length is 28 days.
Magrolimab + Rituximab, Phase 2 Diffuse Large B-Cell lymphomaRituximabParticipants with diffuse large B-cell lymphoma (DLBCL) will receive magrolimab based on RP2DS from Phase 1b portion of the study in combination with rituxumab 375 mg/m\^2.
Magrolimab + R-GemOx, Phase 1b Safety Dose Escalation PhaseRituximabAutologous stem cell transplant (or transplantation) ineligible DLBCL participants will receive 1 mg/kg magrolimab priming dose on Day 1 for Cyle 1 followed by maintenance doses of 30 or 45 mg/kg on Days 8, 11, 15, 22, and 29 for Cycle 1, every week for Cycle 2, and every 2 weeks for each cycle to determine maximum tolerated dose (MTD) + rituxumab 375 mg/m\^2 + gemcitabine 1000 mg/m\^2 + oxaliplatin 100 mg/m\^2. Cycle length is 28 days.
Magrolimab + R-GemOx, Phase 1b Safety Dose Escalation PhaseOxaliplatinAutologous stem cell transplant (or transplantation) ineligible DLBCL participants will receive 1 mg/kg magrolimab priming dose on Day 1 for Cyle 1 followed by maintenance doses of 30 or 45 mg/kg on Days 8, 11, 15, 22, and 29 for Cycle 1, every week for Cycle 2, and every 2 weeks for each cycle to determine maximum tolerated dose (MTD) + rituxumab 375 mg/m\^2 + gemcitabine 1000 mg/m\^2 + oxaliplatin 100 mg/m\^2. Cycle length is 28 days.
Magrolimab + R-GemOx, Phase 1b Dose Expansion PhaseRituximabAutologous stem cell transplant (or transplantation) ineligible DLBCL participants will receive magrolimab at a dose determined from Phase 1b Safety Dose-Escalation Phase in combination with rituxumab 375 mg/m\^2 + gemcitabine 1000 mg/m\^2 + oxaliplatin 100 mg/m\^2.
Magrolimab + R-GemOx, Phase 1b Dose Expansion PhaseGemcitabineAutologous stem cell transplant (or transplantation) ineligible DLBCL participants will receive magrolimab at a dose determined from Phase 1b Safety Dose-Escalation Phase in combination with rituxumab 375 mg/m\^2 + gemcitabine 1000 mg/m\^2 + oxaliplatin 100 mg/m\^2.
Magrolimab + R-GemOx, Phase 1b Dose Expansion PhaseOxaliplatinAutologous stem cell transplant (or transplantation) ineligible DLBCL participants will receive magrolimab at a dose determined from Phase 1b Safety Dose-Escalation Phase in combination with rituxumab 375 mg/m\^2 + gemcitabine 1000 mg/m\^2 + oxaliplatin 100 mg/m\^2.
Magrolimab + Rituximab, Phase 2 Diffuse Large B-Cell lymphomaMagrolimabParticipants with diffuse large B-cell lymphoma (DLBCL) will receive magrolimab based on RP2DS from Phase 1b portion of the study in combination with rituxumab 375 mg/m\^2.
Magrolimab + R-GemOx, Phase 1b Safety Dose Escalation PhaseMagrolimabAutologous stem cell transplant (or transplantation) ineligible DLBCL participants will receive 1 mg/kg magrolimab priming dose on Day 1 for Cyle 1 followed by maintenance doses of 30 or 45 mg/kg on Days 8, 11, 15, 22, and 29 for Cycle 1, every week for Cycle 2, and every 2 weeks for each cycle to determine maximum tolerated dose (MTD) + rituxumab 375 mg/m\^2 + gemcitabine 1000 mg/m\^2 + oxaliplatin 100 mg/m\^2. Cycle length is 28 days.
Primary Outcome Measures
NameTimeMethod
Phase 1b: Percentage of Participants Experiencing Dose-limiting Toxicities (DLTs)Up to 28 days

DLTs refer to toxicities experienced during the first 28 days of study treatment that have been judged to be clinically significant and related to study treatment in participant in Phase 1b.

Percentage of Participants Experiencing Treatment Emergent Adverse EventsFirst dose date up to 5 years
Objective Response Rate as Defined by the Investigator According to the Lugano Classification for LymphomasUp to 5 months

Objective response is defined as complete response (CR) + partial response (PR) determined by Lugano classification for lymphomas.

Secondary Outcome Measures
NameTimeMethod
Progression Free SurvivalUp to 5 years

Progression free survival is measured from dose initiation until the first date of objectively documented disease progression or death.

