MedPath

Clinical Study to Compare the Efficacy and Safety of Ponesimod to Placebo in Subjects With Active Relapsing Multiple Sclerosis Who Are Treated With Dimethyl Fumarate (Tecfidera®)

Phase 3
Terminated
Conditions
Multiple Sclerosis
Interventions
Other: Placebo
Registration Number
NCT02907177
Lead Sponsor
Actelion
Brief Summary

This clinical study compares the efficacy, safety, and tolerability of therapy with ponesimod vs placebo in subjects with active RMS who are treated with DMF (Tecfidera®).

Detailed Description

The study will assess the efficacy, safety, and tolerability of add-on therapy with ponesimod 20 mg vs placebo in adult participants with active relapsing multiple sclerosis (RMS) who are treated with dimethyl fumarate (DMF). Approximately 600 participants who have been receiving DMF for at least 6 months will be randomized in a 1:1 ratio to ponesimod 20 mg or placebo. The study consists of the following study periods: Pre-randomization period; Treatment period; Post-treatment observation period. The study includes one ponesimod treatment arm at the maintenance dose of 20 mg o.d. corresponding to the optimal dose when used as monotherapy based on the Phase 2 dose-finding trial and its ongoing extension. The study includes a placebo comparator arm, but all patients will remain on DMF background therapy throughout the study. Moreover, participants who experience a confirmed relapse or an event of 24-week confirmed disability accumulation (DMF) while on study drug will have the option to switch to an alternative treatment. The treatment period has a variable duration from a minimum of 60 weeks (for the last subject randomized) to a maximum of 156 weeks for the first subjects randomized in the trial and includes a gradual up-titration of ponesimod from a 2 mg starting dose to a 20 mg maintenance dose over a period of 14 days. The total duration of the study will be approximately up to 167 weeks.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
136
Inclusion Criteria
  • Signed informed consent prior to initiation of any study-mandated procedure.
  • Women of childbearing potential must have a negative pregnancy test and use reliable methods of contraception
  • Presenting with a diagnosis of MS as defined by the revised (2010) McDonald Diagnostic Criteria for MS with relapsing course from onset (i.e., relapsing-remitting multiple sclerosis (RRMS), or secondary progressive multiple sclerosis (SPMS) with superimposed relapses).
  • Ongoing treatment with DMF for at least 6 months prior to screening
  • Active disease after at least 3 months of DMF treatment
  • Ambulatory and with an EDSS score between 0 and 6.0 (inclusive).
Exclusion Criteria
  • Lactating or pregnant women and women intending to become pregnant during the study.
  • Presenting with a diagnosis of MS with progressive course from onset (i.e., primary progressive MS or progressive relapsing MS).
  • Evidence of a relapse of MS with onset within 30 days prior to baseline EDSS assessment.
  • Any circumstances or conditions, which, in the opinion of the investigator, may affect full participation in the study or compliance with the protocol.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PonesimodPonesimodPonesimod
PlaceboPlaceboPlacebo
Primary Outcome Measures
NameTimeMethod
Annualized Confirmed Relapse Rate (ARR)Through study completion, an average of 68 weeks

Relapse: occurrence of acute episode of one or more new or worsened symptoms of Multiple sclerosis (MS), not associated with fever/infection and lasting 24 hours after stable 30 days period. Confirmed relapse: increase from baseline at least 0.5 point Expanded Disability Status Scale (EDSS) score or increase of one point in one, two or three Functional Systems (FS), excluding bowel/bladder and cerebral/mental FS. EDSS and FS scores are based on neurological examination for assessing its impairment in MS. Among eight FS, seven are ordinal clinical rating scales ranging from 0-5 or 6 with higher scale indicates overall functional impairment assessing Visual, Brain Stem, Pyramidal, Cerebellar, Sensory, Bowel/Bladder and Cerebral functions. Rating individual FS scores is used to rate EDSS in conjunction with observations and information concerning gait and use of assistance. EDSS is ordinal clinical rating scale ranging from 0 (normal neurological examination) to 10(death due to MS).

