MedPath

A Study of Combination Therapy With Venetoclax, Daratumumab and Dexamethasone (With and Without Bortezomib) in Participants With Relapsed or Refractory Multiple Myeloma

Phase 2
Active, not recruiting
Conditions
Multiple Myeloma
Interventions
Registration Number
NCT03314181
Lead Sponsor
AbbVie
Brief Summary

This is a study of venetoclax, daratumumab, and dexamethasone with and without bortezomib combination therapy to evaluate safety, tolerability, and efficacy of these combinations in participants with relapsed or refractory multiple myeloma. The study will consist of 3 distinct parts: Part 1 includes participants with t(11;14) positive relapsed/refractory (R/R) multiple myeloma who will receive venetoclax in combination with daratumumab and dexamethasone (VenDd); Part 2 includes participants with R/R multiple myeloma who will receive venetoclax in combination with daratumumab, bortezomib, and dexamethasone (VenDVd); Part 3 includes participants with t(11;14) positive R/R multiple myeloma who will receive venetoclax in combination with daratumumab and dexamethasone (VenDd) or daratumumab, bortezomib, and dexamethasone (DVd).

Part 1 and Part 2 are non-randomized and will be initiated with a dose-escalation phase in which increasing doses of venetoclax will be given with fixed doses of daratumumab and dexamethasone (Part 1a) or with fixed doses of daratumumab, bortezomib, and dexamethasone (Part 2a). Each dose escalation phase will be followed by a single-arm, open-label expansion phase. Part 3 will include a randomized, open-label expansion phase with participants receiving venetoclax in combination with daratumumab and dexamethasone (VenDd) or daratumumab, bortezomib, and dexamethasone (DVd).

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
156
Inclusion Criteria
  • Eastern Cooperative Oncology Group (ECOG) performance status <= 2.
  • Participant has relapsed or refractory multiple myeloma with documented evidence of progression that occurred during or after the participant's last treatment regimen based on investigator's determination of International Myeloma Working Group (IMWG) criteria.
  • Measurable disease confirmed by central lab at Screening, defined by at least 1 of the following: Serum M-protein >= 1.0 g/dL (>= 10 g/L), OR Urine M-protein >= 200 mg/24 hours, OR Serum free light chain (FLC) >= 10 mg/dL, provided serum FLC ratio is abnormal in participants who do not have measurable disease by Serum Protein Electrophoresis (SPEP) or Urine Protein Electrophoresis (UPEP) criteria.
  • Participant has received previous multiple myeloma treatment as defined in the protocol.
  • Bone marrow aspirate samples have been collected.
  • To qualify for Part 1 and 3, the participant must be t(11;14) positive as determined by an analytically validated Fluorescent In Situ Hybridization (FISH) assay per central laboratory testing.
  • Participants must have adequate hematologic, renal and hepatic function.
Exclusion Criteria
  • Previous treatment with venetoclax or other B-Cell Lymphoma 2 (BCL-2) inhibitor

  • For participants in Parts 1 and 2: Previous treatment with daratumumab or other anti-CD38 therapy. For participants in Part 3: Prior daratumumab or other anti-CD38 antibody therapy exposure that meets ANY of the following criteria:

    • Failure to achieve at least a PR to most recent therapy with daratumumab or other anti-CD38 therapy.
    • Daratumumab or other anti-CD38 antibody therapy was discontinued due to toxicity.
    • Relapse within 60 days of intensive treatment (at least every other week) of daratumumab or other anti-CD38 antibody therapy.
    • Prior treatment with daratumumab or other anti-CD38 antibody within 6 months prior to first dose of study drug.
  • For participants in Part 2 and 3:

    • Participant is refractory to any proteasome inhibitor, defined as progression on or within 60 days of the last dose of a proteasome inhibitor-containing regimen.
    • Participant has had prior treatment with proteasome inhibitor within 60 days prior to first dose of study drug.
  • Treatment with anti-myeloma chemotherapy, radiotherapy, biological, immunotherapy or an investigational therapy, including targeted small molecule agents within 2 weeks or 5 half-lives (whichever is longer and/or applicable) before first dose.

  • Treatment with anti-myeloma monoclonal antibodies within 6 weeks prior to first dose.

  • Recent corticosteroid therapy at a cumulative dose equivalent to >= 140 mg of prednisone, cumulative dose equivalent to >= 40 mg of dexamethasone, or a single dose equivalent to >= 40 mg of dexamethasone within 2 weeks prior the first dose of study drug.

  • Known central nervous system involvement of multiple myeloma.

  • Significant history of medical conditions as listed in the protocol.