PK Parameter of Magrolimab: AUCtauBefore magrolimab infusion (within 12 hours) on Day 1, 8, and 15 of Cycle 1, Day 1 and 15 of Cycle 2, Day 1 of Cycles 3, 4, 5, 9, and 13 and until safety follow-up visit (30 days ± 7 days after last dose of magrolimab); Cycle length is 28 days

AUCtau is defined as concentration of drug over time (the area under the concentration verses time curve over the dosing interval).

PK Parameter of Magrolimab: AUClastBefore magrolimab infusion (within 12 hours) on Day 1, 8, and 15 of Cycle 1, Day 1 and 15 of Cycle 2, Day 1 of Cycles 3, 4, 5, 9, and 13 and until safety follow-up visit (30 days ± 7 days after last dose of magrolimab); Cycle length is 28 days

AUClast is defined as the concentration of drug from time zero to the last observable concentration.

PK Parameter of Rituximab: AUClastBefore rituximab infusion (within 12 hours) on Day 8 and 15 of Cycle 1, Day 1 of Cycle 2, Day 1 of Cycles 3 - 6; Cycle length is 28 days

AUClast is defined as the concentration of drug from time zero to the last observable concentration.

PK Parameter of Rituximab: AUCtauBefore rituximab infusion (within 12 hours) on Day 8 and 15 of Cycle 1, Day 1 of Cycle 2, Day 1 of Cycles 3 - 6; Cycle length is 28 days

AUCtau is defined as concentration of drug over time (the area under the concentration verses time curve over the dosing interval).

PK Parameter of Magrolimab: CmaxBefore magrolimab infusion (within 12 hours) on Day 1, 8, and 15 of Cycle 1, Day 1 and 15 of Cycle 2, Day 1 of Cycles 3, 4, 5, 9, and 13 and until safety follow-up visit (30 days ± 7 days after last dose of magrolimab); Cycle length is 28 days

Cmax is defined as the maximum observed concentration of drug.

PK Parameter of Rituximab: CmaxBefore rituximab infusion (within 12 hours) on Day 8 and 15 of Cycle 1, Day 1 of Cycle 2, Day 1 of Cycles 3 - 6; Cycle length is 28 days

Cmax is defined as the maximum observed concentration of drug.

Percentage of Participants who Developed Anti-Magrolimab AntibodiesDay 1 of Cycle 1 to 5, Day 1 Cycle 9, 13, and until safety follow-up visit (30 days ± 7 days after last dose of magrolimab); Cycle length is 28 days
Duration of ResponseUp to 5 years

The duration of response is measured from when the first (objective) response is met (i.e., complete response or partial response) until the first date of objectively documented progressive disease.

Objective Rate of Response Defined by the Investigator According to the LYRIC Criteria for LymphomasUp to 5 months

Objective response is defined as complete response + partial response determined by Lymphoma Response to Immunomodulatory Therapy Criteria (LYRIC) criteria.

Overall SurvivalUp to 5 years

Overall Survival is measured from dose initiation until death.

Time to ProgressionFirst dose date up to 5 years

Time to Progression is measured from dose initiation until the first date of objectively documented progressive disease criteria.

Trial Locations

Locations (20)

Georgia Cancer Center at Augusta University

🇺🇸

Augusta, Georgia, United States

Dana Farber Cancer Institute

🇺🇸

Boston, Massachusetts, United States

University of Minnesota Medical Center, Fairview

🇺🇸

Minneapolis, Minnesota, United States

The University of Texas MD Anderson Cancer Center

🇺🇸

Houston, Texas, United States

The Sarah Cannon Research Institute

🇺🇸

Nashville, Tennessee, United States

University of Michigan

🇺🇸

Ann Arbor, Michigan, United States

Hospital of the University of Pennsylvania

🇺🇸

Philadelphia, Pennsylvania, United States

Linear Clinical Research Ltd

🇦🇺

Nedlands, Western Australia, Australia

The Churchill Hospital

🇬🇧

Oxford, United Kingdom

Princess Alexandra Hospital

🇦🇺

Brisbane, Queensland, Australia

University of Chicago Medical Center

🇺🇸

Chicago, Illinois, United States

Stanford Cancer Center

🇺🇸

Stanford, California, United States

National Institutes of Health Clinical Center/ National Cancer Institute

🇺🇸

Bethesda, Maryland, United States

Beth Israel Deaconess Medical Center

🇺🇸

Boston, Massachusetts, United States

Levine Cancer Institute

🇺🇸

Charlotte, North Carolina, United States

Stephenson Cancer Center

🇺🇸

Oklahoma City, Oklahoma, United States

St. Vincent's Hospital Melbourne

🇦🇺

Melbourne, Victoria, Australia

Washington University School of Medicine Siteman Cancer Center

🇺🇸

Saint Louis, Missouri, United States

University of Alabama At Birmingham (Uab)

🇺🇸

Birmingham, Alabama, United States

City of Hope National Medical Center

🇺🇸

Duarte, California, United States

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