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A Study to Assess the Safety, Pharmacokinetics, and Antiviral Activity of ABI-H3733 in Subjects With Chronic Hepatitis B Virus Infection

Phase 1
Completed
Conditions
Chronic Hepatitis B
Interventions
Drug: Placebo
Registration Number
NCT05414981
Lead Sponsor
Assembly Biosciences
Brief Summary

This is a randomized, blinded, placebo-controlled, dose-ranging Phase 1b study of the safety, PK, and antiviral activity of ABI-H3733 in treatment-naïve or off-treatment chronic Hepatitis B virus (cHBV) subjects that are Hepatitis B e antigen (HBeAg) positive or negative. The study will enroll up to 5 sequential cohorts of 10 subjects each, for a total of up to 50 subjects, randomized 8:2 to receive ABI-H3733 or placebo.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
31
Inclusion Criteria
  1. Body mass index (BMI) ≥ 18.0 and < 35.0 kg/m(2), where BMI = weight (kg)/(height [m])(2) with a minimum body weight of 45 kg.
  2. Chronic hepatitis B infection, defined as HBV infection for ≥6 months documented
  3. Treatment-naïve or off-antiviral therapy for ≥24 weeks prior to Screening
  4. Lack of bridging fibrosis or cirrhosis
Exclusion Criteria
  1. Co-infection with human immunodeficiency virus (HIV), hepatitis C virus (HCV), hepatitis D virus (HDV), acute hepatitis A virus (HAV), or acute hepatitis E virus (HEV)
  2. History of liver transplant or evidence of advanced liver disease, cirrhosis, or hepatic decompensation
  3. Clinically significant diseases or conditions
  4. History of hepatocellular carcinoma
  5. Current or prior treatment for cHBV

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
ABI-H3733ABI-H3733-
PlaceboPlacebo-
Primary Outcome Measures
NameTimeMethod
Proportion of subjects with adverse events (AEs), premature treatment discontinuation due to AEs, and abnormal laboratory resultsThrough end of study, up to 56 days
Secondary Outcome Measures
NameTimeMethod
Maximum Plasma Concentration (Cmax) of ABI-H3733 in subjects with cHBVThrough treatment period, up to 28 days
Minimum Plasma Concentration (Cmin) of ABI-H3733 in subjects with cHBVThrough treatment period, up to 28 days
Area Under Plasma Concentration-Time Curve (AUC) of ABI-H3733 in subjects with cHBVThrough treatment period, up to 28 days
Time to Maximum Plasma Concentration (Tmax) of ABI-H3733 in subjects with cHBVThrough treatment period, up to 28 days
Elimination half-life (t1/2) of ABI-H3733 in subjects with cHBVThrough treatment period, up to 28 days
To evaluate the effect of food on Cmax of ABI-H3733 in subjects with cHBVThrough treatment period, up to 28 days
To evaluate the effect of food on AUC of ABI-H3733 in subjects with cHBVThrough treatment period, up to 28 days
To evaluate the effect of food on the proportion of subjects with AEs, premature discontinuation due to AEs and abnormal laboratory resultsThrough treatment period, up to 28 days
To evaluate the changes in HBV DNA (IU/mL or Log IU/mL) in subjects with cHBV by Quantitative PCRThrough treatment period, up to 28 days

Trial Locations

Locations (9)

Diagnostic Consultative Center Aleksandrovska

🇧🇬

Sofia, Sofia City, Bulgaria

National University Hospital

🇸🇬

Singapore, Singapore

Clinical Trials and Research Centre, Singapore General Hospital

🇸🇬

Singapore, Singapore

New Zealand Clinical Research

🇳🇿

Grafton, Auckland, New Zealand

Military Medical Academy Multiprofile Hospital for Active Treatment - Sofia

🇧🇬

Sofia, Bulgaria

Acibadem City Clinic Tokuda Hospital

🇧🇬

Sofia, Bulgaria

Institute of Infectious Diseases - Hospital ARENSIA Exploratory Medicine Research Clinic National Institute of Infectious Diseases "Matei Bals"

🇷🇴

Bucharest, Romania

ICS Arensia Exploratory Medicine Republican Clinical Hospital "Timofei Moșneaga"- Hospital

🇲🇩

Chisinau, Moldova, Republic of

University of Hong Kong

🇭🇰

Hong Kong, Hong Kong

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