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A Study Evaluating the Safety and Efficacy of Venetoclax in Combination With Trastuzumab Emtansine in Patients With Previously Treated HER2-Positive Locally Advanced or Metastatic Breast Cancer

Phase 1
Terminated
Conditions
Breast Cancer
Interventions
Registration Number
NCT04298918
Lead Sponsor
Hoffmann-La Roche
Brief Summary

This two-part study is composed of two stages: a Phase Ib stage consisting of a dose-escalation phase and an expansion phase; and a Phase II, randomized, placebo-controlled, double-blind, multicenter stage. The Phase Ib stage will assess the safety and tolerability, determine the maximum tolerated dose (MTD) and the recommended Phase II dose (RP2D), and evaluate the preliminary efficacy of trastuzumab emtansine in combination with venetoclax in participants with previously treated human epidermal growth factor receptor 2 (HER2) positive unresectable locally advanced breast cancer (LABC) or metastatic breast cancer (MBC). Additional patients may be enrolled in an expansion phase to evaluate the safety, tolerability, and efficacy of trastuzumab emtansine in combination with venetoclax at RP2D in patients with previously treated HER2-positive LABC or MBC who have previously received either trastuzumab emtansine or trastuzumab deruxtecan (DS-8201a). The Phase II randomized stage will evaluate the safety, efficacy, tolerability, and pharmacokinetics of trastuzumab emtansine in combination with venetoclax at RP2D compared with trastuzumab emtansine plus placebo in participants with previously treated HER2-positive LABC or MBC who have not received prior trastuzumab emtansine therapy, either alone or in combination with other anti-cancer therapies.

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
1
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Randomized Phase II Arm 1PlaceboParticipants were to receive trastuzumab emtansine + placebo.
Dose Expansion PhaseVenetoclaxParticipants were to receive venetoclax at the Phase II Recommended Dose (RP2D) in combination with trastuzumab emtansine.
Dose Expansion PhaseTrastuzumab emtansineParticipants were to receive venetoclax at the Phase II Recommended Dose (RP2D) in combination with trastuzumab emtansine.
Dose Escalation PhaseVenetoclaxParticipants received venetoclax in combination with a fixed dose of trastuzumab emtansine.
Dose Escalation PhaseTrastuzumab emtansineParticipants received venetoclax in combination with a fixed dose of trastuzumab emtansine.
Randomized Phase II Arm 1Trastuzumab emtansineParticipants were to receive trastuzumab emtansine + placebo.
Randomized Phase II Arm 2VenetoclaxParticipants were to receive trastuzumab emtansine + venetoclax.
Randomized Phase II Arm 2Trastuzumab emtansineParticipants were to receive trastuzumab emtansine + venetoclax.
Primary Outcome Measures
NameTimeMethod
Phase II: Progression-Free Survival (PFS)Up to 30 months

The study was terminated by the Sponsor. Only 1 participant was enrolled in this study. Based on the low enrolment number, no data is reported here in order to protect and maintain participant privacy/confidentiality.

Dose Escalation: Number of Participants With Adverse EventsBaseline up until 28 days after the last dose of study drug or until initiation of new systemic anti-cancer therapy, whichever occurs first (up to a maximum of 20 weeks).

The study was terminated by the Sponsor. Only 1 participant was enrolled in this study. Based on the low enrolment number, no data is reported here in order to protect and maintain participant privacy/confidentiality.

Expansion Phase: Objective Response Rate (ORR)Up to 30 months

The study was terminated by the Sponsor. Only 1 participant was enrolled in this study. Based on the low enrolment number, no data is reported here in order to protect and maintain participant privacy/confidentiality.

Phase II: ORRUp to 30 months

The study was terminated by the Sponsor. Only 1 participant was enrolled in this study. Based on the low enrolment number, no data is reported here in order to protect and maintain participant privacy/confidentiality.

Secondary Outcome Measures
NameTimeMethod
Phase II: Serum Concentration of Trastuzumab EmtansineAt pre-defined time points from Cycle 1 Day 1 through Cycle 4 Day 1 (cycle = 21 days)

The study was terminated by the Sponsor. Only 1 participant was enrolled in this study. Based on the low enrolment number, no data is reported here in order to protect and maintain participant privacy/confidentiality.

All Phases: Plasma Concentration of VenetoclaxAt pre-defined time points from Cycle 1 Day 8 and/or Cycle 2 Day 1 through Cycle 4 Day 1 (cycle = 21 days)

The study was terminated by the Sponsor. Only 1 participant was enrolled in this study. Based on the low enrolment number, no data is reported here in order to protect and maintain participant privacy/confidentiality.

Expansion Phase and Phase II: Duration of Response (DOR)Up to 30 months

The study was terminated by the Sponsor. Only 1 participant was enrolled in this study. Based on the low enrolment number, no data is reported here in order to protect and maintain participant privacy/confidentiality.

Phase II: Overall Survival (OS)Randomization to death from any cause (up to 30 months)

The study was terminated by the Sponsor. Only 1 participant was enrolled in this study. Based on the low enrolment number, no data is reported here in order to protect and maintain participant privacy/confidentiality.

Expansion Phase and Phase II: Number of Participants With Adverse EventsBaseline up until 28 days after the last dose of study drug or until initiation of new systemic anti-cancer therapy, whichever occurs first (up to a maximum of 20 weeks).

The study was terminated by the Sponsor. Only 1 participant was enrolled in this study. Based on the low enrolment number, no data is reported here in order to protect and maintain participant privacy/confidentiality.

Phase II: Number of Participants With Anti-Drug Antibodies (ADAs) to Trastuzumab EmtansineUp to 30 months

The study was terminated by the Sponsor. Only 1 participant was enrolled in this study. Based on the low enrolment number, no data is reported here in order to protect and maintain participant privacy/confidentiality.

Trial Locations

Locations (3)

Peter MacCallum Cancer Center

🇦🇺

East Melbourne, Victoria, Australia

Asan Medical Center

🇰🇷

Seoul, Korea, Republic of

Samsung Medical Center

🇰🇷

Seoul, Korea, Republic of

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