Secondary Outcome Measures
NameTimeMethod
Percentage of Participants With 12-Week Confirmed Disability Accumulation (CDA) as Assessed by Kaplan Meier Estimate at Week 96Week 96

Percentage of participants with 12-week CDA as assessed by Kaplan Meier estimate at week 96 was defined as an increase of at least 1.5 in Expanded Disability Status Scale (EDSS) for participants with a baseline EDSS score of 0.0 or an increase of at least 1.0 in EDSS for participants with a baseline EDSS score of 1.0 to 5.0, or an increase of at least 0.5 in EDSS for participants with a baseline EDSS score greater than or equal to (\>=) 5.5, which was confirmed after 12 weeks. Baseline EDSS was defined as the last EDSS score recorded prior to randomization. EDSS is an ordinal clinical rating scale ranging from 0 (normal neurological examination) to 10 (death due to MS).

Percentage of Participants Experiencing a Confirmed Relapse as Assessed by Kaplan Meier Estimate at Week 96Week 96

Percentage of participants experiencing a confirmed relapse as assessed by Kaplan Meier estimate at week 96 was reported. The time to first confirmed relapse (in days) is defined as \[Date of first confirmed relapse minus Date of randomization plus 1\] in days. Relapse: Occurrence of acute episode of one or more new symptoms or worsened symptoms of Multiple sclerosis (MS), not related with fever/infection and lasting 24 hours after 30 days stable period.

Number of Participants With Adverse Events (AEs) as a Measure of Safety and TolerabilityUp to 147 Weeks

An AE is any untoward medical event that occurs in a participants administered an investigational product, and it does not necessarily indicate only events with clear causal relationship with the relevant investigational product.

Trial Locations

Locations (119)

Associated Neurologists

🇺🇸

Danbury, Connecticut, United States

Los Angeles Biomedical Research Institute at Harbor-UCLA Medical Center

🇺🇸

Torrance, California, United States

OhioHealth Research Institute

🇺🇸

Columbus, Ohio, United States

Hospital of the University of Pennsylvania

🇺🇸

Philadelphia, Pennsylvania, United States

MS Ambulanz Maida

🇦🇹

Wien, Austria

"University Multiprofile Hospital for Active Treatment - Alexandrovska" EAD, Neurology Clinic

🇧🇬

Sofia, Bulgaria

University Multiprofile Hospital for Active Treatment "Sv. Ivan Rilski" EAD, Neurology Clinic

🇧🇬

Sofia, Bulgaria

Henry Ford Health System - Neurology

🇺🇸

Detroit, Michigan, United States

Neurology and Neuromuscular Center

🇺🇸

Oklahoma City, Oklahoma, United States

Neurology Center of San Antonio

🇺🇸

San Antonio, Texas, United States

IRCCS NEUROMED - Istituto Neurologico Mediterraneo - Unità Operativa di Neurologia I

🇮🇹

Pozzilli, Italy

Neurology Associates - MS Center of Greater Orlando

🇺🇸

Maitland, Florida, United States

Care Access Research - Santa Clarita

🇺🇸

Santa Clarita, California, United States

Aalborg Universitetshospital, Skleroseklinikken Neurologisk afdelning

🇩🇰

Aalborg, Denmark

Pardubicka krajska nemocnice, MS Centrum

🇨🇿

Pardubice, Czechia

Neurology Assoc of Ormond Beach - CNS Trials

🇺🇸

Ormond Beach, Florida, United States

University of Alberta

🇨🇦

Edmonton, Canada

Glostrup Hospital, Neurologisk afdelning

🇩🇰

Glostrup, Denmark

Riverhills Healthcare, Inc.