  • History of other active malignancies including myelodysplatic syndromes (MDS) within the past 3 years with the exceptions of:

    • Basal cell carcinoma of the skin or localized squamous cell carcinoma of the skin.
    • Prostate cancer Gleason grade 6 or lower AND with stable Prostate Specific Antigen (PSA) levels off treatment
    • Previous malignancy with no evidence of disease confirmed and surgically resected (or treated with other modalities) with curative intent and unlikely to impact survival during the duration of the study.
  • Known active severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) infection.

  • Has a hypersensitivity or allergy to any of the components of study therapy, excipient or boron.

  • Known allergies, hypersensitivities, or intolerance to monoclonal antibodies or human proteins, or their excipients, or known sensitivity to mammalian-derived products (see daratumumab prescribing information).

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Arm A, Part 1a: VenDd Dose EscalationDaratumumabVenetoclax (Ven) various doses administered orally, once daily (QD) in combination with daratumumab (D) (1800 mg subcutaneous injection (preferred) or 16 mg/kg intravenous \[IV\]) administered in accordance with prescribing information and dexamethasone (d) (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm A, Part 1a: VenDd Dose EscalationDexamethasoneVenetoclax (Ven) various doses administered orally, once daily (QD) in combination with daratumumab (D) (1800 mg subcutaneous injection (preferred) or 16 mg/kg intravenous \[IV\]) administered in accordance with prescribing information and dexamethasone (d) (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm A, Part 1a: VenDd Dose EscalationVenetoclaxVenetoclax (Ven) various doses administered orally, once daily (QD) in combination with daratumumab (D) (1800 mg subcutaneous injection (preferred) or 16 mg/kg intravenous \[IV\]) administered in accordance with prescribing information and dexamethasone (d) (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm B, Part 1b: VenDd Dose ExpansionDexamethasoneVenetoclax at a dose determined by the dose-escalation phase, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information and dexamethasone (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm B, Part 1b: VenDd Dose ExpansionDaratumumabVenetoclax at a dose determined by the dose-escalation phase, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information and dexamethasone (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm B, Part 1b: VenDd Dose ExpansionVenetoclaxVenetoclax at a dose determined by the dose-escalation phase, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information and dexamethasone (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm D, Part 2a: VenDVd Dose EscalationDexamethasoneVenetoclax at various doses administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection \[preferred\] or IV) Cycles 1-8, Days 1, 4, 8 and 11), and dexamethasone (oral or IV) 20 mg Cycles 1 - 3, Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 20 mg Cycles 4-8, Days 1,2,4,5,8,9,11 and 12; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) Cycle 9+.
Arm D, Part 2a: VenDVd Dose EscalationDaratumumabVenetoclax at various doses administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection \[preferred\] or IV) Cycles 1-8, Days 1, 4, 8 and 11), and dexamethasone (oral or IV) 20 mg Cycles 1 - 3, Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 20 mg Cycles 4-8, Days 1,2,4,5,8,9,11 and 12; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) Cycle 9+.
Arm D, Part 2a: VenDVd Dose EscalationVenetoclaxVenetoclax at various doses administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection \[preferred\] or IV) Cycles 1-8, Days 1, 4, 8 and 11), and dexamethasone (oral or IV) 20 mg Cycles 1 - 3, Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 20 mg Cycles 4-8, Days 1,2,4,5,8,9,11 and 12; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) Cycle 9+.
Arm D, Part 2a: VenDVd Dose EscalationBortezomibVenetoclax at various doses administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection \[preferred\] or IV) Cycles 1-8, Days 1, 4, 8 and 11), and dexamethasone (oral or IV) 20 mg Cycles 1 - 3, Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 20 mg Cycles 4-8, Days 1,2,4,5,8,9,11 and 12; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) Cycle 9+.
Arm E, Part 2b: VenDVd Dose ExpansionDexamethasoneVenetoclax at dose determined by the dose-escalation phase, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection) Cycles 1-8, Days 1, 4, 8 and 11, and dexamethasone (oral or IV) 20 mg Cycles 1 - 3, Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 20 mg Cycles 4-8, Days 1,2,4,5,8,9,11 and 12; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) Cycle 9+.
Arm E, Part 2b: VenDVd Dose ExpansionDaratumumabVenetoclax at dose determined by the dose-escalation phase, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection) Cycles 1-8, Days 1, 4, 8 and 11, and dexamethasone (oral or IV) 20 mg Cycles 1 - 3, Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 20 mg Cycles 4-8, Days 1,2,4,5,8,9,11 and 12; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) Cycle 9+.
Arm E, Part 2b: VenDVd Dose ExpansionVenetoclaxVenetoclax at dose determined by the dose-escalation phase, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection) Cycles 1-8, Days 1, 4, 8 and 11, and dexamethasone (oral or IV) 20 mg Cycles 1 - 3, Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 20 mg Cycles 4-8, Days 1,2,4,5,8,9,11 and 12; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) Cycle 9+.
Arm E, Part 2b: VenDVd Dose ExpansionBortezomibVenetoclax at dose determined by the dose-escalation phase, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection) Cycles 1-8, Days 1, 4, 8 and 11, and dexamethasone (oral or IV) 20 mg Cycles 1 - 3, Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 20 mg Cycles 4-8, Days 1,2,4,5,8,9,11 and 12; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) Cycle 9+.
Arm F: VenDd Dose ExpansionDexamethasoneVenetoclax at a pre-determined dose, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information and dexamethasone (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm F: VenDd Dose ExpansionDaratumumabVenetoclax at a pre-determined dose, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information and dexamethasone (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm F: VenDd Dose ExpansionVenetoclaxVenetoclax at a pre-determined dose, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information and dexamethasone (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm G: VenDd Dose ExpansionDaratumumabVenetoclax at a pre-determined dose, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information and dexamethasone (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm G: VenDd Dose ExpansionVenetoclaxVenetoclax at a pre-determined dose, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information and dexamethasone (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm G: VenDd Dose ExpansionDexamethasoneVenetoclax at a pre-determined dose, administered orally QD in combination with daratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information and dexamethasone (oral or IV) 40 mg weekly (or 20 mg weekly, if necessary, as described in the protocol).
Arm H: DVd DoseDaratumumabDaratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection) Cycles 1-8: Days 1, 4, 8 and 11, and dexamethasone (oral or IV) 20 mg on Cycles 1 - 3: Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) on Cycles 4-8: Days 1,2,4,5,8,9,11 and 12; 20 mg monthly for Cycles 9+: Day 1
Arm H: DVd DoseDexamethasoneDaratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection) Cycles 1-8: Days 1, 4, 8 and 11, and dexamethasone (oral or IV) 20 mg on Cycles 1 - 3: Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) on Cycles 4-8: Days 1,2,4,5,8,9,11 and 12; 20 mg monthly for Cycles 9+: Day 1
Arm H: DVd DoseBortezomibDaratumumab (1800 mg subcutaneous injection (preferred) or 16 mg/kg IV) administered in accordance with prescribing information, bortezomib (1.3 mg/m2 subcutaneous injection) Cycles 1-8: Days 1, 4, 8 and 11, and dexamethasone (oral or IV) 20 mg on Cycles 1 - 3: Days 1, 2, 4, 5, 8, 9, 11,12 and 15; 40 mg weekly (or 20 mg weekly, if necessary as described in the protocol) on Cycles 4-8: Days 1,2,4,5,8,9,11 and 12; 20 mg monthly for Cycles 9+: Day 1
Primary Outcome Measures
NameTimeMethod
Overall Response Rate (ORR)Up to approximately 3.5 years after the last participant is enrolled

