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Drug metabolism related to obesity

Phase 1
Conditions
MedDRA version: 19.1Level: LLTClassification code 10029885Term: Obesity, unspecifiedSystem Organ Class: 100000004861
Therapeutic area: Body processes [G] - Metabolic Phenomena [G03]
Registration Number
EUCTR2014-004554-34-DK
Lead Sponsor
Bispebjerg Hospital
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
ot Recruiting
Sex
All
Target Recruitment
Not specified
Inclusion Criteria

•Obese children (BMI = 99 % percentile)
•Healthy non-obese children (BMI= 90 % percentile)
•Age 11-18 years
•Both genders (block stratified)
•Postmenarche (females)
•Written informed consent from both parents (age<18)
Females included will be post menarche (Tanner stage 4) in order to avoid bias, as maturation of CYP1A2 activity mirrors pubertal growth, which peaks early in females.

Are the trial subjects under 18? yes
Number of subjects for this age range: 68
F.1.2 Adults (18-64 years) no
F.1.2.1 Number of subjects for this age range 0
F.1.3 Elderly (>=65 years) no
F.1.3.1 Number of subjects for this age range 0

Exclusion Criteria

•Acute or chronic Liver diseases
•Other chronic diseases, except from allergic rhinitis, rash etc.
•Intake of drugs known to induce of inhibit CYP2E1-, CYP3A4 and/or CYP1A2, including paracetamol, ciprofloxacin, azithromycin, ketoconazol, estradiol etc.
•Citrus fruit
•Alcohol intake within minimum 72 hours
•Caffeine (Coca Cola©, coffee and tea) intake 48 h prior to administration of the caffeine-probe
•Smoking 96 hours prior to administration of the caffeine-probe, screening test will be performed (nicotine metabolite: cotinine)
•Kidney disease and dialysis
•Pregnancy (test will be performed)
•Known hypersensitivity to chlorzoxazone, midazolam or caffeine
•vigorous exercise 24 hours before administration

Study & Design

Study Type
Interventional clinical trial of medicinal product
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
Secondary Outcome Measures
NameTimeMethod
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