🇺🇸

Cincinnati, Ohio, United States

Hôpital Universitaire Carémeau, Service de Neurologie

🇫🇷

Nimes, France

Hopital Gui de Chauliac - CHU Montpellier

🇫🇷

Montpellier, France

The MS Center of Vero Beach

🇺🇸

Vero Beach, Florida, United States

Nemocnice Jihlava, Neurologické oddělení

🇨🇿

Jihlava, Czechia

Bradenton Research Center

🇺🇸

Bradenton, Florida, United States

Fort Wayne Neurological Center - North Office

🇺🇸

Fort Wayne, Indiana, United States

Univ of New Mexico - Health Sciences Center

🇺🇸

Albuquerque, New Mexico, United States

Austin Health - Neuro-Immunology Clinical Research, Education and Support Service

🇦🇺

Heidelberg, Victoria, Australia

SC3 Research - Pasadena

🇺🇸

Pasadena, California, United States

AOU San Martino di Genova, Dipartimento di Neuroscienze, Riabilitazione, Oftalmologia, Genetica e Scienze Materno-Infantili (DINOGMI)

🇮🇹

Genova, Italy

Uzsoki utcai Kórház, Neurológiai Osztály

🇭🇺

Budapest, Hungary

AFL Arzneimittelforschung Leipzig GmbH

🇩🇪

Leipzig, Germany

Universitätsklinikum Giessen Klinik und Poliklinik für Neurologie

🇩🇪

Giessen, Germany

Fakultní nemocnice Hradec Králové, Neurologická klinika

🇨🇿

Hradec Králové, Czechia

CHRU de Lille - Hôpital Roger Salengro, Service de Neurologie

🇫🇷

Lille, France

Centre Hospitalier Sud Francilien - Service de Neurologie

🇫🇷

Corbeil-Essonnes, France

Fakultní nemocnice u sv. Anny Brno, RS Centrum

🇨🇿

Brno, Czechia

Hôpital Avicenne, Service de Neurologie

🇫🇷

Bobigny, France

CHU de Dijon - Hôpital François Miterrand, Service de Neurologie

🇫🇷

Dijon, France

Hosp Gabriel Montpied, Dept Neurology

🇫🇷

Clermont Ferrand, France

Medical Center of Athens - Neurology Dpt

🇬🇷

Marousi, Greece

CHI POISSY-Saint Germay en Laye_Service de Neurologie et Réeducation

🇫🇷

Poissy, France

Hosp Pontchaillou, Dept Cardiology

🇫🇷

Rennes, France

Hosp Charles Nicolle Dept Neurology

🇫🇷

Rouen, France

Fondazione Istituto San Raffaele , Unità Operativa di Neurologia

🇮🇹

Cefalù, Italy

Università degli Studi di Firenze - Azienda Ospedaliero Universitaria Careggi - CTO - SOD Neurologia 2

🇮🇹

Firenze, Italy

Medizinische Hochschule Hannover, Neurologie

🇩🇪

Hannover, Germany

Naval Hospital of Athens - Neurology Dpt

🇬🇷

Athens, Greece

General Hospital of Thessaloniki

🇬🇷

Thessaloniki, Greece

Istituto Neurologico Carlo Besta, UOC Neurologia 4, Neuroimmunologia e Malattie Neuromuscolari, Centro Sclerosi Multipla

🇮🇹

Milano, Italy

Azienda Ospedaliera Universitaria (AOU) "Federico II" - Centro Regionale Per la Sclerosi Multipla c/o Clinica Neurologica II - Dipartimento di Scienze

🇮🇹

Napoli, Italy

AOU Università degli Studi della Campania L. Vanvitelli - I° Policlinico - DAI di Medicina Interna e Specialistica CS, Centro Sclerosi Multipla

🇮🇹

Napoli, Italy

Azienda Ospedaliero Universitaria San Luigi Gonzaga - Centro Sclerosi Multipla CRESM

