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Safety and Efficacy of Terbogrel in Patients With Primary Pulmonary Hypertension

Phase 2
Completed
Conditions
Hypertension, Pulmonary
Interventions
Registration Number
NCT02223481
Lead Sponsor
Boehringer Ingelheim
Brief Summary

This study sought to determine whether terbogrel was an effective treatment for primary pulmonary hypertension (PPH) by comparing its efficacy and safety to that of placebo.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
71
Inclusion Criteria
  • Primary pulmonary hypertension and New York Health Association (NYHA) chronic heart failure (CHF) functional class II-III
  • Ability to walk >= 50 meters on the 6 minute walk test
  • Resting mean pulmonary artery pressure > 25 mmHg
  • Mean right atrial pressure <= 20 mmHg
  • Pulmonary capillary wedge pressure <= 15 mmHg
  • Cardiac index > 2.5 L/min2
  • SvO2 sat. > 63%
  • Male of female at least 18 years old
  • Signed written informed consent
Exclusion Criteria
  • Secondary pulmonary hypertension due to lung or systemic diseases
  • Pregnant of nursing women, or women of childbearing potential who are not using adequate methods of birth control
  • Concurrent systematic use of aspirin, aspirin like drugs, or non-steroidal anti-inflammatory drugs (NSAIDs)
  • Surgery of bleeding from gastrointestinal, genitourinary tract, cerebrum or retina within past 6 weeks
  • History of bleeding diathesis or a platelet count less than 70,000/mm3
  • Exercise limited by factors other than fatigue or exertional dyspnea, such as arthritis, claudication, angina, chronic obstructive pulmonary disease, or bronchial asthma
  • Myocardial infarction, stroke, or transient ischemic attack within the preceding six months
  • Systolic blood pressure < 90 mmHg or > 180 mmHg, or diastolic blood pressure > 110 mmHg
  • Known drug or alcohol dependency within one year of entry into the study
  • Known hypersensitivity to any component of the study formulation, epoprostenol, nitric oxide, or adenosine
  • Psychiatric or other illness or condition which, in the opinion of the principal investigator, may interfere with study participation, compliance, or other elements of the protocol
  • Participation in an evaluation of an investigational drug within the past 30 days
  • Portal hypertension or cirrhosis of the liver
  • Congenital heart disease e.g., atrial septal defect; patent foramen ovale does not exclude patient from the study
  • Appetite suppressants such as fenfluramine, dexfenfluramine, and inhibitors of serotonin uptake known to be associated with primary pulmonary hypertension, received within 3 months of entry into the study
  • HIV positive
  • Vasodilators. Patients will not receive Ca-channel blockers during the study unless the medication was started prior to the study and the patient has been on a stable dose for at least one month prior to entry

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Terbogrel low doseTerbogrel low dose-
Terbogrel high doseTerbogrel high dose-
PlaceboPlacebo-
Primary Outcome Measures
NameTimeMethod
Change in pulmonary vascular resistance (PVR)baseline, after 3 months of treatment
Change in distance walked in 6 minutesbaseline, after 3 months of treatment
Secondary Outcome Measures
NameTimeMethod
Change in pulmonary artery pressure (PAP)baseline, after 3 months of treatment
Change in chronic heart failure indexbaseline, after 3 months of treatment

questionnaire

Change in quality of life by SF-36 questionnairebaseline, after 3 months of treatment
Change in cardiac index (CI)baseline, after 3 months of treatment
Change in venous oxygen saturation (SvO2 sat.)baseline, after 3 months of treatment
Change in dyspnea/fatigue ratingbaseline, after 3 months of treatment
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