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Radiation Dosimetry, Metabolism, Pharmacokinetics, Safety and Tolerability and PET Imaging With BAY94-9392 in Healthy Volunteers and Patients With Cancer or Inflammation

Phase 1
Completed
Conditions
Diagnostic Imaging
Neoplasms
Interventions
Registration Number
NCT01103310
Lead Sponsor
Life Molecular Imaging SA
Brief Summary

Visual assessment of diagnostic PET/CT (positron emission tomography/computed tomography) images obtained after a single intravenous injection of BAY94-9392 in patients with cancer or inflammation.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
46
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Arm 1BAY94-9392Cancer patients, single intravenous bolus injection of 300 MBq BAY94-9392 on day one of the treatment period, PET/CT
Arm 2BAY94-9392Healthy volunteers, single intravenous bolus injection of 300 MBq BAY94-9392 on day one of the treatment period, whole body PET/CT for determination of effective dose, kinetics of BAY94-9392 in blood
Primary Outcome Measures
NameTimeMethod
Visual assessment of lesionDay of study drug administration
Secondary Outcome Measures
NameTimeMethod
Serum creatinineAt least twice within 2 days after treatment
Serum proteinAt least twice within 2 days after treatment
Quantitative analysis of BAY94-9392 uptake into lesions (Standardized Uptake Values = SUVs)Day of study drug administration
Electrocardiogram (ECG)At least twice within 2 days after treatment
Blood pressureAt least twice within 2 days after treatment
Serum GOT (Glutamate-Oxalacetate-Transaminase)At least twice within 2 days after treatment
Adverse events collectionContinuously for at least 4 days after treatment
Radiation doses per organ (µGy/MBq)Day of study drug administration
Doses per organ (µSv/MBq)Day of study drug administration
Higher organ dose (HT)Day of study drug administration
Effective dose (µSv/MBq)Day of study drug administration
Effective dose resulting from the total administered diagnostic activity of 300 MBq +/- 10%Day of study drug administration
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