🇮🇹

Orbassano, Italy

Azienda Ospedaliera Universitaria Senese - Dipartimento di Scienze Neurologiche e neurosensoriali - UOSA Neurologia Sperimentale

🇮🇹

Siena, Italy

Unidad de Investigacion en Salud de Chihuahua SC, Médica Sur, Unidad de Neurociencias

🇲🇽

Tlalpan, DF, Mexico

Uniwersytecki Szpital Kliniczny w Bialymstoku, Klinika Neurologii i Oddziat Udarowy

🇵🇱

Bialystok, Poland

Azienda Ospedaliera S. Andrea di Roma - Unità Operativa Complessa di Neurologia

🇮🇹

Roma, Italy

B&B Robert Bonek, Pawel Bochniak S.C

🇵🇱

Bydgoszcz, Poland

Neuro-Medic Janusz Zbrojkiewicz Poradnia Weilospecjalistyczna

🇵🇱

Katowice, Poland

Centrum Terapii SM

🇵🇱

Katowice, Poland

Neuro-Clinic, LLC

🇷🇺

Moscow, Russian Federation

Complejo Hospitalario Universitario de Santiago de Compostela (CHUS) - Neurology Department 2

🇪🇸

Santiago de Compostela, Spain

Hospital Santa Caterina - Neurology Department

🇪🇸

Salt, Spain

Hosp Gregorio Marañón, Neurology

🇪🇸

Madrid, Spain

Univeritätsspital Basel Neurologie, Neurologische Klinik und Poliklinik

🇨🇭

Basel, Switzerland

Queen Square MS Centre / NMR research Unit UCL Institute of Neurology

🇬🇧

London, United Kingdom

Nuffield Department of Clinical Neurosciences, John Radcliffe Hospital

🇬🇧

Oxford, United Kingdom

Moscow State Budgetary Healthcare Institution Pirogov City Clinical Hospital No. 1 of Moscow Health Department

🇷🇺

Moscow, Russian Federation

Moscow State Budgetary Healthcare Institution City Clinical Hospital No. 24 of Moscow Health Department

🇷🇺

Moscow, Russian Federation

Helios Klinikum Erfurt

🇩🇪

Erfurt, Germany

Gemeinschaftspraxis Dr. med. Joachim Springub / Wolfgang Schwarz, Studienzentrum Nord-West (Study Center)

🇩🇪

Westerstede, Germany

Universitätsklinikum Münster, Klinik für Allgemeine Neurologie

🇩🇪

Münster, Germany

Medizinzentrum Siegerland Weidenau

🇩🇪

Siegen, Germany

University of Kansas Med Center

🇺🇸

Kansas City, Kansas, United States

Krajská zdravotní a.s. - Nemonice Teplice o.z., RS Centrum

🇨🇿

Teplice, Czechia

Mountain View Clinical Research, Inc

🇺🇸

Denver, Colorado, United States

University of Colorado Hospital

🇺🇸

Aurora, Colorado, United States

Hospital Universitario Virgen Macarena - Neurofisiology Department

🇪🇸

Sevilla, Spain

Advanced Neuroscience Institute

🇺🇸

Franklin, Tennessee, United States

University Hospitals of North Midlands NHS Trust

🇬🇧

Stoke-on-Trent, United Kingdom

Royal Hallamshire Hospital

🇬🇧

Sheffield, United Kingdom

Aeginition Hospital - Neurology Department

🇬🇷

Athens, Greece

Neuro-Pain Medical Center

🇺🇸

Fresno, California, United States

UAB Dpt of Neurology

🇺🇸

Birmingham, Alabama, United States

Suncoast Neuroscience Associates, Inc

🇺🇸

Saint Petersburg, Florida, United States

NYU Langone Medical Center - MS Comprehensive Care Center

🇺🇸

New York, New York, United States

Thomas Jefferson University Hospital - Dpt Neurology MS Center

🇺🇸

Philadelphia, Pennsylvania, United States

Medizinische Universität Wien, Universitätsklinik für Neurologie

🇦🇹

Wien, Austria

"Multiprofile Hospital for Active Treatment of Neurology and Psychiatry - Sveti Naum" EAD - Neurology Clinic for Movement Disorders

