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Pharmacokinetics Of Alprazolam Sublingual Tablet Versus Conventional Tablet

Phase 1
Completed
Conditions
Anxiety Disorder
Interventions
Registration Number
NCT01256151
Lead Sponsor
Pfizer's Upjohn has merged with Mylan to form Viatris Inc.
Brief Summary

To assess if the sublingual tablet will have similar pharmacokinetics as the conventional tablet of alprazolam.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
28
Inclusion Criteria
  • Healthy male and/or female subjects between the ages of 18 and 55 years, inclusive.
  • Body Mass Index (BMI) of 17.5 to 30.5 kg/m2.
  • Signed informed consent.
Exclusion Criteria
  • Evidence or history of clinically significant abnormalities
  • Positive drug screen, excessive alcohol and tobacco use

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Alprazolam sublingual tabletAlprazolam sublingualAlprazolam sublingual tablet
Alprazolam conventional tabletAlprazolam tabletAlprazolam conventional tablet
Primary Outcome Measures
NameTimeMethod
Peak concentration of alprazolam72 hours
Area under the curve (AUC) from time zero to last measurable time of alprazolam72 hours
Secondary Outcome Measures
NameTimeMethod
AUC% extrapolated72 hours
Time of Cmax72 hours
Area under the curve from time zero to infinity72 hours
half-life of alprazolam72 hours
Clinically significant safety laboratory testsScreening, Day 0, Day 4
Clincally significant vital signsScreening, Day 4
Clinically significant adverse events1 month

Trial Locations

Locations (1)

Pfizer Investigational Site

🇺🇸

New Haven, Connecticut, United States

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