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Efficacy and Safety of Combination Ambrisentan and Tadalafil in Patients With Portopulmonary Hypertension

Phase 4
Withdrawn
Conditions
Portopulmonary Hypertension
Pulmonary Hypertension
Cirrhosis, Liver
Interventions
Registration Number
NCT03309592
Lead Sponsor
Ochsner Health System
Brief Summary

The purpose of this study is to evaluate the efficacy and safety of the combination of ambrisentan and tadalafil in reducing mPAP to below 35mmHg in patients with moderate to severe Portopulmonary Hypertension (POPH) as a means to candidacy for liver transplantation.

Detailed Description

The outcome of liver transplantation (LT) in the presence of moderate to severe POPH is significantly poor with a 50% reported mortality rate in LT recipients having a mean pulmonary artery pressure (mPAP) \>35 mmHg and 100% when the mPAP is greater than 50 mmHg; therefore, making moderate to severe POPH a contraindication to liver transplants. Those recipients with significant pulmonary artery pressure (PAP) may be denied the opportunity for transplant unless the mPAP is brought below 35 mmHg with medical treatment. This study will test the efficacy \& safety of the combination of using ambrisentan and tadalfil in reducing the Pulmonary Arterial Pressure to below 35 mmHg in patients with moderate to severe POPH as a means to candidacy for liver transplantation.

Recruitment & Eligibility

Status
WITHDRAWN
Sex
All
Target Recruitment
Not specified
Inclusion Criteria
  • Child-Pugh Class Class A & B Cirrhosis
  • mPAP ≥35mmHg
  • Pulmonary Capillary Wedge Pressure (PWCP) <15mmHg on Right Heart Catheterization's (RHCs)
  • mPAP > 50mmHg will be considered eligible unless they are World Health Organization (WHO) Functional Class IV
Exclusion Criteria
  • End stage renal disease on hemodialysis (ESRD on HD)

  • Renal dysfunction and GFR < 30

  • AST, ALT > 5 times the upper limit of normal

  • Total bilirubin ≥ 6.0

  • INR > 2

    • Initially, Child-Pugh Class C patients will be excluded; however, after the first 5 patients are included, if there is no signal of worsening liver function, the protocol may be amended to include patients with Class C cirrhosis.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Combination TherapyAmbrisentan PillQualifying participants will begin combination therapy with ambrisentan pill 5 mg daily and tadalafil pill 20 mg. After one week of therapy, patients will increase tadalafil pill to 40 mg daily and continue ambrisentan pill 5 mg daily. On day 15, patients will increase ambrisentan pill to 10 mg daily and continue at 40 mg of tadalafil pill daily.
Combination TherapyTadalafil PillQualifying participants will begin combination therapy with ambrisentan pill 5 mg daily and tadalafil pill 20 mg. After one week of therapy, patients will increase tadalafil pill to 40 mg daily and continue ambrisentan pill 5 mg daily. On day 15, patients will increase ambrisentan pill to 10 mg daily and continue at 40 mg of tadalafil pill daily.
Primary Outcome Measures
NameTimeMethod
Reduction in mPAP to 35mmHg2 months post initiation of therapy

A Right Heart Catheterization will be performed in order to see if there's a reduction in mPAP to less than 35mmHg from baseline

Secondary Outcome Measures
NameTimeMethod
Post-Transplant Survival Outcome: Alive or Dead at 30 daysPost-op Day 1 and 30

Post-transplant survival comparing subjects with or without history of POPH

Liver Function test measured by AST (iu/L)baseline, 1 month, 2 month, 3 month, 6 month, 9 month, 12 months/end of treatment, 1 month post transplant

AST will be done to monitor and measure the degree of cirrhosis on the liver as well as the overall function of the liver

Right Ventricular (RV) Function in centimetersBaseline, 1-month, 6-month and 12 months post therapy and 1-month post transplant

Tricuspid Annular Plane Systolic Excursion (TAPSE) measured in centimeters

Biomarker of Right ventricular failurebaseline, 1 month, 2 month, 3 month, 6 month, 9 month, 12 months/end of treatment, 1 month post transplant

serum BNP

New York Heart Association Functional classbaseline, 1 month, 2 month, 3 month, 6 month, 9 month, 12 months/end of treatment, 1 month post transplant

NYHA FC will be assessed by clinician at baseline and each subsequent visit

Blood Pressure2 months post therapy

Systemic Blood pressure

mPAP Reduction2 months post initiation of therapy

Percent reduction in mPAP will be assessed and measured from baseline via RHC

Kidney function evaluation through measurement of Creatinine levels (mg/dL)baseline, 1 month, 2 month, 3 month, 6 month, 9 month, 12 months/end of treatment, 1 month post transplant

Comprehensive metabolic panel will be completed at 2 months post therapy to assess kidney function

Liver Function test measured by ALT (iu/L)baseline, 1 month, 2 month, 3 month, 6 month, 9 month, 12 months/end of treatment, 1 month post transplant

ALT test will be done to monitor and measure the degree of cirrhosis on the liver as well as the overall function of the liver

Liver Function test measured by Bilirubin (mg/dL)baseline, 1 month, 2 month, 3 month, 6 month, 9 month, 12 months/end of treatment, 1 month post transplant

Bilirubin test will be done to monitor and measure the degree of cirrhosis on the liver as well as the overall function of the liver

Liver Function test measured by INRbaseline, 1 month, 2 month, 3 month, 6 month, 9 month, 12 months/end of treatment, 1 month post transplant

INR test will be done to monitor and measure the degree of cirrhosis on the liver as well as the overall function of the liver

Right Ventricular (RV) Size in centimetersBaseline, 1-month, 6-month and 12 months post therapy, 1 month post transplant

To measure Right Ventricular Size in centimeters

Right Ventricular (RV) Qualitative Systolic Function: assessment that is categorized as normal, mildly depressed, moderately depressed or severely depressedBaseline, 1-month, 6-month and 12 months post therapy, 1 month post transplant

To measure Right Ventricular Qualitative Systolic Function assessment that is categorized as normal, mildly depressed, moderately depressed or severely depressed

Change in 6 Minute Walk Distancebaseline, 1 month, 2 month, 3 month, 6 month, 9 month, 12 months/end of treatment, 1 month post transplant

6 Minute walk will be performed at baseline and each study visit

Trial Locations

Locations (1)

Ochsner Clinic Foundation

🇺🇸

New Orleans, Louisiana, United States

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