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Phase 2 Study of DS-8500a in Patients With Type 2 Diabetes

Phase 2
Completed
Conditions
Type 2 Diabetes Mellitus
Interventions
Drug: 10mg DS-8500a tablet
Drug: 75mg DS-8500a tablet
Drug: placebo
Registration Number
NCT02222350
Lead Sponsor
Daiichi Sankyo Co., Ltd.
Brief Summary

The objective of this study is to evaluate the efficacy and safety of DS-8500a compared with placebo in Japanese patients with Type 2 Diabetes Mellitus.

Detailed Description

The objective of this study is to evaluate the efficacy and safety of DS-8500a 10 mg and 75 mg administered orally, once daily, for 28 days, compared with placebo, in Japanese patients with Type 2 Diabetes Mellitus in a double-blind, placebo-controlled parallel-group design. The primary endpoint is the change in 24-hour weighted mean glucose at day 28 from baseline. The safety, pharmacokinetics, and pharmacodynamics of DS-8500a will be evaluated as well.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
100
Inclusion Criteria
  • Patients aged ≥ 20 years at the time of informed consent
  • Japanese patients with type 2 diabetes
  • Patients who have HbA1c ≥ 7.0% and < 10.0% if untreated with antidiabetic agent.
  • Patients who have HbA1c ≥ 6.5% and < 9.5% if treated with antidiabetic agent.
Exclusion Criteria
  • Patients aged ≥ 70 years at the time of informed consent
  • Patients with a history of type 1 diabetes or diabetic ketoacidosis
  • Patients receiving or requiring treatment with insulin
  • Patients with a body mass index (BMI) of < 18.5 kg/m2 or ≥ 35.0 kg/m2
  • Patients with an estimated glomerular filtration rate (eGFR), < 45 mL/min per 1.73 m2
  • Patients with fasting plasma glucose ≥ 240 mg/dL

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
DS-8500a 10mg once daily10mg DS-8500a tablet10mg DS-8500a tablet given orally once daily
DS8500a 75 mg once daily75mg DS-8500a tablet75mg DS-8500a tablet given orally once daily
placebo to match DS-8500a tabletplaceboplacebo matching DS-8500a tablet
Primary Outcome Measures
NameTimeMethod
change in 24-hour weighted mean blood glucoseDay -1 (baseline) to Day 28
Secondary Outcome Measures
NameTimeMethod
change in blood HbA1c levelDay -1 (baseline) to Days 14 and 28

Change in the parameter at Day 14 or 28 from Day -1

change in blood fasting plasma glucose levelDay -1 (baseline) to Days 7, 14, 21, 28
change in blood insulin levelDay -1 (baseline) to Days 14 and 28

Change in the parameter at Day 14 or 28 from Day -1

change in blood active GLP-1 levelDay -1 (baseline) to Days 14 and 28

Change in the parameter at Day 14 or 28 from Day -1

change in 24 hour weighted mean blood glucoseDay -1 (baseline) to Day 14
change in blood plasma glucose levelDay -1 (baseline) to Days 14 and 28

Change in the parameter at Day 14 or 28 from Day -1

change in blood C-peptide levelDay -1 (baseline) to Days 14 and 28

Change in the parameter at Day 14 or 28 from Day -1

change in blood glycoalbumin levelDay -1 (baseline) to Days 14 and 28

Change in the parameter at Day 14 or 28 from Day -1

change in blood PYY levelDay -1 (baseline) to Days 14 and 28

Change in the parameter at Day 14 or 28 from Day -1

Number of subjects experiencing adverse events as a measure of safetyDay -1 (baseline) to Day 28

Number of subjects experiencing adverse events

change in postprandial plasma glucose levelDay -1 (baseline) to Days 14 and 28

Change in postprandial plasma glucose level (2 hours after a meal) at Day 14 or 28 from Day -1

pharmacokinetic profile of DS-8500aDay -1 (baseline) to Day 28

Pharmacokinetic profile of DS-8500a in Japanese subjects with type 2 diabetes mellitus. i.e. Tmax, Cmax, AUC, t1/2

Trial Locations

Locations (1)

Heishinkai Medical Group Incorporated OCROM Clinic

🇯🇵

Kasuga, Osaka, Japan

Heishinkai Medical Group Incorporated OCROM Clinic
🇯🇵Kasuga, Osaka, Japan
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