MedPath

Buspirone for Weak or Absent Esophageal Peristalsis

Phase 4
Recruiting
Conditions
Dysphagia, Esophageal
Interventions
Registration Number
NCT05629325
Lead Sponsor
Universitaire Ziekenhuizen KU Leuven
Brief Summary

This is a randomized, double-blind, placebo-controlled, cross-over clinical trial of buspirone in patients with complaints of dysphagia due to poor esophageal motility. The goal of this clinical trial is to study the effect of buspirone on esophageal motility by performing high resolution impedance manometry (HRiM).

Detailed Description

Esophageal motility disorders can be characterized by poor esophageal motility with impaired clearance of the esophagus. Examples are Ineffective Esophageal Motility (IEM, \>70% of the swallows are ineffective or ≥50% are failed) and Absent Contractility (100% failed peristalsis). Both might be the underlying cause for dysphagia.

Several studies have shown that poor esophageal motility can be manipulated by pharmacological means. Buspirone, a 5-HT1A agonist, is able to significantly increase distal esophageal wave amplitude and duration in healthy volunteers, suggesting it may be effective in IEM. At the moment, findings in patients with IEM are not consistent and depend on the dose and treatment duration.

This cross-over trial will examine the use of buspirone in patients with dysphagia, with the intent of using a higher dose. We will use impedance/manometry and pressure flow analysis to liquid, viscous and solid boluses to evaluate the symptomatic and manometric effect of buspirone.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
25
Inclusion Criteria

Patients can participate in this study if:

  1. A minimum of 18 years old;

  2. Ineffective Esophageal Motility (IEM) or absent contractility, as determined on HRM in the last three months before inclusion in the study, using the Chicago classification v4.0 (1).

    IEM is defined as >70% ineffective or ≥50% failed swallows with a normal integrated relaxation pressure (IRP4). IEM includes a weak contraction (DCI ≥ 100 mmHg·s·cm and <450 mmHg·s·cm), failed peristalsis (DCI < 100 mmHg·s·cm), or fragmented peristalsis (a large break (>5 cm length) in the 20-mmHg isobaric contour with DCI > 450 mmHg·s·cm).

    Absent contractility is defined as 100% failed swallows (DCI < 100 mmHg·s·cm), with a normal IRP4.

  3. Have completed a gastro-duodenoscopy, within 12 months, showing no anatomical abnormality of the stomach or esophagus, which can explain the patients' symptoms.

  4. History of dysphagia for at least 2 months, at least twice per week in the last month.

  5. Sexually active women of childbearing potential participating in the study must be using an appropriate form of contraception. Medically acceptable forms of contraception include oral contraceptives, injectable or implantable methods, intrauterine devices, or properly used barrier contraception. If the female patient has not been on oral, injectable, implantable or intrauterine contraception, a urinary pregnancy test will be performed prior to administration of Buspirone/Placebo.

  6. Subjects must be capable of understanding and be willing to provide signed and dated written voluntary informed consent before any protocol-specific screening procedures are performed.

Exclusion Criteria

Patients cannot participate in this study if:

  1. Endoscopic signs of severe erosive esophagitis (grade C or D, Los Angeles classification) on endoscopy performed off PPI treatment in the 12 months prior to screening, or ≥ grade B when endoscopy is performed during PPI treatment.
  2. Systemic diseases, known to affect esophageal motility (i.e. systemic sclerosis)
  3. Surgery in the thorax or in the upper part of the abdomen (appendectomy and cholecystectomy are allowed).
  4. Hiatal hernia ≥3 cm
  5. QT c>450 ms.
  6. Use of medication that effect cholinergic function such as anticholinergics, tricyclic antidepressants.
  7. Concomitant promotility agents such as prucalopride or domperidone.
  8. Concomitant use of more than one benzodiazepine.
  9. Significant neurological, respiratory, hepatic, renal, hematological, cardiovascular, metabolic or gastrointestinal cerebrovascular disease as judged by the investigator.
  10. Major psychiatric disorder.
  11. Pregnancy or breastfeeding.
  12. History of poor compliance.
  13. History of/or current psychiatric illness that would interfere with ability to comply with protocol requirements or give informed consent.
  14. History of alcohol or drug abuse that would interfere with ability to comply with protocol requirements.

