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Open Label Safety & Pharmacodynamic Study 24Wk w/DIO-902 Combo w/Metformin & Atorvastatin in T2DM Patients

Phase 2
Terminated
Conditions
Type 2 Diabetes
Interventions
Registration Number
NCT00622089
Lead Sponsor
DiObex
Brief Summary

DiObex Inc. is developing an experimental drug (DIO-902) that is made up of part of the ketoconazole molecule for the treatment of elevated blood glucose associated with type 2 diabetes mellitus. Ketoconazole (Nizoral®) is a drug available by prescription for the treatment of fungal infections however DIO-902 is an investigational drug. DIO-902 may lower blood glucose by lowering levels of a naturally occurring hormone called cortisol. Elevated cortisol may contribute to the development of type 2 diabetes.

Detailed Description

To maintain the blind in Protocol DIO-502, subjects will be re-randomized at Study Visit 1 to one of three doses of DIO-902: 150, 300 or 450 mg QHS. All subjects receiving DIO-902 placebo and 50% of subjects receiving DIO-902 will be re-randomized to one of three DIO-902 doses. The remaining 50% of subjects receiving DIO-902 will be assigned to their original DIO-902 dose. The re- randomization will be performed by a group independent of study conduct to ensure the treatment status of the subject while in Protocol DIO-502 remains blinded. In addition, subjects will continue on the same dose of metformin that they had been taking during the conduct of Protocol DIO-502. Subjects will continue on atorvastatin 10 mg for the first 4 weeks of this protocol. Thereafter, at Study Visits 3 and 4, the dose of atorvastatin may be increased up to a maximum of 40 mg daily in order to achieve LDL-cholesterol/non-HDL cholesterol goals specified within the protocol. In addition, after Study Visit 4 (Week 12) subjects with HbA1c levels of \> 7.5% (0.075 Hb Fract.) will undergo a one time titration of their oral hypoglycemic regimen as per the algorithm provided in the protocol.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
150
Inclusion Criteria
  • Participated in DIO-502
Exclusion Criteria
  • Did not participate in DIO-502

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
1DIO-902150mg DIO-902 + 10mg Atorvastatin
2.DIO-902300mg DIO-902 + 10mg Atorvastatin
3DIO-902450mg DIO-902 + 10mg Atorvastatin
Primary Outcome Measures
NameTimeMethod
The following parameters will be evaluated at Week 12 and Week 24: • Proportion of subjects who reach the lipid goal as defined in the protocol from baseline • Proportion of subjects who meet the HbA1c goal as defined in the protocol from baseline24 weeks
Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (24)

Dr. Terence Hart

🇺🇸

Muscle Shoals, Alabama, United States

Genova Research

🇺🇸

Tucson, Arizona, United States

Research Solutions

🇺🇸

Jonesboro, Arkansas, United States

Arkansas Primary Care Clinic

🇺🇸

Little Rock, Arkansas, United States

Advanced Medical Research

🇺🇸

Lakewood, California, United States

Mills-Peninsula Helath Services

🇺🇸

San Mateo, California, United States

Diabetes Research Goup University of Hawaii at Manoa

🇺🇸

Honolulu, Hawaii, United States

Creighton Diabetes Center

🇺🇸

Omaha, Nebraska, United States

AHS Oklahoma Physician Group

🇺🇸

Tulsa, Oklahoma, United States

Covance Clinical Research Unit - Dr. Andrew Ahmann

🇺🇸

Portland, Oregon, United States

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Dr. Terence Hart
🇺🇸Muscle Shoals, Alabama, United States

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