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A Trial of PEGPH20 in Combination With Avelumab in Chemotherapy Resistant Pancreatic Cancer

Early Phase 1
Terminated
Conditions
Pancreatic Cancer
Pancreatic Ductal Adenocarcinoma
Interventions
Registration Number
NCT03481920
Lead Sponsor
PH Research, S.L.
Brief Summary

The purpose of this study is to evaluate the pharmacodynamics, safety and efficacy of PEGPH20 in combination with Avelumab in adult patients with chemotherapy resistant advanced or locally advanced pancreatic ductal adenocarcinoma (PDAC). This is a multi-center, open-label, non-randomized trial.

Detailed Description

The reported response rate with check-point inhibitors in PDAC is 0 %. This study tests the hypothesis that elimination of HA in pancreas tumor microenvironment mediated by PEG PH20 will result in increased tumor vascularization and vessel patency as well as stromal remodeling with increase immune infiltrate. These effects may facilitate the activity of check-point inhibitors like avelumab by at least two mechanisms including increase in drug delivery and increasing immune infiltrate.

The purpose of this study is to evaluate the pharmacodynamics, safety and efficacy of PEGPH20 in combination with Avelumab in adult patients with chemotherapy resistant advanced or locally advanced pancreatic ductal adenocarcinoma (PDAC). This is a multi-center, open-label, non-randomized trial.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
7
Inclusion Criteria
  • Signed, written IRB/IEC-approved Informed Consent Form

  • Histologically or cytologically-confirmed pancreatic ductal adenocarcinoma (PDAC).

  • Accessible tumor for two repeated tumor biopsies.

  • Progression to first line treatment for locally advanced or advanced disease. Prior adjuvant chemotherapy or chemoradiation therapy for early disease is allowed.

  • Age ≥18 years.

  • Radiologically measurable disease per RECIST v1.1.

  • Performance-status ECOG 0 -2.

  • Life expectancy ≥ 3 months.

  • Resolved acute effects of any prior therapy to baseline or Grade ≤1 severity

  • Screening laboratory:

    1. Hematologic: ANC ≥ 1.5 × 109/L, platelet count ≥ 100 × 109/L, and hemoglobin ≥ 9 g/dL
    2. Hepatic: Total bilirubin level ≤ 1.5 × the ULN range and AST and ALT levels ≤ 2.5 × ULN or AST and ALT levels ≤ 5 X ULN (for subjects with documented metastatic disease to the liver)
    3. Renal: Estimated creatinine clearance ≥ 30 mL/min according to the Cockcroft-Gault formula or serum creatinine ≤ 2.0 mg/dL.
    4. Albumin ≥2.5 g/dL.
    5. Coagulation: PT time and INR within normal limits (+/-15%). PTT within normal limits (+/-15%).
  • If a subject requires anticoagulation, treatment must be modified to enoxaparin.

  • Negative serum pregnancy test if female subject is of childbearing potential.

  • Patients who are willing and able to comply with scheduled visits, treatment plans, laboratory tests, biopsies when required, and other procedures.

Exclusion Criteria
  • Clinical evidence of DVT, PE, prior history of CVA or history of TIA within 12 months or other known TE event present during the screening period
  • Current use of megestrol acetate (use within 10 days of Day 1).
  • Contraindication to heparin as per institutional guidelines.
  • Another primary cancer within the last 3 years currently requiring antineoplastic treatment within the exception of non-melanoma skin cancer, early-stage prostate cancer, or curatively treated cervical carcinoma in-situ.
  • Current use of immunosuppressive medication within 2 weeks of study participation, EXCEPT for those listed in protocol
  • Active autoimmune disease that might deteriorate when receiving an immuno-stimulatory agent: Patients with diabetes type I, vitiligo, psoriasis, or hypo- or hyperthyroid diseases not requiring immunosuppressive treatment are eligible.
  • Prior organ transplantation including allogenic stem-cell transplantation.
  • Active infection requiring systemic therapy.
  • Known infection with human immunodeficiency virus, Hepatitis B, or Hepatitis C
  • Known prior severe hypersensitivity to investigational product, hyaluronidase, or any component in its formulations, including known severe hypersensitivity reactions to monoclonal antibodies (NCI CTCAE v4.03 Grade ≥ 3).
  • Any history of anaphylaxis or uncontrolled asthma (that is, 3 or more features of partially controlled asthma).
  • Clinically significant (i.e., active) cardiovascular disease: myocardial infarction (< 6 months prior to enrollment), unstable angina, congestive heart failure (≥ New York Heart Association Classification Class II), or serious cardiac arrhythmia requiring medication.
  • Prior cerebrovascular accident/stroke.
  • Clinically significant carotid artery disease (e.g. prior carotid surgery, symptomatic and/or requires treatment)
  • Inability to comply with study and follow-up procedures as judged by the Investigator.
  • Known alcohol or drug abuse.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
PEGPH20 + AvelumabPEGylated Recombinant Human Hyaluronidase (PEGPH20)PEGPH20, a multi-site PEGylated enzyme generated by conjugating N-hydroxysuccinimidyl ester of methoxypoly(ethylene glycol)-butanoic acid (MSBA30K/B or PEG) and recombinant human hyaluronidase (rHuPH20). PEGPH20 has a half-life of approximately 2 days, thereby enabling systemic activity and sustained duration of action to degrade HA. In many different tumor types tested in murine xenograft models, response to PEGPH20 has been shown to be more robust for tumors characterized by higher HA expression.
PEGPH20 + AvelumabAvelumabPEGPH20, a multi-site PEGylated enzyme generated by conjugating N-hydroxysuccinimidyl ester of methoxypoly(ethylene glycol)-butanoic acid (MSBA30K/B or PEG) and recombinant human hyaluronidase (rHuPH20). PEGPH20 has a half-life of approximately 2 days, thereby enabling systemic activity and sustained duration of action to degrade HA. In many different tumor types tested in murine xenograft models, response to PEGPH20 has been shown to be more robust for tumors characterized by higher HA expression.
Primary Outcome Measures
NameTimeMethod
Determine ORR as per RECIST v1.1 criteria6 months from trial treatment initiation cycle 1/day 1. Each treatment cycle is 14 days

Determine ORR as per RECIST v1.1 criteria

To assess the safety of this combination in patients with PDAC.Initiation of trial treatment cycle 1/day 1 through 30 days after last dose of trial treatment

graded by National Cancer Institute Common Terminology Criteria for Adverse Events (NCI CTCAE) version 4.03

Secondary Outcome Measures
NameTimeMethod
Changes in CA 19,9 levesUp to 4 weeks

Measured in UI/ML

Determine OS (OVERALL SURVIVAL)From date of treatment initiation cycle 1/day 1 until death from any cause, assessed up to 36 months

The length of time from either the date of diagnosis or the start of treatment for a disease, such as cancer, that patients diagnosed with the disease are still alive

Determine PFS (PROGRESSION FREE SURVIVAL)From date of treatment initiation cycle 1/day 1 until progression, assessed up to 24 months

The length of time during and after the treatment of a disease, such as cancer, that a patient lives with the disease but it does not get worse.

Trial Locations

Locations (3)

Hospital Universitario La Paz

🇪🇸

Madrid, Spain

Hospital Universitario Fuenlabrada

🇪🇸

Fuenlabrada, Madrid, Spain

Hospital Ramon y Cajal

🇪🇸

Madrid, Spain

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