🇧🇬

Sofia, Bulgaria

Hospital - Revalidatie & MS Centrum Overpelt_Neurology Department

🇧🇪

Overpelt, Belgium

Hôpital Central - CHU Nancy, Département Neurologie

🇫🇷

Nancy, France

Neurologische Klinik und Poliklinik - Universitätsklinikum Carl Gustav Carus, Zentrum für klinische Neurowissenschaften

🇩🇪

Dresden, Germany

Universitätsmedizin Greifswald - Körperschaft des öffentlichen Rechts - Klinik und Poliklinik für Neurologie

🇩🇪

Greifswald, Germany

Zentrum für klinische Forschung Dr. med. Irma Schöll

🇩🇪

Bad Homburg, Germany

NeuroPoint GmbH, Gesellschaft für vorbeugende Gesundheitspflege

🇩🇪

Ulm, Germany

401 Military Hospital of Athens - Neurology Dept

🇬🇷

Athens, Greece

Desarrollo Ético en Investigación Clínica S.C .

🇲🇽

Guadalajara, Jalisco, Mexico

COPERNICUS - Podmiot Leczniczy Sp. z o.o.

🇵🇱

Gdansk, Poland

Unidad de Investigación de Salud en Chihuahua

🇲🇽

Chihuahua, Mexico

State Budgetary Healthcare Institution Regional Clinical Hospital No 3

🇷🇺

Chelyabinsk, Russian Federation

Center of Professional Therapy, LLC

🇷🇺

Krasnodar, Russian Federation

Moscow State Budgetary Healthcare Institution Filatov City Clinical Hospital No.15 of Moscow Health Department

🇷🇺

Moscow, Russian Federation

Hospital Santa Creu I Sant Pau - Neurology Dpt

🇪🇸

Barcelona, Spain

Hosp Virgen de la Arrixaca, Neurology

🇪🇸

El Palmar, Spain

Hospital Clinico San Carlos, Neurology

🇪🇸

Madrid, Spain

Centro de Neurologia Avanzada, Neurology

🇪🇸

Sevilla, Spain

Axis Heilsa S. de R.L. de C.V. (Althian)

🇲🇽

Nuevo Leon, Monterrey, Mexico

Hospital - Universitair Gent __Neurology Department

🇧🇪

Gent, Belgium

Hospital universitair Brussels_neurology department

🇧🇪

Brussels, Belgium

Pest Megyei Flór Ferenc Kórház, Neurológia és Stroke ambulancia

🇭🇺

Kistarcsa, Hungary

WroMedica, J. Bielicka A. Strzałkowska SC

🇵🇱

Wroclaw, Poland

Valeomed EGÉSZSÉGÜGYI KÖZPONT

🇭🇺

Esztergom, Hungary

Centro Hospitalar de Lisboa Central

🇵🇹

Lisboa, Portugal

Hospital de Santa Maria - Neurology Department

🇵🇹

Lisboa, Portugal

Centrum Kompleksowej Rehabilitacji

🇵🇱

Konstancin-Jeziorna, Poland

Centrum Opieki Zdrowotnej Orkan - Med.

🇵🇱

Ksawerów, Poland

Instytut Psychiatrii i Neurologii, II Klinika Neurologiczna

🇵🇱

Warszawa, Poland

Centro Hospitalar de São João, E.P.E. - Hospital de São João - Neurology Department

🇵🇹

Porto, Portugal

Ospedale Regionale di Lugano - Civico e Italiano, Neurologia, Lugano

🇨🇭

Lugano, Switzerland

MidAmerica Neuroscience Research Foundation/Rowe Neurology

🇺🇸

Lenexa, Kansas, United States

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