ORR is defined as the percentage of participants with documented partial response (PR) or better based on International Myeloma Working Group (IMWG) criteria.

Duration of Response (DOR)Up to approximately 3.5 years after the last participant is enrolled

DOR is defined as the number of days from the participant's date of first documented response (PR or better) to the date of first documented disease progression or death due to multiple myeloma, whichever occurs first.

Very Good Partial Response or Better Response Rate (VGPR)Up to approximately 3.5 years after the last participant is enrolled

VGPR or better response rate is defined as the proportion of participants with documented VGPR or better (sCR, CR. or VGPR) based on IMWG criteria.

Complete Response (CR) or Better RateUp to approximately 3.5 years after the last participant is enrolled

CR or better response is defined as the percentage of participants with documented response of CR or better (stringent complete response \[sCR\] or CR) based on IMWG criteria.

Time to Response (TTR)Up to approximately 3.5 years after the last participant is enrolled

TTR is defined as the number of days from the date of treatment start (for subjects enrolled prior to randomization start) or randomization (for randomized subjects) to the date of first documented response of PR or better.

Time to Progression (TTP)Up to approximately 3.5 years after the last participant is enrolled

TTP is defined as the number of days from the date of treatment start (for subjects enrolled prior to randomization start) or randomization (for randomized subjects) to the date of first documented PD or death due to MM, whichever occurs first.

Progression-Free Survival (PFS)Up to approximately 3.5 years after the last participant is enrolled

PFS is defined as the number of days from the date of treatment start (for subjects enrolled prior to randomization start) or randomization (for randomized subjects) to the date of the first documented PD or death due to any cause, whichever occurs first.

Overall Survival (OS)Up to approximately 3.5 years after the last participant is enrolled

OS is defined as the number of days from the date of treatment start (for subjects enrolled prior to randomization start) or randomization (for randomized subjects) to the date of death.

