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Study of the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of REGN3918 in Healthy Volunteers

Phase 1
Completed
Conditions
Healthy Volunteers
Interventions
Drug: Placebo
Registration Number
NCT03115996
Lead Sponsor
Regeneron Pharmaceuticals
Brief Summary

To evaluate the safety and tolerability of single ascending intravenous (IV) and subcutaneous (SC) doses and a multiple dose regimen.

Detailed Description

Participants will be randomized to single IV or SC or multiple dose treatment with REGN3918 or matched placebo.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
56
Inclusion Criteria

A subject must meet the follow criteria to be eligible for inclusion in the study:

  1. Males and females from 18 to 50 years of age.
  2. Subject is judged to be in good health based on medical history, physical examination, vital sign measurements and laboratory safety tests performed at screening and/or prior to administration of initial dose of study drug
  3. The subject has a body mass index less than 30 kg/m2
  4. Willingness to undergo vaccination and antibiotic prophylaxis against N. meningitides.

Key

Exclusion Criteria

A subject who meets any of the following criteria will be excluded from the study:

  1. Any clinically significant physical examination abnormalities observed during the screening visit.
  2. Hospitalization for any reason within 30 days of the screening visit
  3. Persistent chronic or active recurring infection requiring treatment with antibiotics, antivirals, or antifungals.
  4. Subject has a history of meningococcal infection.
  5. Carriers of Neisseria meningitides based on cultures from naso-pharyngeal swabs during screening.
  6. Subject has had a splenectomy.
  7. Known allergy to penicillin class antibiotics
  8. Known or suspected complement deficiency, or abnormal complement C3, C4 or CH50 during screening.
  9. Recent (within the previous 2 months) bacterial, protozoal, viral or parasite infection requiring systemic treatment.
  10. History of tuberculosis or systemic fungal diseases
  11. HIV infection or HIV seropositivity at the screening visit
  12. Positive HBsAg, HBcAb, or hepatitis C antibody at the screening visit
  13. History of malignancy (except non-melanoma skin cancer or cervical in-situ)
  14. Pregnant or breastfeeding women
  15. Women of childbearing potential and men who are unwilling to practice highly effective contraception prior to the initial dose/start of the first treatment, during the study, and for at least 6 months after the last dose

Note: Other protocol defined Inclusion/Exclusion criteria may apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Placebo (Cohorts 1-4 & 6a)PlaceboCohorts 1-4 and 6a will receive placebo
REGN3918 (Cohorts 1-4 & 6a)REGN3918Cohorts 1-4 and 6a will receive sequential ascending doses of REGN3918
REGN3918 (Cohort 5 & 6b)REGN3918Cohort 5 and 6b will receive multiple doses of REGN3918
Placebo (Cohort 5 & 6b)PlaceboCohort 5 and 6b will receive placebo
Primary Outcome Measures
NameTimeMethod
Incidence of treatment emergent adverse events (TEAEs)Up to 20 weeks
Severity of TEAEsUp to 20 weeks
Secondary Outcome Measures
NameTimeMethod
Pharmacodynamics profile of REGN3918Up to 20 weeks

Assessed by CH50 assay over time

Pharmacokinetic profile of REGN3918; single dose IV and SCUp to 20 weeks

Assessed via serum concentrations of REGN3918 over time; Area under the Curve (AUC)

Pharmacokinetic profile of REGN3918; single dose IV and repeated SC dosesUp to 20 weeks

Assessed via serum concentrations of REGN3918 over time; peak concentration Cmax

Pharmacokinetic exploratory analysisUp to 20 weeks

Peak concentration Cmax

Immunogenicity of REGN3918Up to 20 weeks

Assessed by measurement of anti-drug antibodies (ADA)

Trial Locations

Locations (1)

Covance Clinical Research Unit (CRU) Ltd.

🇬🇧

Leeds, United Kingdom

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