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Assessing Long Term Safety and Tolerability of PXT3003 in Patients With Charcot-Marie-Tooth Disease Type 1A

Phase 3
Active, not recruiting
Conditions
Charcot-Marie-Tooth Disease, Type IA
Interventions
Registration Number
NCT03023540
Lead Sponsor
Pharnext S.C.A.
Brief Summary

All randomised patients with Charcot-Marie-Tooth Type 1A (CMT1A) who completed the primary study CLN-PXT3003-02, i.e. treatment with PXT3003 or placebo, are eligible to continue in the extension study CLN-PXT3003-03.

Period 1: Patients randomised to PXT3003 dose 1 or placebo in the primary study (CLN-PXT3003-02) continued in the extension study on PXT3003 dose 1 (5 mL). Patients randomised to PXT3003 dose 2 (5 mL) in the primary study (CLN-PXT3003-02) continued in the extension study on PXT3003 dose 2 or PXT3003 twice dose 1 (2x5 mL).

Period 2: All patients continue on twice dose 1 (2X5mL).

Detailed Description

PXT3003 is a rational design, fixed combination of low-dose (RS) baclofen, naltrexone hydrochloride and D-sorbitol. The use of PXT3003 in a multicenter, randomised, placebo controlled phase II study (CLN-PXT3003-01) was well-tolerated and safe in patients with CMT1A for the three dose-levels investigated (Attarian et al., 2014). The intermediate and high dose of PXT3003 demonstrated an improvement of disability in this patient population.

Subsequently a multicenter, randomised, placebo controlled phase III study (CLN-PXT3003-02) to assess the efficacy and safety of PXT3003 in the treatment of patients with CMT1A was initiated in December 2015. In March 2017 the first patients completed the 15-month treatment with PXT3003 and rolled over into the extension study CLN-PXT3003-03.

During Period 1 (9 months), patients that were randomised to PXT3003 dose 1 or placebo in the primary study (CLN-PXT3003-02) continued in the extension study on PXT3003 dose 1 (5 mL). Patients randomised to PXT3003 dose 2 (5 mL) in the primary study (CLN-PXT3003-02) continued in the extension study on on PXT3003 dose 2 or PXT3003 twice dose 1 (2x5 mL). During Period 2, all patients continue on twice dose 1 (2X5mL).

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
187
Inclusion Criteria

Not provided

Exclusion Criteria
  • Any clinically significant change in health status that, in the opinion of the Investigator, would prevent the subject from participating in this study or successfully completing this study
  • Any unauthorized concomitant treatments, as study CLN-PXT3003-02 (e.g. including but not limited to baclofen, naltrexone,sorbitol (pharmaceutical form), opioids, levothyroxin, and potentially neurotoxic drugs such as amiodarone, chloroquine, cancer drugs susceptible to induce peripheral neuropathy)

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PXT3003 dose 2PXT3003Period 1, PXT3003: Liquid oral solution (1.2 mg/mL baclofen, 0.14 mg/mL naltrexone HCl and 420 mg/mL D-sorbitol), 5 mL bid (taken morning and evening with food) for 9 consecutive months Period 2, PXT3003: Liquid oral solution (0.6 mg/mL baclofen, 0.07 mg/mL naltrexone HCl and 210 mg/mL D-sorbitol), 10 mL bid (taken morning and evening with food)
PXT3003 dose 1PXT3003Period 1, PXT3003 : Liquid oral solution (0.6 mg/mL baclofen, 0.07 mg/mL naltrexone HCl and 210 mg/mL D-sorbitol), 5 mL bid (taken morning and evening with food) for 9 consecutive months
Primary Outcome Measures
NameTimeMethod
Incidence of treatment-emergent adverse events (TEAEs) related to PXT3003 during the follow-up in patients with CMT1A9 or 24 months

Incidence of treatment-emergent adverse events (TEAEs) related to PXT3003 during the follow-up in patients with CMT1A

Secondary Outcome Measures
NameTimeMethod
Incidence of adverse events leading to withdrawal of study drug9 or 24 months

Incidence of adverse events leading to withdrawal of study drug

Charcot-Marie-Tooth Neuropathy Score - version 2 (CMTNS-V2), and its sub-items9 or 24 months