Secondary Outcome Measures
NameTimeMethod
AUC0-24 of VenetoclaxUp to approximately 1 year

Area under the plasma concentration-time curve (AUC) over the dose interval (AUC0-24) of venetoclax.

Minimal Residual Disease (MRD)Up to 12 months after confirmation of Complete Response (CR) or Stringent Complete Response (sCR)

MRD negativity in bone marrow aspirates is defined at 10\^-5 threshold as assessed by next generation sequencing (NGS) in participants at the time of suspected CR/sCR, and at 6 and 12 months post confirmation of CR/sCR for participants who maintained this response.

Tmax of VenetoclaxUp to approximately 1 year

Time to Cmax (Tmax) of Venetoclax

Cmax of VenetoclaxUp to approximately 1 year

Maximum observed plasma concentration (Cmax) of venetoclax

Trial Locations

Locations (40)

Eastern Health /ID# 165850

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Box Hill, Victoria, Australia

Cross Cancer Institute /ID# 203114

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Edmonton, Alberta, Canada

Kameda General Hospital /ID# 225246

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Kamogawa-shi, Chiba, Japan

Oregon Health and Science University /ID# 166822

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Portland, Oregon, United States

Dana-Farber Cancer Institute /ID# 166886

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Boston, Massachusetts, United States

Univ of Colorado Cancer Center /ID# 167331

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Aurora, Colorado, United States

Beth Israel Deaconess Medical Center /ID# 210904

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Boston, Massachusetts, United States

Emory University, Winship Cancer Institute /ID# 165427

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Atlanta, Georgia, United States

The University of Chicago Medical Center /ID# 165429

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Chicago, Illinois, United States

Atrium Health Carolinas Medical Center /ID# 164948

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Charlotte, North Carolina, United States

Duke Cancer Center /ID# 165104

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Durham, North Carolina, United States

Sygehus Lillebalt, Vejle /ID# 164418

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Vejle, Syddanmark, Denmark

CHU Limoges - Dupuytren 1 /ID# 224759

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Limoges CEDEX 1, Franche-Comte, France

The Kinghorn Cancer Centre /ID# 165431

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Darlinghurst, New South Wales, Australia

Tom Baker Cancer Centre /ID# 167822

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Calgary, Alberta, Canada

Odense University Hospital /ID# 164417

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Odense, Syddanmark, Denmark

University Hospital Cologne /ID# 166037

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Cologne, Germany

AP-HP - Hopital Saint-Louis /ID# 224758

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Paris, France

Gifu Municipal Hospital /ID# 240381

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Gifu-shi, Gifu, Japan

St George Hospital /ID# 171063

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Kogarah, New South Wales, Australia

Duplicate_Roswell Park Comprehensive Cancer Center /ID# 169615

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Buffalo, New York, United States

Weill Cornell Medicine/NYP /ID# 167605

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New York, New York, United States

University of Washington /ID# 164884

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Seattle, Washington, United States

Royal Adelaide Hospital /ID# 171060

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Adelaide, South Australia, Australia

Moffitt Cancer Center /ID# 169614

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Tampa, Florida, United States

Wake Forest Baptist Health /ID# 224447

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Winston-Salem, North Carolina, United States

Duplicate_Royal Perth Hospital /ID# 224895

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Perth, Western Australia, Australia

Duplicate_Aarhus University Hospital /ID# 164509

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Aarhus N, Midtjylland, Denmark

Rigshospitalet /ID# 164420

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Copenhagen Ø, Hovedstaden, Denmark

St Vincent's Hospital Melbourne /ID# 165853

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Fitzroy Melbourne, Victoria, Australia

Universitaetsklinikum Freiburg /ID# 166036

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Freiburg, Baden-Wuerttemberg, Germany

Institut Gustave Roussy /ID# 164807

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Villejuif Cedex, Val-de-Marne, France

Royal Victoria Hospital / McGill University Health Centre /ID# 167824

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Montreal, Quebec, Canada

CHU Poitiers - La miletrie /ID# 164806

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Poitiers, Vienne, France

Hackensack Univ Med Ctr /ID# 225111

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Hackensack, New Jersey, United States

Peter MacCallum Cancer Ctr /ID# 164742

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Melbourne, Victoria, Australia

CHRU Tours - Hopital Bretonneau /ID# 164795

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Tours CEDEX 9, Indre-et-Loire, France

Nagoya City University Hospital /ID# 225273

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Nagoya shi, Aichi, Japan

Matsuyama Red Cross Hospital /ID# 225196

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Matsuyama-shi, Ehime, Japan

CHU de Nantes, Hotel Dieu -HME /ID# 164767

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Nantes, Pays-de-la-Loire, France

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