MedPath

A Study of Nemonoxacin Malate Sodium Chloride Injection Administered by Intravenous Infusion

Phase 1
Completed
Conditions
Healthy
Interventions
Registration Number
NCT01529957
Lead Sponsor
TaiGen Biotechnology Co., Ltd.
Brief Summary

The purpose of this study is to evaluate the safety and tolerability of nemonoxacin in healthy Chinese volunteers.

Detailed Description

Single dose safety and tolerability study: evaluate safety and tolerability of intravenous infusion nemonoxacin 25mg, 50mg, 125mg, 250mg, 500mg, 750mg, 1000mg and 1250mg.

Single dose pharmacokinetic (PK) study:evaluate PK profile of doses of 250mg, 500mg or 750mg intravenous infusion nemonoxacin .

Multiple dose study: evaluate PK profile of doses of 500mg, 650mg or 750mg intravenous infusion nemonoxacin after consecutive 10 days.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
176
Inclusion Criteria
  1. Healthy male or female, aged 18 ~45
  2. A male volunteer should be willing to use a double-barrier contraception until the study is completed, and should not make his partner pregnant during the study and within 3 months after completing the study
  3. Volunteers who have never used any tobacco or nicotine-containing product within three months before use of the investigational product
  4. Volunteers who are willing to abstain from caffeine- or xanthine- containing drinks or food within 24h before being enrolled in the study and throughout the study,such as coffee and tea,chocolate,alcohol, grapefruit juice,orange juice,etc.
  5. The body mass index (BMI) of the volunteer must be 19~24, and the weight of a male should be at least 50kg,and that of a female should be at least 45kg.
  6. Volunteers who are able to sign the informed consent form (ICF) of their own accord.
Exclusion Criteria
  1. History of diabetes,or cardiovascular,hepatic or renal disease.
  2. Had surgery or trauma within 6 months prior to this study
  3. Alcohol or drug abuse
  4. HIV, HBV or HCV positive
  5. subject used any known hepatic enzyme inducer/hepatic enzyme inhibitor product within 30 days prior to the study
  6. Used any prescribed drug (including traditional chinese medicine) within 14 days prior to the study
  7. Donated 400ml of blood or plasma within 3 months prior to this study
  8. Have an abnormal laboratory examination value that exceeds the normal range by 10%
  9. Drug allergies
  10. Have cardiac disorders or have a family history of cardiac disorders
  11. Have abnormal 12-lead ECG during screening
  12. Pregnant or lactating
  13. Participated in any study within 3 months prior to this study
  14. according to the investigator's judgment, affect the safety or efficacy evaluation.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Nemonoxacin Malate Sodium Chloride 50 mgNemonoxacin Malate Sodium ChlorideNemonoxacin Malate Sodium Chloride 50 mg
Nemonoxacin Malate Sodium Chloride 125 mgNemonoxacin Malate Sodium ChlorideNemonoxacin Malate Sodium Chloride 125 mg
Nemonoxacin Malate Sodium Chloride 750 mgNemonoxacin Malate Sodium ChlorideNemonoxacin Malate Sodium Chloride 750 mg
Nemonoxacin Malate Sodium Chloride 25 mgNemonoxacin Malate Sodium ChlorideNemonoxacin Malate Sodium Chloride 25 mg
placebolNemonoxacin Malate Sodium Chlorideplacebol
Nemonoxacin Malate Sodium Chloride 250 mgNemonoxacin Malate Sodium ChlorideNemonoxacin Malate Sodium Chloride 250 mg
Nemonoxacin Malate Sodium Chloride 500 mgNemonoxacin Malate Sodium ChlorideNemonoxacin Malate Sodium Chloride 500 mg
Nemonoxacin Malate Sodium Chloride 650 mgNemonoxacin Malate Sodium ChlorideNemonoxacin Malate Sodium Chloride 650 mg
Nemonoxacin Malate Sodium Chloride 1000 mgNemonoxacin Malate Sodium ChlorideNemonoxacin Malate Sodium Chloride 1000 mg
Nemonoxacin Malate Sodium Chloride 1250 mgNemonoxacin Malate Sodium ChlorideNemonoxacin Malate Sodium Chloride 1250 mg
Primary Outcome Measures
NameTimeMethod
Adverse event assessment in healthy Chinese volunteer46days
Maximum tolerated single dose of nemonoxacin in healthy Chinese volunteers32days
Secondary Outcome Measures
NameTimeMethod
Pharmacokinetic profile of nemonoxacin in healthy Chinese volunteers4days

Trial Locations

Locations (26)

Guangzhou Red Cross Hospital

πŸ‡¨πŸ‡³

Guangzhou, China

Third Military Medical University, Third Affiliated Hospital

πŸ‡¨πŸ‡³

Chongqing, China

Zhen Hospital, Capital Medical University Beijing

πŸ‡¨πŸ‡³

Beijing, China

Second Affiliated Hospital of Nanchang University

πŸ‡¨πŸ‡³

Jiangxi, China

Shanghai Changzheng Hospital

πŸ‡¨πŸ‡³

Shanghai, China

Shanghai Pudong New Area, Oriental Hospital

πŸ‡¨πŸ‡³

Shanghai, China

Kunming General Hospital of Chengdu Military Region

πŸ‡¨πŸ‡³

Chengdu, China

West China Hospital of Sichuan University

πŸ‡¨πŸ‡³

Chengdu, China

Second Affiliated Hospital, Third Military Medical University

πŸ‡¨πŸ‡³

Chongqing, China

Third Military Medical University First Affiliated Hospital

πŸ‡¨πŸ‡³

Chongqing, China

Second Affiliated Hospital of Dalian Medical University

πŸ‡¨πŸ‡³

Dalian, China

Gansu Provincial People's Hospital

πŸ‡¨πŸ‡³

Gansu, China

Second Affiliated Hospital of Sun Yat-sen

πŸ‡¨πŸ‡³

Guangzhou, China

Hangzhou First People's Hospital

πŸ‡¨πŸ‡³

Hangzhou, China

Xiangya Hospital, Central South University

πŸ‡¨πŸ‡³

Hunan, China

Jiangxi Provincial People's Hospital

πŸ‡¨πŸ‡³

Jiangxi, China

Shengjing Hospital of China Medical University

πŸ‡¨πŸ‡³

Liaoning, China

Peking University First Hospital

πŸ‡¨πŸ‡³

Peking, China

Peking University People's Hospital

πŸ‡¨πŸ‡³

Peking, China

Affiliated Hospital of Qingdao University Medical College

πŸ‡¨πŸ‡³

Qingdao, China

Second Affiliated Hospital of Xi'an Jiaotong University

πŸ‡¨πŸ‡³

Xi'an, China

Third Xiangya Hospital, Central South University

πŸ‡¨πŸ‡³

Hunan, China

Institute of Antibiotics, Huashan Hospital, Fundan University

πŸ‡¨πŸ‡³

Shanghai, China

First Affiliated Hospital,Zhejiang University School of Medicine

πŸ‡¨πŸ‡³

Zhejiang, China

People's Liberation Army General Hospital of Shenyang Military Region

πŸ‡¨πŸ‡³

Shenyang, China

Huai'an First Hospital of Nanjing Medical University

πŸ‡¨πŸ‡³

Nanjing, China

Β© Copyright 2025. All Rights Reserved by MedPath