Charcot-Marie-Tooth Neuropathy Score - version 2 (CMTNS-V2), and its sub-items

Time to walk 10 meters9 or 24 months

Time to walk 10 meters

Incidence of all TEAEs and their evaluation of type/nature, severity/intensity, seriousness, duration, relationship to study drug, and outcome9 or 24 months

Incidence of all TEAEs and their evaluation of type/nature, severity/intensity, seriousness, duration, relationship to study drug, and outcome

Overall Neuropathy Limitation Scale (ONLS) score, and its arm and leg sub-items9 or 24 months

Overall Neuropathy Limitation Scale (ONLS) score, and its arm and leg sub-items

Nine-hole Peg Test (9-HPT)9 or 24 months

Nine-hole Peg Test (9-HPT)

Compound Muscle Action Potential (CMAP) on ulnar nerve9 or 24 months

Compound Muscle Action Potential (CMAP) on ulnar nerve

Nerve conduction velocity (NCV)9 or 24 months

Nerve conduction velocity (NCV)

Visual analog scale on self-assessment of individualized main impairment in daily activities (defined at baseline with the patient)9 or 24 months

Visual analog scale on self-assessment of individualized main impairment in daily activities (defined at baseline with the patient)

Quantified Muscular Testing (QMT) by hand grip and foot dorsiflexion dynamometry (mean of both sides)9 or 24 months

Quantified Muscular Testing (QMT) by hand grip and foot dorsiflexion dynamometry (mean of both sides)

Sensory Nerve Action Potential (SNAP) on radial nerve9 or 24 months

Sensory Nerve Action Potential (SNAP) on radial nerve

Quality of Life (EQ-5D)9 or 24 months

Quality of Life (EQ-5D)

Trial Locations

Locations (23)

Departement of Neurology, UZ Leuven

🇧🇪

Leuven, Belgium

Servicio de Neurologia, Hospital Universitario i Politécnic La Fe

🇪🇸

Valencia, Spain

Department of Neurology, Salford Royal NHS Foundation Trust

🇬🇧

Salford, Manchester, United Kingdom

Department of Neurology, McKnight Brain Institute

🇺🇸

Gainesville, Florida, United States

Department of Neurology, Cedars-Sinai Medical Center

🇺🇸

Los Angeles, California, United States

Brigham and Women's Hospital

🇺🇸

Boston, Massachusetts, United States

University of Michigan Health System

🇺🇸

Ann Arbor, Michigan, United States

Department of Neurology, University of Minnesota

🇺🇸

Minneapolis, Minnesota, United States

Department of Neurology and Psichiatry, Saint Louis University

🇺🇸

Saint Louis, Missouri, United States

Peripheral Neuropathy Center, Neurological Institue Building, Columbia University Medical Center

🇺🇸

New York, New York, United States

Saint Luke's Rehabilitation Institute

🇺🇸

Spokane, Washington, United States

University Hospital of Quebec

🇨🇦

Quebec, Canada

Cntre de Reference des Maladies Neuromusculaires, Hopital Swynghedauwl, CHU Lille

🇫🇷

Lille, France

Service de Neurologie et du Sommeil, CHU Lyon Sud

🇫🇷

Lyon, France

Centre de Reference des Maladie Neuromusculaires, CHU la Timone

🇫🇷

Marseille, France

Centre de Reference des Maladie Neuromusculaires, Hotel Dieu, CHU de Nantes

🇫🇷

Nantes, France

Service de Neurologie, Hopital Kremlin Bicetre

🇫🇷

Paris, France

Departement of Neurology, Academic Medical Center

🇳🇱

Amsterdam, Netherlands

Department of neurology, Hospital Univesitario de Bellvitge

🇪🇸

Barcelona, Spain

Servicio de Neurologia, Hospital Universitario La Paz

🇪🇸

Madrid, Spain

Centro de Diagnostico y Tratamiento, Hospital Universitario Virgen del Rocio

🇪🇸

Sevilla, Spain

Centre de Reference des Neuropathies Peripheriques Rare, Hopital Dupuytren, CHU Limoges

🇫🇷

Limoges, France

University of Kansas Medical Center

🇺🇸

Kansas City, Kansas, United States

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