MedPath

Oral Docetaxel for Prostate Cancer

Phase 1
Completed
Conditions
Metastatic prostate cancer
Cancer - Prostate
Registration Number
ACTRN12616000983404
Lead Sponsor
Kinex Pharmaceuticals Inc
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
Completed
Sex
Male
Target Recruitment
11
Inclusion Criteria

Eligible participants must be males at least 18 years of age with metastatic prostate cancer who are scheduled to receive their prescribed dose of treatment with IV docetaxel. Patients may be receiving steroid treatment or ADT for prostate cancer, but other concomitant cancer chemotherapy is not permitted.
They must have:
- adequate hematologic status as demonstrated by not requiring transfusion support or granulocyte-colony stimulating factor (G-CSF);
- Adequate liver function as demonstrated by: Total bilirubin of less than the upper limit of normal (ULN); Aspartate transaminase (AST) and alanine aminotransferase (ALT) less than/equal to 1.5 times ULN; Alkaline phosphatase (ALP) less than/equal to 2.5 times ULN or less than 5 times ULN if bone metastases are present
- Adequate renal function as demonstrated by serum creatinine less than/equal to 177 micromole/L or creatinine clearance greater than 60 mL/min as calculated by the Cockcroft and Gault formula
Participants must have an Eastern Cooperative Oncology Group (ECOG) performance status of 0 to 1; Life expectancy of at least 6 months; Willing to fast for 8 hours before and 4 hours after Oradoxel administration; Willing to abstain from alcohol consumption from 3 days prior Study Period 1 through to the Final Visit; Willing to refrain from caffeine consumption for 12 hours prior to each dose of study drug through the completion of protocol-specified PK sampling time-points; Sexually active participants must use a barrier method of contraception during the study and agree to continue the use of contraception for at least 30 days after the last dose of study drug.

Exclusion Criteria

Eligible participants must not be
- currently taking a prohibited concomitant medication;
- have unresolved toxicity from prior chemotherapy (participants must have recovered from all significant toxicity to less than or equal to Grade 1 CTCAE toxicity from previous anticancer treatments or previous investigational agents);
- planning to receive other medical, surgical, or radiological treatments for prostate cancer during the course of this study;
- received investigational agents within 14 days or 5 half-lives prior to the first study dosing day, whichever is longer;
- uncontrolled intercurrent illness; no major surgery to the upper gastrointestinal (GI) tract, or have a history of GI disease or other medical condition that, in the opinion of the Investigator may interfere with oral drug absorption;
- known history of allergy to docetaxel, Cremophor (Registered Trademark), or polysorbate 80 (Tween 80);
- any other condition which the Investigator believes would make participation in the study not acceptable.

Study & Design

Study Type
Interventional
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
Secondary Outcome Measures
NameTimeMethod
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