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Buspirone => Washout => PlaceboBuspirone Hydrochloride 10 MGPatients will take Buspirone hydrochloride 10mg oral once a day (in the evening) for 3 days, twice a day (morning and evening) for 4 days, three times a day for 2 weeks and 20mg oral three times a day for one week. Esophageal motility will be assessed with high resolution impedance manometry (HRiM) after 4 weeks of treatment. Patients will also report their perceived symptoms of dysphagia during the HRiM. A washout period of two weeks will take place. Afterwards, the second treatment period starts. Patients will take Placebo oral once a day (in the evening) for 3 days, twice a day (morning and evening) for 4 days, three times a day for 2 weeks and 20mg oral three times a day for one week. Esophageal motility will also be assessed with high resolution impedance manometry (HRiM) after 4 weeks of treatment. Patients will again report their perceived symptoms of dysphagia during the HRiM.
Placebo => Washout => BuspironeBuspirone Hydrochloride 10 MGPatients will take Placebo oral once a day (in the evening) for 3 days, twice a day (morning and evening) for 4 days, three times a day for 2 weeks and 20mg oral three times a day for one week. Esophageal motility will be assessed with high resolution impedance manometry (HRiM) after 4 weeks of treatment. Patients will also report their perceived symptoms of dysphagia during the HRiM. A washout period of two weeks will take place. Afterwards, the second treatment period starts. Patients will take Buspirone hydrochloride oral once a day (in the evening) for 3 days, twice a day (morning and evening) for 4 days, three times a day for 2 weeks and 20mg oral three times a day for one week. Esophageal motility will also be assessed with high resolution impedance manometry (HRiM) after 4 weeks of treatment. Patients will again report their perceived symptoms of dysphagia during the HRiM.
Buspirone => Washout => PlaceboPlaceboPatients will take Buspirone hydrochloride 10mg oral once a day (in the evening) for 3 days, twice a day (morning and evening) for 4 days, three times a day for 2 weeks and 20mg oral three times a day for one week. Esophageal motility will be assessed with high resolution impedance manometry (HRiM) after 4 weeks of treatment. Patients will also report their perceived symptoms of dysphagia during the HRiM. A washout period of two weeks will take place. Afterwards, the second treatment period starts. Patients will take Placebo oral once a day (in the evening) for 3 days, twice a day (morning and evening) for 4 days, three times a day for 2 weeks and 20mg oral three times a day for one week. Esophageal motility will also be assessed with high resolution impedance manometry (HRiM) after 4 weeks of treatment. Patients will again report their perceived symptoms of dysphagia during the HRiM.
Placebo => Washout => BuspironePlaceboPatients will take Placebo oral once a day (in the evening) for 3 days, twice a day (morning and evening) for 4 days, three times a day for 2 weeks and 20mg oral three times a day for one week. Esophageal motility will be assessed with high resolution impedance manometry (HRiM) after 4 weeks of treatment. Patients will also report their perceived symptoms of dysphagia during the HRiM. A washout period of two weeks will take place. Afterwards, the second treatment period starts. Patients will take Buspirone hydrochloride oral once a day (in the evening) for 3 days, twice a day (morning and evening) for 4 days, three times a day for 2 weeks and 20mg oral three times a day for one week. Esophageal motility will also be assessed with high resolution impedance manometry (HRiM) after 4 weeks of treatment. Patients will again report their perceived symptoms of dysphagia during the HRiM.
Primary Outcome Measures
NameTimeMethod
HRiM Manometric Features: DCI 5ml supineDuring manometric assessment after 4 weeks of treatment

Changes in distal contractile integral (DCI, in mmHg\*s\*cm) between buspirone and placebo. DCI is established on HRiM. As primary endpoint, we will focus on the values for DCI for the liquid bolus, 5 ml in supine position.

Secondary Outcome Measures
NameTimeMethod
HRiM Manometric Features: PFIDuring manometric assessment after 4 weeks of treatment

Pressure Flow Index (PFI, -)

Mayo Dysphagia QuestionnaireAt baseline and after 4 weeks of treatment

Symptom questionnaire

HRiM Manometric Features: DCIDuring manometric assessment after 4 weeks of treatment

Distal Esophageal Contractile Integral (DCI, mmHg.s.cm)

HRiM Manometric Features: Largest Break SizeDuring manometric assessment after 4 weeks of treatment

Largest Break Size (cm)

HRiM Manometric Features: DPEDuring manometric assessment after 4 weeks of treatment

Distension Pressure Emptying Phase (DPE, mmHg)

HRiM Manometric Features: RPDuring manometric assessment after 4 weeks of treatment

Distal Ramp Pressure (RP, mmHg/s)

HRiM Manometric Features: BPTDuring manometric assessment after 4 weeks of treatment

Bolus Presence Time (BPT, s)

HRiM Manometric Features: BFTDuring manometric assessment after 4 weeks of treatment

Bolus Flow Time (BFT, s)

Overall Treatment Evaluation (OTE)At baseline and after 4 weeks of treatment

Symptoms questionnaire

Overall Symptom Severity (OSS)At baseline and after 4 weeks of treatment

Symptom questionnaire

HRiM Manometric Features: DLDuring manometric assessment after 4 weeks of treatment

Distal Latency (DL, s)

HRiM Manometric Features: LES-CDDuring manometric assessment after 4 weeks of treatment

Lower Esophageal Sphincter - Crural Diaphragm (LES-CD, mm)

HRiM Manometric Features: IRP4sDuring manometric assessment after 4 weeks of treatment

Integrated Relaxation Pressure EGJ 4sec (IRP4s, mmHg)

HRiM Manometric Features: EGJ Rest.PDuring manometric assessment after 4 weeks of treatment

EGJ Resting Pressure (EGJ Rest.P, mmHg)

Bolus passage scoreDuring manometric assessment after 4 weeks of treatment

Patients will evaluate the perception of each swallow during the manometric assessment via the following Likert score: 1-Normal, 2-Slow passage of bolus, 3-Stepwise passage, 4-Partial Blockage, 5-Complete Blockage.

HRiM Manometric Features: PCIDuring manometric assessment after 4 weeks of treatment

Pharyngeal Esophageal Contractile Integral (PCI es., mm.Hg.s.cm)

HRiM Manometric Features: IRDuring manometric assessment after 4 weeks of treatment

Impedance Ratio (IR, -)

HRiM Manometric Features: DPADuring manometric assessment after 4 weeks of treatment

Distension Pressure Accommodation Phase (DPA, mmHg)

HRiM Manometric Features: CSIDuring manometric assessment after 4 weeks of treatment

Contractile Segment Impedance (CSI, Ohm)

HRiM Manometric Features: EGJCIDuring manometric assessment after 4 weeks of treatment

EGJ Contractile Integral (EGJCI, mmHg.cm)

Trial Locations

Locations (1)

University Hospitals Leuven

🇧🇪

Leuven, Vlaams-Brabant, Belgium

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